DE69734742D1 - Arzneizusammensetzungen enthaltend Ascomycinderivate - Google Patents

Arzneizusammensetzungen enthaltend Ascomycinderivate

Info

Publication number
DE69734742D1
DE69734742D1 DE69734742T DE69734742T DE69734742D1 DE 69734742 D1 DE69734742 D1 DE 69734742D1 DE 69734742 T DE69734742 T DE 69734742T DE 69734742 T DE69734742 T DE 69734742T DE 69734742 D1 DE69734742 D1 DE 69734742D1
Authority
DE
Germany
Prior art keywords
pharmaceutical compositions
compositions containing
phosphatidylglycerol
sub
salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69734742T
Other languages
English (en)
Other versions
DE69734742T2 (de
Inventor
Harry Tiemessen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis AG filed Critical Novartis AG
Publication of DE69734742D1 publication Critical patent/DE69734742D1/de
Application granted granted Critical
Publication of DE69734742T2 publication Critical patent/DE69734742T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12—Carboxylic acids; Salts or anhydrides thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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    • A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
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    • A61P7/06—Antianaemics

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Diabetes (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Dispersion Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Biomedical Technology (AREA)
  • Virology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Neurosurgery (AREA)
  • Transplantation (AREA)
DE69734742T 1996-01-19 1997-01-20 Arzneizusammensetzungen enthaltend Ascomycinderivate Expired - Lifetime DE69734742T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9601120.0A GB9601120D0 (en) 1996-01-19 1996-01-19 Organic compounds
GB9601120 1996-01-19

Publications (2)

Publication Number Publication Date
DE69734742D1 true DE69734742D1 (de) 2005-12-29
DE69734742T2 DE69734742T2 (de) 2006-07-27

Family

ID=10787276

Family Applications (3)

Application Number Title Priority Date Filing Date
DE69721729T Expired - Lifetime DE69721729T2 (de) 1996-01-19 1997-01-20 [3'-DESOXY-3-OXO-MeBmt]1-[Val]2-CICLOSPORIN ENTHALTENDE ARZNEIMITTELEMULSION
DE69734253T Expired - Lifetime DE69734253T2 (de) 1996-01-19 1997-01-20 Arzneizusammensetzungen enthaltend Rapamycinderivate
DE69734742T Expired - Lifetime DE69734742T2 (de) 1996-01-19 1997-01-20 Arzneizusammensetzungen enthaltend Ascomycinderivate

Family Applications Before (2)

Application Number Title Priority Date Filing Date
DE69721729T Expired - Lifetime DE69721729T2 (de) 1996-01-19 1997-01-20 [3'-DESOXY-3-OXO-MeBmt]1-[Val]2-CICLOSPORIN ENTHALTENDE ARZNEIMITTELEMULSION
DE69734253T Expired - Lifetime DE69734253T2 (de) 1996-01-19 1997-01-20 Arzneizusammensetzungen enthaltend Rapamycinderivate

Country Status (14)

Country Link
US (2) US6239102B1 (de)
EP (4) EP0874621B1 (de)
JP (2) JP4077386B2 (de)
KR (1) KR100485146B1 (de)
AT (4) ATE304842T1 (de)
AU (1) AU1543497A (de)
CA (2) CA2678707A1 (de)
DE (3) DE69721729T2 (de)
DK (4) DK0874621T3 (de)
ES (4) ES2365734T3 (de)
GB (1) GB9601120D0 (de)
HK (3) HK1054183B (de)
PT (2) PT1679064E (de)
WO (1) WO1997025977A1 (de)

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ATE239449T1 (de) 2003-05-15
ES2247245T3 (es) 2006-03-01
EP1679064A2 (de) 2006-07-12
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JP4077386B2 (ja) 2008-04-16
PT874621E (pt) 2003-09-30
EP1679064A3 (de) 2009-10-07
EP1273288A1 (de) 2003-01-08
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DK1679064T3 (da) 2011-09-12
DE69721729T2 (de) 2003-12-11
GB9601120D0 (en) 1996-03-20
CA2240339A1 (en) 1997-07-24
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WO1997025977A1 (en) 1997-07-24
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ATE310504T1 (de) 2005-12-15
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