DK141622B - Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive 1-(3,5-dihydroxyfenyl)-2-aminoætanolderivater eller syreadditionssalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive 1-(3,5-dihydroxyfenyl)-2-aminoætanolderivater eller syreadditionssalte deraf. Download PDF

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Publication number
DK141622B
DK141622B DK439776AA DK439776A DK141622B DK 141622 B DK141622 B DK 141622B DK 439776A A DK439776A A DK 439776AA DK 439776 A DK439776 A DK 439776A DK 141622 B DK141622 B DK 141622B
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DK
Denmark
Prior art keywords
compound
group
general formula
carbon atoms
dihydroxyphenyl
Prior art date
Application number
DK439776AA
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Danish (da)
English (en)
Other versions
DK439776A (de
Inventor
Kjell Ingvar Leopold Wetterlin
Leif Aake Svensson
Lars Magnus Soerenby
Original Assignee
Draco Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Draco Ab filed Critical Draco Ab
Publication of DK439776A publication Critical patent/DK439776A/da
Publication of DK141622B publication Critical patent/DK141622B/da

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/04Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reaction of ammonia or amines with olefin oxides or halohydrins
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/70Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
    • C07C45/71Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • C07D265/321,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings with oxygen atoms directly attached to ring carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Immunology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
DK439776AA 1975-10-01 1976-09-30 Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive 1-(3,5-dihydroxyfenyl)-2-aminoætanolderivater eller syreadditionssalte deraf. DK141622B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE7510988A SE7510988L (sv) 1975-10-01 1975-10-01 Nya farmaceutiskt aktiva foreningar
SE7510988 1975-10-01

Publications (2)

Publication Number Publication Date
DK439776A DK439776A (de) 1977-04-02
DK141622B true DK141622B (da) 1980-05-12

Family

ID=20325688

Family Applications (1)

Application Number Title Priority Date Filing Date
DK439776AA DK141622B (da) 1975-10-01 1976-09-30 Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive 1-(3,5-dihydroxyfenyl)-2-aminoætanolderivater eller syreadditionssalte deraf.

Country Status (19)

Country Link
JP (1) JPS5242840A (de)
AT (1) AT347427B (de)
AU (1) AU503212B2 (de)
BE (1) BE846837A (de)
CS (2) CS199643B2 (de)
DD (1) DD126278A5 (de)
DE (1) DE2640972A1 (de)
DK (1) DK141622B (de)
ES (1) ES451979A1 (de)
FI (1) FI762660A (de)
FR (1) FR2326183A1 (de)
GB (1) GB1542317A (de)
LU (1) LU75916A1 (de)
NL (1) NL7610845A (de)
NO (1) NO763345L (de)
NZ (1) NZ182165A (de)
SE (1) SE7510988L (de)
SU (2) SU638252A3 (de)
ZA (1) ZA765331B (de)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4419364A (en) 1980-07-09 1983-12-06 Aktiebolaget Draco Bronchospasmolytic carbamate derivatives

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0103830A3 (de) * 1982-09-22 1985-07-31 Bayer Ag Wachstumsfördernde Phenylethylamin-Derivate
EP1636191A2 (de) 2003-06-17 2006-03-22 Arena Pharmaceuticals, Inc. Für die behandlung von mit dem 5ht2c rezeptor assoziierten krankheiten geeignete benzazepinderivative
CA2646044A1 (en) 2006-04-03 2007-10-25 Arena Pharmaceuticals, Inc. Processes for the preparation of 8-chloro-1-methyl-2,3,4,5-tetrahydro-1h-3-benzazepine and intermediates related thereto
CA2670285A1 (en) 2006-12-05 2008-06-12 Arena Pharmaceuticals, Inc. Processes for preparing (r)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1h-3-benzazepine and intermediates thereof
WO2009111004A1 (en) 2008-03-04 2009-09-11 Arena Pharmaceuticals, Inc. Processes for the preparation of intermediates related to the 5-ht2c agonist (r)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1h-3-benzazepine
CN102648170A (zh) 2009-06-18 2012-08-22 艾尼纳制药公司 制备5-ht2c受体激动剂的方法
US9045431B2 (en) 2010-06-02 2015-06-02 Arena Pharmaceuticals, Inc. Processes for the preparation of 5-HT2C receptor agonists
MX2013002418A (es) 2010-09-01 2013-08-01 Arena Pharm Inc Administracion de lorcaserina a individuos con daño renal.
SG188361A1 (en) 2010-09-01 2013-04-30 Arena Pharm Inc Non-hygroscopic salts of 5-ht2c agonists
CN103189053A (zh) 2010-09-01 2013-07-03 艾尼纳制药公司 用于体重控制的5-ht2c激动剂的调节释放剂型
JP2013539470A (ja) 2010-09-01 2013-10-24 アリーナ ファーマシューティカルズ, インコーポレイテッド ロルカセリンと光学活性な酸との塩
BR112015007779A2 (pt) 2012-10-09 2017-07-04 Arena Pharm Inc célula de fluxo de permeabilidade e sistema de condutância hidráulica

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4419364A (en) 1980-07-09 1983-12-06 Aktiebolaget Draco Bronchospasmolytic carbamate derivatives

Also Published As

Publication number Publication date
CS199644B2 (en) 1980-07-31
ES451979A1 (es) 1978-01-01
FI762660A (de) 1977-04-02
LU75916A1 (de) 1978-05-16
SU674669A3 (ru) 1979-07-15
NO763345L (de) 1977-04-04
NL7610845A (nl) 1977-04-05
JPS5242840A (en) 1977-04-04
SU638252A3 (ru) 1978-12-15
GB1542317A (en) 1979-03-14
SE7510988L (sv) 1977-04-02
AU503212B2 (en) 1979-08-30
ATA682376A (de) 1978-05-15
BE846837A (fr) 1977-04-01
ZA765331B (en) 1977-08-31
DE2640972A1 (de) 1977-04-14
AT347427B (de) 1978-12-27
FR2326183A1 (fr) 1977-04-29
CS199643B2 (en) 1980-07-31
DK439776A (de) 1977-04-02
DD126278A5 (de) 1977-07-06
NZ182165A (en) 1978-07-10
AU1812276A (en) 1978-04-06

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