AU2003246811A1 - Terphenyl derivatives, preparation thereof, compositions containing same - Google Patents
Terphenyl derivatives, preparation thereof, compositions containing sameInfo
- Publication number
- AU2003246811A1 AU2003246811A1 AU2003246811A AU2003246811A AU2003246811A1 AU 2003246811 A1 AU2003246811 A1 AU 2003246811A1 AU 2003246811 A AU2003246811 A AU 2003246811A AU 2003246811 A AU2003246811 A AU 2003246811A AU 2003246811 A1 AU2003246811 A1 AU 2003246811A1
- Authority
- AU
- Australia
- Prior art keywords
- preparation
- compositions containing
- containing same
- terphenyl derivatives
- sub
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
- C07D295/28—Nitrogen atoms
- C07D295/32—Nitrogen atoms acylated with carboxylic or carbonic acids, or their nitrogen or sulfur analogues
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- C07C233/69—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of an acyclic saturated carbon skeleton
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- C07C233/78—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
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- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
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- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C07D209/16—Tryptamines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/16—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with acylated ring nitrogen atom
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- C07D211/92—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
- C07D211/98—Nitrogen atom
-
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- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/14—All rings being cycloaliphatic
- C07C2602/22—All rings being cycloaliphatic the ring system containing eight carbon atoms, e.g. pentalene
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Immunology (AREA)
- Reproductive Health (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Hospice & Palliative Care (AREA)
- Rheumatology (AREA)
- Pulmonology (AREA)
- Psychology (AREA)
- Ophthalmology & Optometry (AREA)
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- Pregnancy & Childbirth (AREA)
- Gastroenterology & Hepatology (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR02/04567 | 2002-04-11 | ||
| FR0204567A FR2838439B1 (fr) | 2002-04-11 | 2002-04-11 | Derives de terphenyle, leur preparation, les compositions pharmaceutqiues en contenant |
| PCT/FR2003/001134 WO2003084943A2 (fr) | 2002-04-11 | 2003-04-10 | Derives de terphenyle, leur preparation, les compositions pharmaceutiques en contenant |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2003246811A1 true AU2003246811A1 (en) | 2003-10-20 |
| AU2003246811A8 AU2003246811A8 (en) | 2003-10-20 |
Family
ID=28459770
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2003246811A Abandoned AU2003246811A1 (en) | 2002-04-11 | 2003-04-10 | Terphenyl derivatives, preparation thereof, compositions containing same |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US7390924B2 (enExample) |
| EP (1) | EP1497274B1 (enExample) |
| JP (1) | JP4634717B2 (enExample) |
| CN (1) | CN100432062C (enExample) |
| AT (1) | ATE339408T1 (enExample) |
| AU (1) | AU2003246811A1 (enExample) |
| BR (1) | BR0309106A (enExample) |
| CA (1) | CA2481392A1 (enExample) |
| DE (1) | DE60308349T2 (enExample) |
| FR (1) | FR2838439B1 (enExample) |
| MX (1) | MXPA04009981A (enExample) |
| PL (1) | PL374024A1 (enExample) |
| WO (1) | WO2003084943A2 (enExample) |
Families Citing this family (59)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7271266B2 (en) | 2002-03-28 | 2007-09-18 | Merck & Co., Inc. | Substituted 2,3-diphenyl pyridines |
| WO2004029204A2 (en) | 2002-09-27 | 2004-04-08 | Merck & Co., Inc. | Substituted pyrimidines |
| US7129239B2 (en) | 2002-10-28 | 2006-10-31 | Pfizer Inc. | Purine compounds and uses thereof |
| US7247628B2 (en) | 2002-12-12 | 2007-07-24 | Pfizer, Inc. | Cannabinoid receptor ligands and uses thereof |
| US7772188B2 (en) | 2003-01-28 | 2010-08-10 | Ironwood Pharmaceuticals, Inc. | Methods and compositions for the treatment of gastrointestinal disorders |
| US7329658B2 (en) | 2003-02-06 | 2008-02-12 | Pfizer Inc | Cannabinoid receptor ligands and uses thereof |
| US7176210B2 (en) | 2003-02-10 | 2007-02-13 | Pfizer Inc. | Cannabinoid receptor ligands and uses thereof |
