DE69703294T2 - Zusammensetzungen die konjugate von cis-docosahexaenoic-säure und taxotere enthalten - Google Patents

Zusammensetzungen die konjugate von cis-docosahexaenoic-säure und taxotere enthalten

Info

Publication number
DE69703294T2
DE69703294T2 DE69703294T DE69703294T DE69703294T2 DE 69703294 T2 DE69703294 T2 DE 69703294T2 DE 69703294 T DE69703294 T DE 69703294T DE 69703294 T DE69703294 T DE 69703294T DE 69703294 T2 DE69703294 T2 DE 69703294T2
Authority
DE
Germany
Prior art keywords
conjugate
composition
pharmaceutical composition
acid
taxotere
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69703294T
Other languages
German (de)
English (en)
Other versions
DE69703294D1 (de
Inventor
O. Bradley
E. Shashoua
S. Swindell
L. Webb
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
American Regent Inc
Original Assignee
Protarga Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Protarga Inc filed Critical Protarga Inc
Publication of DE69703294D1 publication Critical patent/DE69703294D1/de
Application granted granted Critical
Publication of DE69703294T2 publication Critical patent/DE69703294T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/542—Carboxylic acids, e.g. a fatty acid or an amino acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
DE69703294T 1996-05-22 1997-05-22 Zusammensetzungen die konjugate von cis-docosahexaenoic-säure und taxotere enthalten Expired - Lifetime DE69703294T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US65142996A 1996-05-22 1996-05-22
PCT/US1997/008866 WO1997044026A1 (en) 1996-05-22 1997-05-22 Compositions comprising conjugates of cis-docosahexaenoic acid and taxotere

Publications (2)

Publication Number Publication Date
DE69703294D1 DE69703294D1 (de) 2000-11-16
DE69703294T2 true DE69703294T2 (de) 2001-05-17

Family

ID=24612833

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69703294T Expired - Lifetime DE69703294T2 (de) 1996-05-22 1997-05-22 Zusammensetzungen die konjugate von cis-docosahexaenoic-säure und taxotere enthalten

Country Status (9)

Country Link
US (1) US6080877A (enExample)
EP (1) EP0914116B1 (enExample)
JP (1) JP4172726B2 (enExample)
AT (1) ATE196844T1 (enExample)
CA (1) CA2255615C (enExample)
DE (1) DE69703294T2 (enExample)
DK (1) DK0914116T3 (enExample)
ES (1) ES2151277T3 (enExample)
WO (1) WO1997044026A1 (enExample)

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Also Published As

Publication number Publication date
DE69703294D1 (de) 2000-11-16
US6080877A (en) 2000-06-27
AU722912B2 (en) 2000-08-17
EP0914116A1 (en) 1999-05-12
ATE196844T1 (de) 2000-10-15
CA2255615A1 (en) 1997-11-27
AU3142497A (en) 1997-12-09
ES2151277T3 (es) 2000-12-16
DK0914116T3 (da) 2000-11-20
JP2000511188A (ja) 2000-08-29
WO1997044026A1 (en) 1997-11-27
EP0914116B1 (en) 2000-10-11
CA2255615C (en) 2006-08-29
JP4172726B2 (ja) 2008-10-29

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