DE60308349T2 - Terphenylderivate, deren herstellung und zusammensetzungen, die diese enthalten - Google Patents
Terphenylderivate, deren herstellung und zusammensetzungen, die diese enthalten Download PDFInfo
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- DE60308349T2 DE60308349T2 DE60308349T DE60308349T DE60308349T2 DE 60308349 T2 DE60308349 T2 DE 60308349T2 DE 60308349 T DE60308349 T DE 60308349T DE 60308349 T DE60308349 T DE 60308349T DE 60308349 T2 DE60308349 T2 DE 60308349T2
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- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
- C07D295/28—Nitrogen atoms
- C07D295/32—Nitrogen atoms acylated with carboxylic or carbonic acids, or their nitrogen or sulfur analogues
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- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/16—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with acylated ring nitrogen atom
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- C07D211/98—Nitrogen atom
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- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/14—All rings being cycloaliphatic
- C07C2602/22—All rings being cycloaliphatic the ring system containing eight carbon atoms, e.g. pentalene
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Diabetes (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Endocrinology (AREA)
- Ophthalmology & Optometry (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
- Oncology (AREA)
- Reproductive Health (AREA)
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- Communicable Diseases (AREA)
- Hospice & Palliative Care (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0204567A FR2838439B1 (fr) | 2002-04-11 | 2002-04-11 | Derives de terphenyle, leur preparation, les compositions pharmaceutqiues en contenant |
| FR0204567 | 2002-04-11 | ||
| PCT/FR2003/001134 WO2003084943A2 (fr) | 2002-04-11 | 2003-04-10 | Derives de terphenyle, leur preparation, les compositions pharmaceutiques en contenant |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE60308349D1 DE60308349D1 (de) | 2006-10-26 |
| DE60308349T2 true DE60308349T2 (de) | 2007-04-19 |
Family
ID=28459770
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE60308349T Expired - Lifetime DE60308349T2 (de) | 2002-04-11 | 2003-04-10 | Terphenylderivate, deren herstellung und zusammensetzungen, die diese enthalten |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US7390924B2 (enExample) |
| EP (1) | EP1497274B1 (enExample) |
| JP (1) | JP4634717B2 (enExample) |
| CN (1) | CN100432062C (enExample) |
| AT (1) | ATE339408T1 (enExample) |
| AU (1) | AU2003246811A1 (enExample) |
| BR (1) | BR0309106A (enExample) |
| CA (1) | CA2481392A1 (enExample) |
| DE (1) | DE60308349T2 (enExample) |
| FR (1) | FR2838439B1 (enExample) |
| MX (1) | MXPA04009981A (enExample) |
| PL (1) | PL374024A1 (enExample) |
| WO (1) | WO2003084943A2 (enExample) |
Families Citing this family (59)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1492784A4 (en) | 2002-03-28 | 2006-03-29 | Merck & Co Inc | SUBSTITUTED 2,3-DIPHENYLPYRIDINES |
| AU2003275242B2 (en) | 2002-09-27 | 2010-03-04 | Merck Sharp & Dohme Corp. | Substituted pyrimidines |
| US7129239B2 (en) | 2002-10-28 | 2006-10-31 | Pfizer Inc. | Purine compounds and uses thereof |
| US7247628B2 (en) | 2002-12-12 | 2007-07-24 | Pfizer, Inc. | Cannabinoid receptor ligands and uses thereof |
| US7772188B2 (en) | 2003-01-28 | 2010-08-10 | Ironwood Pharmaceuticals, Inc. | Methods and compositions for the treatment of gastrointestinal disorders |
| US7329658B2 (en) | 2003-02-06 | 2008-02-12 | Pfizer Inc | Cannabinoid receptor ligands and uses thereof |
| US7176210B2 (en) | 2003-02-10 | 2007-02-13 | Pfizer Inc. | Cannabinoid receptor ligands and uses thereof |
| US7141669B2 (en) | 2003-04-23 | 2006-11-28 | Pfizer Inc. | Cannabiniod receptor ligands and uses thereof |
| US7268133B2 (en) | 2003-04-23 | 2007-09-11 | Pfizer, Inc. Patent Department | Cannabinoid receptor ligands and uses thereof |
