DE60326080D1 - Thiadiazoldioxide und thiadiazoloxide als cxc- und cc-chemokinrezeptor liganden - Google Patents

Thiadiazoldioxide und thiadiazoloxide als cxc- und cc-chemokinrezeptor liganden

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Publication number
DE60326080D1
DE60326080D1 DE60326080T DE60326080T DE60326080D1 DE 60326080 D1 DE60326080 D1 DE 60326080D1 DE 60326080 T DE60326080 T DE 60326080T DE 60326080 T DE60326080 T DE 60326080T DE 60326080 D1 DE60326080 D1 DE 60326080D1
Authority
DE
Germany
Prior art keywords
und
thiadiazoloxide
thiadiazoldioxide
chemokinrezeptor
liganden
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60326080T
Other languages
German (de)
English (en)
Inventor
Arthur G Taveras
Jianhua Chao
Purakkattle J Biju
Younong Yu
Jay S Fine
William Hipkin
Cynthia J Aki
Robert J Merritt
Ge Li
John J Baldwin
Gaifa Lai
Minglang Wu
Evan A Hecker
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Sharp and Dohme LLC
Pharmacopeia LLC
Original Assignee
Pharmacopeia Inc
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacopeia Inc, Schering Corp filed Critical Pharmacopeia Inc
Application granted granted Critical
Publication of DE60326080D1 publication Critical patent/DE60326080D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
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AU2003288922A1 (en) 2004-05-04
MY139601A (en) 2009-10-30
ES2321186T3 (es) 2009-06-03
JP2006508079A (ja) 2006-03-09
AR043052A1 (es) 2005-07-13
JP2010270151A (ja) 2010-12-02
CN1720240A (zh) 2006-01-11
HK1072432A1 (en) 2005-10-28
MXPA05003867A (es) 2005-11-23
PE20040570A1 (es) 2004-08-30
US20040186142A1 (en) 2004-09-23
WO2004033440A1 (en) 2004-04-22
WO2004033440A8 (en) 2005-06-02
EP1551818A1 (en) 2005-07-13
ATE422203T1 (de) 2009-02-15
TW200413342A (en) 2004-08-01
CA2501535A1 (en) 2004-04-22
CN1720240B (zh) 2010-10-27
US7691856B2 (en) 2010-04-06
JP4664074B2 (ja) 2011-04-06
US20070264230A1 (en) 2007-11-15

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