DK141780B - Analogifremgangsmåde til fremstilling af 1,4-benzodiazepinderivater. - Google Patents

Analogifremgangsmåde til fremstilling af 1,4-benzodiazepinderivater. Download PDF

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Publication number
DK141780B
DK141780B DK576868AA DK576868A DK141780B DK 141780 B DK141780 B DK 141780B DK 576868A A DK576868A A DK 576868AA DK 576868 A DK576868 A DK 576868A DK 141780 B DK141780 B DK 141780B
Authority
DK
Denmark
Prior art keywords
tetrahydro
benzodiazepin
reaction
chloro
phenyl
Prior art date
Application number
DK576868AA
Other languages
Danish (da)
English (en)
Other versions
DK141780C (no
Inventor
Tetsuo Miyadera
Toshiharu Kamioka
Hiromu Takagi
Mitsunobu Fukunaga
Yoichi Kawano
Ryuji Tachikawa
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP43076013A external-priority patent/JPS4830076B1/ja
Application filed by Sankyo Co filed Critical Sankyo Co
Priority to DK573272A priority Critical patent/DK141699B/da
Publication of DK141780B publication Critical patent/DK141780B/da
Application granted granted Critical
Publication of DK141780C publication Critical patent/DK141780C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/02—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK576868AA 1967-11-27 1968-11-26 Analogifremgangsmåde til fremstilling af 1,4-benzodiazepinderivater. DK141780B (da)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DK573272A DK141699B (da) 1967-11-27 1972-11-17 Aminoacetylaminobenzophenon-forbindelser til anvendelse som mellemprodukt ved fremstilling af terapeutisk aktive 5-phenyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-2-on-forbindelser.

Applications Claiming Priority (22)

Application Number Priority Date Filing Date Title
JP7600567 1967-11-27
JP7600767 1967-11-27
JP7600867 1967-11-27
JP7600567 1967-11-27
JP7600767 1967-11-27
JP7600867 1967-11-27
JP4572268 1968-07-01
JP4572268 1968-07-01
JP6270068 1968-08-31
JP6269968 1968-08-31
JP6270068 1968-08-31
JP6269968 1968-08-31
JP7601368 1968-10-18
JP7601268 1968-10-18
JP7601268 1968-10-18
JP43076013A JPS4830076B1 (no) 1968-10-18 1968-10-18
JP7749868 1968-10-24
JP7749968 1968-10-24
JP7749968 1968-10-24
JP7749868 1968-10-24
JP7876868 1968-10-29
JP7876868 1968-10-29

Publications (2)

Publication Number Publication Date
DK141780B true DK141780B (da) 1980-06-16
DK141780C DK141780C (no) 1980-12-01

Family

ID=27581992

Family Applications (1)

Application Number Title Priority Date Filing Date
DK576868AA DK141780B (da) 1967-11-27 1968-11-26 Analogifremgangsmåde til fremstilling af 1,4-benzodiazepinderivater.

Country Status (14)

Country Link
US (2) US3914215A (no)
AT (1) AT299203B (no)
CA (1) CA1038381A (no)
CH (1) CH518302A (no)
DE (1) DE1817923C3 (no)
DK (1) DK141780B (no)
FI (1) FI49048C (no)
GB (1) GB1254736A (no)
IE (1) IE32894B1 (no)
IL (2) IL31094A (no)
NL (1) NL170957C (no)
NO (1) NO127055B (no)
SE (1) SE346791B (no)
YU (3) YU36709B (no)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK153152B (da) * 1968-10-24 1988-06-20 Sankyo Co Fremgangsmaade til fremstilling af benzodiazepinforbindelser

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH574443A5 (no) * 1970-04-06 1976-04-15 Hoffmann La Roche
LU65340A1 (no) * 1972-05-12 1973-11-22
US3928415A (en) * 1973-05-08 1975-12-23 Cassella Farbwerke Mainkur Ag Benzophenone derivatives and process for their production II
JPS584035B2 (ja) * 1974-05-07 1983-01-24 武田薬品工業株式会社 イコウカンカゴウブツノ セイゾウホウ
US4007219A (en) * 1974-08-20 1977-02-08 Hoffmann-La Roche Inc. Benzophenone glycinamide derivatives
FR2403330A1 (fr) * 1977-06-16 1979-04-13 Fabre Sa Pierre Nouveaux derives de benzoyl-2-chloro-4-glycinanilides substitues, leur procede de preparation et leur application en tant que medicaments
FR2436776A1 (fr) * 1978-09-25 1980-04-18 Fabre Sa Pierre Nouveaux derives d'ortho chloro benzoyl-2 chloro-4 glycylanilide, leur preparation et leur application en tant que medicaments
FR2459793A1 (fr) * 1979-06-25 1981-01-16 Fabre Sa Pierre Nouveaux derives de benzoyl-2 nitro-4 anilides, leur preparation et leur application en tant que medicaments
US4289770A (en) * 1980-06-13 1981-09-15 Pierre Fabre S.A. 2-Benzoyl-4-nitroanilides and their use as medicaments
FR2525214B1 (fr) * 1982-04-16 1986-02-07 Fabre Sa Pierre Nouveaux derives d'halogeno benzoyl-2 nitro-4 glycylanilides, leur procede de preparation et leur application en therapeutique

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3371085A (en) * 1959-12-10 1968-02-27 Hoffmann La Roche 5-aryl-3h-1,4-benzodiazepin-2(1h)-ones

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK153152B (da) * 1968-10-24 1988-06-20 Sankyo Co Fremgangsmaade til fremstilling af benzodiazepinforbindelser

Also Published As

Publication number Publication date
US3772371A (en) 1973-11-13
CH518302A (de) 1972-01-31
NL6816789A (no) 1969-05-29
FI49048B (no) 1974-12-02
SE346791B (no) 1972-07-17
CA1038381A (en) 1978-09-12
YU41664B (en) 1987-12-31
YU229879A (en) 1983-12-31
YU36709B (en) 1984-08-31
US3914215A (en) 1975-10-21
NL170957B (nl) 1982-08-16
DE1817923A1 (de) 1974-06-06
IL31094A0 (en) 1969-01-29
IE32894B1 (en) 1974-01-09
NO127055B (no) 1973-04-30
DK141780C (no) 1980-12-01
YU279468A (en) 1982-06-18
IE32894L (en) 1969-05-27
IL31094A (en) 1972-09-28
DE1817923B2 (de) 1977-11-24
YU229779A (en) 1983-01-21
IL39770A (en) 1972-10-29
FI49048C (fi) 1975-03-10
NL170957C (nl) 1983-01-17
YU41413B (en) 1987-04-30
GB1254736A (en) 1971-11-24
DE1817923C3 (de) 1978-08-03
AT299203B (de) 1972-06-12

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