AU2003288922A1 - Thiadiazoledioxides and thiadiazoleoxides as cxc- and cc-chemokine receptor ligands - Google Patents

Thiadiazoledioxides and thiadiazoleoxides as cxc- and cc-chemokine receptor ligands

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Publication number
AU2003288922A1
AU2003288922A1 AU2003288922A AU2003288922A AU2003288922A1 AU 2003288922 A1 AU2003288922 A1 AU 2003288922A1 AU 2003288922 A AU2003288922 A AU 2003288922A AU 2003288922 A AU2003288922 A AU 2003288922A AU 2003288922 A1 AU2003288922 A1 AU 2003288922A1
Authority
AU
Australia
Prior art keywords
thiadiazoleoxides
thiadiazoledioxides
cxc
chemokine receptor
receptor ligands
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003288922A
Other languages
English (en)
Inventor
Cynthia J. Aki
John J. Baldwin
Purakkattle J. Biju
Jianhua Chao
Jay S. Fine
Evan A. Hecker
William Hipkin
Gaifa Lai
Ge Li
J. Robert Merritt
Arthur G. Taveras
Minglang Wu
Younong Yu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacopeia LLC
Original Assignee
Pharmacopeia Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacopeia Inc filed Critical Pharmacopeia Inc
Publication of AU2003288922A1 publication Critical patent/AU2003288922A1/en
Abandoned legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
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US20040186142A1 (en) 2004-09-23
PE20040570A1 (es) 2004-08-30
CN1720240B (zh) 2010-10-27
WO2004033440A1 (en) 2004-04-22
WO2004033440A8 (en) 2005-06-02
JP2010270151A (ja) 2010-12-02
DE60326080D1 (en) 2009-03-19
MXPA05003867A (es) 2005-11-23
HK1072432A1 (en) 2005-10-28
TW200413342A (en) 2004-08-01
JP2006508079A (ja) 2006-03-09
EP1551818B1 (en) 2009-02-04
ES2321186T3 (es) 2009-06-03
EP1551818A1 (en) 2005-07-13
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MY139601A (en) 2009-10-30
US7691856B2 (en) 2010-04-06
JP4664074B2 (ja) 2011-04-06
CA2501535A1 (en) 2004-04-22
AR043052A1 (es) 2005-07-13

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