DE602004010829D1 - Adamantan- und azabicyclooctan- und -nonanderivate, verfahren zu deren herstellung und deren verwendung als dpp-iv-inhibitoren - Google Patents

Adamantan- und azabicyclooctan- und -nonanderivate, verfahren zu deren herstellung und deren verwendung als dpp-iv-inhibitoren

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Publication number
DE602004010829D1
DE602004010829D1 DE602004010829T DE602004010829T DE602004010829D1 DE 602004010829 D1 DE602004010829 D1 DE 602004010829D1 DE 602004010829 T DE602004010829 T DE 602004010829T DE 602004010829 T DE602004010829 T DE 602004010829T DE 602004010829 D1 DE602004010829 D1 DE 602004010829D1
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Germany
Prior art keywords
preparation
nonanderivates
azabicyclooctanese
adamantan
dpp
Prior art date
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Expired - Lifetime
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DE602004010829T
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English (en)
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DE602004010829T2 (de
Inventor
Peter Aranyi
Imre Bata
Sandor Batori
Eva Boronkay
Philippe Bovy
Zoltan Kapui
Edit Susan
Tibor Szabo
Katalin Urban-Szabo
Marton Varga
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Sanofi Aventis France
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Sanofi Aventis France
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Publication of DE602004010829D1 publication Critical patent/DE602004010829D1/de
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    • C04BLIME, MAGNESIA; SLAG; CEMENTS; COMPOSITIONS THEREOF, e.g. MORTARS, CONCRETE OR LIKE BUILDING MATERIALS; ARTIFICIAL STONE; CERAMICS; REFRACTORIES; TREATMENT OF NATURAL STONE
    • C04B35/00Shaped ceramic products characterised by their composition; Ceramics compositions; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/622Forming processes; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/626Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B
    • C04B35/63Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
    • C04B35/632Organic additives
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    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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DE602004010829T 2003-08-29 2004-08-27 Adamantan- und azabicyclooctan- und -nonanderivate, verfahren zu deren herstellung und deren verwendung als dpp-iv-inhibitoren Expired - Lifetime DE602004010829T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
HU0302788A HU227684B1 (en) 2003-08-29 2003-08-29 Adamantane and azabicyclo-octane and nonane derivatives and their use as dpp-iv inhibitors
HU0302788 2003-08-29
PCT/HU2004/000088 WO2005021536A2 (en) 2003-08-29 2004-08-27 Adamantane and azabicyclo-octane and nonane derivatives, process of their preparation and their use as dpp-iv inhibitors

Publications (2)

Publication Number Publication Date
DE602004010829D1 true DE602004010829D1 (de) 2008-01-31
DE602004010829T2 DE602004010829T2 (de) 2008-12-11

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CA2537123A1 (en) 2005-03-10
JP4853965B2 (ja) 2012-01-11
WO2005021536A3 (en) 2005-10-13
US7652021B2 (en) 2010-01-26
JP2007504120A (ja) 2007-03-01
IL173802A (en) 2011-08-31
US20060276487A1 (en) 2006-12-07
US20100160328A1 (en) 2010-06-24
HUP0302788A3 (en) 2008-09-29
EP1664031B1 (de) 2007-12-19
CN1845921A (zh) 2006-10-11
MXPA06002345A (es) 2006-05-19
ATE381559T1 (de) 2008-01-15
AU2004268832A1 (en) 2005-03-10
BRPI0413973A (pt) 2006-10-31
IL173802A0 (en) 2006-07-05
WO2005021536A2 (en) 2005-03-10
EP1664031A2 (de) 2006-06-07
HU227684B1 (en) 2011-11-28
DE602004010829T2 (de) 2008-12-11
HUP0302788A2 (en) 2007-09-28
HU0302788D0 (en) 2003-10-28
AU2004268832B2 (en) 2011-04-28
KR20060121838A (ko) 2006-11-29

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