DK0996621T3 - Triazolo[4,5-d]pyrimidin-derivater som anti-trombotiske midler - Google Patents

Triazolo[4,5-d]pyrimidin-derivater som anti-trombotiske midler

Info

Publication number
DK0996621T3
DK0996621T3 DK98934107T DK98934107T DK0996621T3 DK 0996621 T3 DK0996621 T3 DK 0996621T3 DK 98934107 T DK98934107 T DK 98934107T DK 98934107 T DK98934107 T DK 98934107T DK 0996621 T3 DK0996621 T3 DK 0996621T3
Authority
DK
Denmark
Prior art keywords
triazolo
pyrimidine derivatives
thrombotic agents
thrombotic
agents
Prior art date
Application number
DK98934107T
Other languages
Danish (da)
English (en)
Inventor
Simon Guile
Anthony Ingall
Brian Springthorpe
Paul Willis
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26663042&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK0996621(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from SE9702775A external-priority patent/SE9702775D0/xx
Priority claimed from SE9702773A external-priority patent/SE9702773D0/xx
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Application granted granted Critical
Publication of DK0996621T3 publication Critical patent/DK0996621T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/04—Drugs for disorders of the respiratory system for throat disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Otolaryngology (AREA)
  • Urology & Nephrology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
DK98934107T 1997-07-22 1998-07-15 Triazolo[4,5-d]pyrimidin-derivater som anti-trombotiske midler DK0996621T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE9702775A SE9702775D0 (sv) 1997-07-22 1997-07-22 Novel compounds
SE9702773A SE9702773D0 (sv) 1997-07-22 1997-07-22 Novel compounds
PCT/SE1998/001393 WO1999005143A1 (en) 1997-07-22 1998-07-15 Novel compounds

Publications (1)

Publication Number Publication Date
DK0996621T3 true DK0996621T3 (da) 2004-02-02

Family

ID=26663042

Family Applications (1)

Application Number Title Priority Date Filing Date
DK98934107T DK0996621T3 (da) 1997-07-22 1998-07-15 Triazolo[4,5-d]pyrimidin-derivater som anti-trombotiske midler

Country Status (31)

Country Link
EP (1) EP0996621B1 (ja)
JP (1) JP4187406B2 (ja)
KR (2) KR20050084540A (ja)
CN (1) CN1154650C (ja)
AR (2) AR017014A1 (ja)
AT (1) ATE251161T1 (ja)
AU (1) AU745381B2 (ja)
BR (1) BR9810802B1 (ja)
CA (1) CA2296665C (ja)
CZ (1) CZ302629B6 (ja)
DE (1) DE69818668T2 (ja)
DK (1) DK0996621T3 (ja)
EE (1) EE04193B1 (ja)
EG (1) EG24412A (ja)
ES (1) ES2207846T3 (ja)
HK (1) HK1026421A1 (ja)
HU (1) HU230074B1 (ja)
IL (2) IL133959A0 (ja)
IS (1) IS2236B (ja)
MY (1) MY123196A (ja)
NO (1) NO315854B1 (ja)
NZ (1) NZ502381A (ja)
PL (1) PL200325B1 (ja)
PT (1) PT996621E (ja)
RU (1) RU2225407C2 (ja)
SA (1) SA98190487B1 (ja)
SK (1) SK284199B6 (ja)
TR (1) TR200000197T2 (ja)
TW (1) TW530058B (ja)
UA (1) UA66801C2 (ja)
WO (1) WO1999005143A1 (ja)

Families Citing this family (79)

