DK1273289T3 - Farmaceutiske sammensætninger indeholdende ascomycinderivater - Google Patents

Farmaceutiske sammensætninger indeholdende ascomycinderivater

Info

Publication number
DK1273289T3
DK1273289T3 DK02022257T DK02022257T DK1273289T3 DK 1273289 T3 DK1273289 T3 DK 1273289T3 DK 02022257 T DK02022257 T DK 02022257T DK 02022257 T DK02022257 T DK 02022257T DK 1273289 T3 DK1273289 T3 DK 1273289T3
Authority
DK
Denmark
Prior art keywords
pharmaceutical compositions
compositions containing
phosphatidylglycerol
sub
salt
Prior art date
Application number
DK02022257T
Other languages
English (en)
Inventor
Harry Tiemessen
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Application granted granted Critical
Publication of DK1273289T3 publication Critical patent/DK1273289T3/da

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12—Carboxylic acids; Salts or anhydrides thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
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    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
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Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Diabetes (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dispersion Chemistry (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurology (AREA)
  • Obesity (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Virology (AREA)
  • Endocrinology (AREA)
  • Transplantation (AREA)
  • Emergency Medicine (AREA)
DK02022257T 1996-01-19 1997-01-20 Farmaceutiske sammensætninger indeholdende ascomycinderivater DK1273289T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9601120.0A GB9601120D0 (en) 1996-01-19 1996-01-19 Organic compounds
EP97901563A EP0874621B1 (en) 1996-01-19 1997-01-20 [3'-DESOXY-3-OXO-MeBmT]1-[Val]2-CICLOSPORIN-CONTAINING EMULSION PHARMACEUTICAL COMPOSITIONS

Publications (1)

Publication Number Publication Date
DK1273289T3 true DK1273289T3 (da) 2006-03-20

Family

ID=10787276

Family Applications (4)

Application Number Title Priority Date Filing Date
DK05018663.4T DK1679064T3 (da) 1996-01-19 1997-01-20 Farmaceutiske sammensætninger indeholdende rapamycinderivater
DK97901563T DK0874621T3 (da) 1996-01-19 1997-01-20 Lægemiddelemulsion indeholdende [3'-desoxy-3-oxy-MeBmt]1-[Val]2-ciclosporin
DK02022257T DK1273289T3 (da) 1996-01-19 1997-01-20 Farmaceutiske sammensætninger indeholdende ascomycinderivater
DK02022256T DK1273288T3 (da) 1996-01-19 1997-01-20 Lægemiddelsammensætning indeholdende rapamycinderivater

Family Applications Before (2)

Application Number Title Priority Date Filing Date
DK05018663.4T DK1679064T3 (da) 1996-01-19 1997-01-20 Farmaceutiske sammensætninger indeholdende rapamycinderivater
DK97901563T DK0874621T3 (da) 1996-01-19 1997-01-20 Lægemiddelemulsion indeholdende [3'-desoxy-3-oxy-MeBmt]1-[Val]2-ciclosporin

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK02022256T DK1273288T3 (da) 1996-01-19 1997-01-20 Lægemiddelsammensætning indeholdende rapamycinderivater

Country Status (14)

Country Link
US (2) US6239102B1 (da)
EP (4) EP0874621B1 (da)
JP (2) JP4077386B2 (da)
KR (1) KR100485146B1 (da)
AT (4) ATE239449T1 (da)
AU (1) AU1543497A (da)
CA (2) CA2240339C (da)
DE (3) DE69721729T2 (da)
DK (4) DK1679064T3 (da)
ES (4) ES2253483T3 (da)
GB (1) GB9601120D0 (da)
HK (3) HK1054183B (da)
PT (2) PT874621E (da)
WO (1) WO1997025977A1 (da)

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ATE510532T1 (de) 2011-06-15
EP1273288B1 (en) 2005-09-21
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HK1054183B (zh) 2006-07-28
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EP1273288A1 (en) 2003-01-08
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JP4077386B2 (ja) 2008-04-16
PT1679064E (pt) 2011-07-25
DE69721729T2 (de) 2003-12-11
WO1997025977A1 (en) 1997-07-24
HK1053973B (zh) 2006-09-29
ES2247245T3 (es) 2006-03-01
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ATE239449T1 (de) 2003-05-15
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