CA2501535A1 - Thiadiazoledioxides and thiadiazoleoxides as cxc- and cc-chemokine receptor ligands - Google Patents

Thiadiazoledioxides and thiadiazoleoxides as cxc- and cc-chemokine receptor ligands Download PDF

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Publication number
CA2501535A1
CA2501535A1 CA002501535A CA2501535A CA2501535A1 CA 2501535 A1 CA2501535 A1 CA 2501535A1 CA 002501535 A CA002501535 A CA 002501535A CA 2501535 A CA2501535 A CA 2501535A CA 2501535 A1 CA2501535 A1 CA 2501535A1
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Canada
Prior art keywords
group
compound
pharmaceutically acceptable
formula
substituted
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Abandoned
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CA002501535A
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English (en)
French (fr)
Inventor
Arthur G. Taveras
Jianhua Chao
Purakkattle J. Biju
Younong Yu
Jay S. Fine
William Hipkin
Cynthia J. Aki
J. Robert Merritt
Ge Li
John J. Baldwin
Gaifa Lai
Minglang Wu
Evan A. Hecker
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Merck Sharp & Dohme LLC
Pharmacopeia LLC
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Individual
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Publication of CA2501535A1 publication Critical patent/CA2501535A1/en
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
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US20040186142A1 (en) 2004-09-23
WO2004033440A1 (en) 2004-04-22
WO2004033440A8 (en) 2005-06-02
JP2010270151A (ja) 2010-12-02
US20070264230A1 (en) 2007-11-15
AU2003288922A1 (en) 2004-05-04
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CN1720240B (zh) 2010-10-27
AR043052A1 (es) 2005-07-13
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JP4664074B2 (ja) 2011-04-06
ATE422203T1 (de) 2009-02-15
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MXPA05003867A (es) 2005-11-23
HK1072432A1 (en) 2005-10-28
US7691856B2 (en) 2010-04-06
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