* Cited by examiner, † Cited by third party
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TWI229674B (en) 1998-12-04 2005-03-21 Astra Pharma Prod Novel triazolo[4,5-d]pyrimidine compounds, pharmaceutical composition containing the same, their process for preparation and uses
SE9903290D0 (sv) * 1999-09-15 1999-09-15 Astra Pharma Prod Novel compounds
SE9904129D0 (sv) 1999-11-15 1999-11-15 Astra Pharma Prod Novel compounds
SE9904128D0 (sv) * 1999-11-15 1999-11-15 Astra Pharma Prod Novel compounds
GB0013487D0 (en) * 2000-06-02 2000-07-26 Astrazeneca Ab Novel process
GB0013488D0 (en) 2000-06-02 2000-07-26 Astrazeneca Ab Chemical compound
GB0013407D0 (en) * 2000-06-02 2000-07-26 Astrazeneca Ab Forms of a chemical compound
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SE0004098D0 (sv) 2000-11-09 2000-11-09 Astrazeneca Ab Novel compounds
SE0004099D0 (sv) * 2000-11-09 2000-11-09 Astrazeneca Ab Novel compounds
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US7504497B2 (en) 2003-10-21 2009-03-17 Inspire Pharmaceuticals, Inc. Orally bioavailable compounds and methods for inhibiting platelet aggregation
SE0401001D0 (sv) 2004-03-31 2004-03-31 Astrazeneca Ab Chemical process
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GB0615620D0 (en) 2006-08-05 2006-09-13 Astrazeneca Ab A process for the preparation of optically active intermediates
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US9006449B2 (en) * 2010-07-29 2015-04-14 Oryzon Genomics, S.A. Cyclopropylamine derivatives useful as LSD1 inhibitors
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CN107573333B (zh) * 2013-04-10 2019-10-18 江苏恒瑞医药股份有限公司 替格瑞洛的中间体及其制备方法和替格瑞洛的制备方法
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TR201601835A2 (tr) 2016-02-12 2017-08-21 Ali Raif Ilac Sanayi Ve Ticaret Anonim Sirketi Ti̇kagrelor i̇çeren formülasyonlar i̇çi̇n üreti̇m yöntemi̇
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WO2023213198A1 (zh) * 2022-05-04 2023-11-09 华东师范大学 芳香稠环化合物作为trek-1激活剂的用途、包含其的药物组合物、镇痛剂
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Also Published As

Publication number Publication date
RU2225407C2 (ru) 2004-03-10
BR9810802B1 (pt) 2010-10-19
NZ502381A (en) 2001-12-21
CN1270590A (zh) 2000-10-18
IS5354A (is) 2000-01-20
EP0996621A1 (en) 2000-05-03
JP4187406B2 (ja) 2008-11-26
NO20000312L (no) 2000-03-21
HU230074B1 (hu) 2015-06-29
AR017014A1 (es) 2001-08-22
PL200325B1 (pl) 2008-12-31
MY123196A (en) 2006-05-31
ATE251161T1 (de) 2003-10-15
KR100535837B1 (ko) 2006-01-12
DE69818668D1 (de) 2003-11-06
DE69818668T2 (de) 2004-08-12
NO315854B1 (no) 2003-11-03
CN1154650C (zh) 2004-06-23
AR077553A2 (es) 2011-09-07
BR9810802A (pt) 2000-09-12
KR20010022083A (ko) 2001-03-15
SK284199B6 (sk) 2004-10-05
ES2207846T3 (es) 2004-06-01
CA2296665C (en) 2008-06-10
NO20000312D0 (no) 2000-01-21
HUP0004333A2 (hu) 2001-04-28
TR200000197T2 (tr) 2000-06-21
PL338516A1 (en) 2000-11-06
JP2001510842A (ja) 2001-08-07
AU745381B2 (en) 2002-03-21
EE200000044A (et) 2000-10-16
UA66801C2 (uk) 2004-06-15
IL133959A0 (en) 2001-04-30
EE04193B1 (et) 2003-12-15
HUP0004333A3 (en) 2001-11-28
EG24412A (en) 2009-05-25
PT996621E (pt) 2004-02-27
IS2236B (is) 2007-05-15
CA2296665A1 (en) 1999-02-04
EP0996621B1 (en) 2003-10-01
KR20050084540A (ko) 2005-08-26
IL133959A (en) 2007-10-31
WO1999005143A1 (en) 1999-02-04
CZ2000233A3 (cs) 2000-07-12
HK1026421A1 (en) 2000-12-15
TW530058B (en) 2003-05-01
SK188199A3 (en) 2000-10-09
CZ302629B6 (cs) 2011-08-10
AU8370698A (en) 1999-02-16
SA98190487B1 (ar) 2006-08-20

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