| US7145012B2 (en) | 2003-04-23 | 2006-12-05 | Pfizer Inc. | Cannabinoid receptor ligands and uses thereof |
| US7232823B2 (en) | 2003-06-09 | 2007-06-19 | Pfizer, Inc. | Cannabinoid receptor ligands and uses thereof |
| FR2856684B1 (fr) | 2003-06-26 | 2008-04-11 | Sanofi Synthelabo | Derives de diphenylpyridine, leur preparation et leur application en therapeutique |
| WO2005075450A2 (en) | 2004-01-28 | 2005-08-18 | F. Hoffmann-La Roche Ag | Spiro-benzodioxoles and their use as cb1 antagonists |
| EP1574211A1 (en) * | 2004-03-09 | 2005-09-14 | Inserm | Use of antagonists of the CB1 receptor for the manufacture of a composition useful for the treatment of hepatic diseases |
| US20080125403A1 (en) | 2004-04-02 | 2008-05-29 | Merck & Co., Inc. | Method of Treating Men with Metabolic and Anthropometric Disorders |
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| WO2012120055A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| EP2766349B1 (de) | 2011-03-08 | 2016-06-01 | Sanofi | Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
| US8846666B2 (en) | 2011-03-08 | 2014-09-30 | Sanofi | Oxathiazine derivatives which are substituted with benzyl or heteromethylene groups, method for producing them, their use as medicine and drug containing said derivatives and the use thereof |
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| WO2012120054A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
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| PL3004138T3 (pl) | 2013-06-05 | 2024-07-29 | Bausch Health Ireland Limited | Ultra-oczyszczeni agoniści peptydowi cyklazy guanylanowej C, sposób ich uzyskiwania i ich zastosowanie |
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| WO2018159650A1 (ja) * | 2017-02-28 | 2018-09-07 | 東レ株式会社 | グアニジン誘導体及びその医薬用途 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4916145A (en) * | 1987-07-10 | 1990-04-10 | Hoffmann-La Roche Inc. | Substituted n-[(pyridyl)alkyl]aryl-carboxamide |
| FR2800375B1 (fr) * | 1999-11-03 | 2004-07-23 | Sanofi Synthelabo | Derives tricycliques d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant |
-
2002
- 2002-04-11 FR FR0204567A patent/FR2838439B1/fr not_active Expired - Fee Related
-
2003
- 2003-04-10 EP EP03745842A patent/EP1497274B1/fr not_active Expired - Lifetime
- 2003-04-10 US US10/511,040 patent/US7390924B2/en not_active Expired - Fee Related
- 2003-04-10 MX MXPA04009981A patent/MXPA04009981A/es active IP Right Grant
- 2003-04-10 CA CA002481392A patent/CA2481392A1/fr not_active Abandoned
- 2003-04-10 DE DE60308349T patent/DE60308349T2/de not_active Expired - Lifetime
- 2003-04-10 WO PCT/FR2003/001134 patent/WO2003084943A2/fr not_active Ceased
- 2003-04-10 AU AU2003246811A patent/AU2003246811A1/en not_active Abandoned
- 2003-04-10 CN CNB038130068A patent/CN100432062C/zh not_active Expired - Fee Related
- 2003-04-10 JP JP2003582140A patent/JP4634717B2/ja not_active Expired - Fee Related
- 2003-04-10 PL PL03374024A patent/PL374024A1/xx not_active Application Discontinuation
- 2003-04-10 BR BR0309106-6A patent/BR0309106A/pt not_active IP Right Cessation
- 2003-04-10 AT AT03745842T patent/ATE339408T1/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| CN100432062C (zh) | 2008-11-12 |
| JP4634717B2 (ja) | 2011-02-16 |
| MXPA04009981A (es) | 2005-07-01 |
| CN1659157A (zh) | 2005-08-24 |
| BR0309106A (pt) | 2005-02-01 |
| DE60308349D1 (de) | 2006-10-26 |
| CA2481392A1 (fr) | 2003-10-16 |
| EP1497274B1 (fr) | 2006-09-13 |
| FR2838439A1 (fr) | 2003-10-17 |
| EP1497274A2 (fr) | 2005-01-19 |
| AU2003246811A8 (en) | 2003-10-20 |
| PL374024A1 (en) | 2005-09-19 |
| FR2838439B1 (fr) | 2005-05-20 |
| JP2005534620A (ja) | 2005-11-17 |
| US20060167049A1 (en) | 2006-07-27 |
| WO2003084943A2 (fr) | 2003-10-16 |
| ATE339408T1 (de) | 2006-10-15 |
| WO2003084943A9 (fr) | 2004-06-10 |
| AU2003246811A1 (en) | 2003-10-20 |
| WO2003084943A3 (fr) | 2004-04-01 |
| US7390924B2 (en) | 2008-06-24 |
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