DK1414439T3 - Nye pyrroler med hypolipidæmiske og hypocholesterolæmiske aktiviteter, fremgangsmåde til deres fremstilling og farmaceutiske sammensætninger indeholdende dem og deres anvendelse indenfor medicin - Google Patents

Nye pyrroler med hypolipidæmiske og hypocholesterolæmiske aktiviteter, fremgangsmåde til deres fremstilling og farmaceutiske sammensætninger indeholdende dem og deres anvendelse indenfor medicin

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Publication number
DK1414439T3
DK1414439T3 DK02751609.5T DK02751609T DK1414439T3 DK 1414439 T3 DK1414439 T3 DK 1414439T3 DK 02751609 T DK02751609 T DK 02751609T DK 1414439 T3 DK1414439 T3 DK 1414439T3
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Prior art keywords
compositions containing
medicine
pharmaceutically acceptable
pharmaceutical compositions
hypolipidemic
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DK02751609.5T
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English (en)
Inventor
Braj Bhushan Lohray
Vidya Bhushan Lohray
Vijay Kumar Barot
Saurin Khimshankar Raval
Preeti Saurin Raval
Sujay Basu
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Cadila Healthcare Ltd
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Publication of DK1414439T3 publication Critical patent/DK1414439T3/da

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/325—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
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    • C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07—ORGANIC CHEMISTRY
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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
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DK02751609.5T 2001-07-26 2002-07-25 Nye pyrroler med hypolipidæmiske og hypocholesterolæmiske aktiviteter, fremgangsmåde til deres fremstilling og farmaceutiske sammensætninger indeholdende dem og deres anvendelse indenfor medicin DK1414439T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN711MU2001 2001-07-26
PCT/IN2002/000155 WO2003009841A1 (en) 2001-07-26 2002-07-25 Novel pyrroles having hypolipidemic hypocholesteremic activities, process for their preparation and pharmaceutical compositions containing them and their use in medicine

Publications (1)

Publication Number Publication Date
DK1414439T3 true DK1414439T3 (da) 2011-07-18

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DK02751609.5T DK1414439T3 (da) 2001-07-26 2002-07-25 Nye pyrroler med hypolipidæmiske og hypocholesterolæmiske aktiviteter, fremgangsmåde til deres fremstilling og farmaceutiske sammensætninger indeholdende dem og deres anvendelse indenfor medicin

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US (6) US6987123B2 (da)
EP (1) EP1414439B1 (da)
JP (2) JP4313194B2 (da)
KR (2) KR20060094545A (da)
CN (1) CN100450477C (da)
AP (1) AP1808A (da)
AR (1) AR036347A1 (da)
AT (1) ATE507828T1 (da)
AU (1) AU2002355205B2 (da)
BR (1) BRPI0211665B8 (da)
CA (1) CA2454863C (da)
CO (1) CO5390079A1 (da)
CY (1) CY1111876T1 (da)
DE (1) DE60239939D1 (da)
DK (1) DK1414439T3 (da)
EA (1) EA006858B1 (da)
ES (1) ES2366279T3 (da)
HR (1) HRP20040138B1 (da)
IL (1) IL160042A (da)
MX (1) MXPA04000758A (da)
MY (1) MY140057A (da)
NO (1) NO326698B1 (da)
NZ (2) NZ550375A (da)
OA (1) OA12702A (da)
PL (1) PL224397B1 (da)
PT (1) PT1414439E (da)
RS (1) RS51837B (da)
SI (1) SI1414439T1 (da)
UA (1) UA76992C2 (da)
WO (1) WO2003009841A1 (da)
ZA (1) ZA200400563B (da)

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US20050288373A1 (en) * 2002-10-24 2005-12-29 Ron Eyal S Methods of treating various conditions by administration of sustained release L-arginine
JP2007516227A (ja) * 2003-05-16 2007-06-21 アンビット バイオサイエンシス コーポレーション ピロール化合物およびその使用
US20050182125A1 (en) * 2003-05-16 2005-08-18 Ambit Biosciences Corporation Pyrrole compounds and uses thereof
US20040248972A1 (en) * 2003-05-16 2004-12-09 Ambit Biosciences Corporation Compounds and uses thereof
US7767152B2 (en) * 2003-08-11 2010-08-03 Sakura Finetek U.S.A., Inc. Reagent container and slide reaction retaining tray, and method of operation
US9518899B2 (en) * 2003-08-11 2016-12-13 Sakura Finetek U.S.A., Inc. Automated reagent dispensing system and method of operation
US7744817B2 (en) * 2003-08-11 2010-06-29 Sakura Finetek U.S.A., Inc. Manifold assembly
PL1773768T3 (pl) * 2004-07-30 2019-03-29 Exelixis, Inc. Pochodne pirolu jako środki farmaceutyczne
US20110092566A1 (en) * 2004-11-19 2011-04-21 Srivastava Satish K Treatment of cancer with aldose reductase inhibitors
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