| US7145012B2 (en) | 2003-04-23 | 2006-12-05 | Pfizer Inc. | Cannabinoid receptor ligands and uses thereof |
| US7268133B2 (en) | 2003-04-23 | 2007-09-11 | Pfizer, Inc. Patent Department | Cannabinoid receptor ligands and uses thereof |
| US7141669B2 (en) | 2003-04-23 | 2006-11-28 | Pfizer Inc. | Cannabiniod receptor ligands and uses thereof |
| US7232823B2 (en) | 2003-06-09 | 2007-06-19 | Pfizer, Inc. | Cannabinoid receptor ligands and uses thereof |
| FR2856684B1 (fr) * | 2003-06-26 | 2008-04-11 | Sanofi Synthelabo | Derives de diphenylpyridine, leur preparation et leur application en therapeutique |
| JP4436369B2 (ja) | 2004-01-28 | 2010-03-24 | エフ.ホフマン−ラ ロシュ アーゲー | スピロ−ベンゾジオキソール類およびそれらのcb1アンタゴニストとしての使用 |
| EP1574211A1 (en) * | 2004-03-09 | 2005-09-14 | Inserm | Use of antagonists of the CB1 receptor for the manufacture of a composition useful for the treatment of hepatic diseases |
| EP1734963A4 (en) | 2004-04-02 | 2008-06-18 | Merck & Co Inc | METHOD FOR TREATING PEOPLE WITH METABOLIC AND ANTHROPOMETRIC DISORDER |
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| EP2683703B1 (de) | 2011-03-08 | 2015-05-27 | Sanofi | Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
| WO2012120053A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| US8846666B2 (en) | 2011-03-08 | 2014-09-30 | Sanofi | Oxathiazine derivatives which are substituted with benzyl or heteromethylene groups, method for producing them, their use as medicine and drug containing said derivatives and the use thereof |
| EP2683702B1 (de) | 2011-03-08 | 2014-12-24 | Sanofi | Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
| EP2683705B1 (de) | 2011-03-08 | 2015-04-22 | Sanofi | Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| WO2012120051A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Mit adamantan- oder noradamantan substituierte benzyl-oxathiazinderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
| WO2012120056A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
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| WO2018159650A1 (ja) * | 2017-02-28 | 2018-09-07 | 東レ株式会社 | グアニジン誘導体及びその医薬用途 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4916145A (en) * | 1987-07-10 | 1990-04-10 | Hoffmann-La Roche Inc. | Substituted n-[(pyridyl)alkyl]aryl-carboxamide |
| FR2800375B1 (fr) * | 1999-11-03 | 2004-07-23 | Sanofi Synthelabo | Derives tricycliques d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant |
-
2002
- 2002-04-11 FR FR0204567A patent/FR2838439B1/fr not_active Expired - Fee Related
-
2003
- 2003-04-10 AU AU2003246811A patent/AU2003246811A1/en not_active Abandoned
- 2003-04-10 EP EP03745842A patent/EP1497274B1/fr not_active Expired - Lifetime
- 2003-04-10 BR BR0309106-6A patent/BR0309106A/pt not_active IP Right Cessation
- 2003-04-10 DE DE60308349T patent/DE60308349T2/de not_active Expired - Lifetime
- 2003-04-10 CN CNB038130068A patent/CN100432062C/zh not_active Expired - Fee Related
- 2003-04-10 AT AT03745842T patent/ATE339408T1/de not_active IP Right Cessation
- 2003-04-10 MX MXPA04009981A patent/MXPA04009981A/es active IP Right Grant
- 2003-04-10 US US10/511,040 patent/US7390924B2/en not_active Expired - Fee Related
- 2003-04-10 JP JP2003582140A patent/JP4634717B2/ja not_active Expired - Fee Related
- 2003-04-10 CA CA002481392A patent/CA2481392A1/fr not_active Abandoned
- 2003-04-10 PL PL03374024A patent/PL374024A1/xx not_active Application Discontinuation
- 2003-04-10 WO PCT/FR2003/001134 patent/WO2003084943A2/fr not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2003084943A2 (fr) | 2003-10-16 |
| DE60308349D1 (de) | 2006-10-26 |
| DE60308349T2 (de) | 2007-04-19 |
| ATE339408T1 (de) | 2006-10-15 |
| WO2003084943A3 (fr) | 2004-04-01 |
| MXPA04009981A (es) | 2005-07-01 |
| WO2003084943A9 (fr) | 2004-06-10 |
| BR0309106A (pt) | 2005-02-01 |
| FR2838439B1 (fr) | 2005-05-20 |
| JP4634717B2 (ja) | 2011-02-16 |
| JP2005534620A (ja) | 2005-11-17 |
| CA2481392A1 (fr) | 2003-10-16 |
| CN1659157A (zh) | 2005-08-24 |
| AU2003246811A8 (en) | 2003-10-20 |
| EP1497274A2 (fr) | 2005-01-19 |
| PL374024A1 (en) | 2005-09-19 |
| US7390924B2 (en) | 2008-06-24 |
| EP1497274B1 (fr) | 2006-09-13 |
| FR2838439A1 (fr) | 2003-10-17 |
| CN100432062C (zh) | 2008-11-12 |
| US20060167049A1 (en) | 2006-07-27 |
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