DE60144570D1 - Verfahren zur herstellung von optisch aktiven sulfonamiden und zwischenprodukte zur deren synthese - Google Patents

Verfahren zur herstellung von optisch aktiven sulfonamiden und zwischenprodukte zur deren synthese

Info

Publication number
DE60144570D1
DE60144570D1 DE60144570T DE60144570T DE60144570D1 DE 60144570 D1 DE60144570 D1 DE 60144570D1 DE 60144570 T DE60144570 T DE 60144570T DE 60144570 T DE60144570 T DE 60144570T DE 60144570 D1 DE60144570 D1 DE 60144570D1
Authority
DE
Germany
Prior art keywords
optically active
optionally substituted
intermediates
synthesis
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60144570T
Other languages
English (en)
Inventor
Tomomi Ikemoto
Atsuko Nishiguchi
Kiminori Tomimatsu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Takeda Pharmaceutical Co Ltd
Original Assignee
Takeda Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical Co Ltd filed Critical Takeda Pharmaceutical Co Ltd
Application granted granted Critical
Publication of DE60144570D1 publication Critical patent/DE60144570D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/50—Compounds containing any of the groups, X being a hetero atom, Y being any atom
    • C07C311/51—Y being a hydrogen or a carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C07C303/40—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reactions not involving the formation of sulfonamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/42—Separation; Purification; Stabilisation; Use of additives
    • C07C303/44—Separation; Purification
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/14—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/16—Systems containing only non-condensed rings with a six-membered ring the ring being unsaturated
DE60144570T 2000-10-18 2001-10-17 Verfahren zur herstellung von optisch aktiven sulfonamiden und zwischenprodukte zur deren synthese Expired - Lifetime DE60144570D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2000323309 2000-10-18
PCT/JP2001/009120 WO2002032859A1 (fr) 2000-10-18 2001-10-17 Procede de preparation de sulfonamides optiquement actifs et intermediaires pour leur synthese

Publications (1)

Publication Number Publication Date
DE60144570D1 true DE60144570D1 (de) 2011-06-16

Family

ID=18801004

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60144570T Expired - Lifetime DE60144570D1 (de) 2000-10-18 2001-10-17 Verfahren zur herstellung von optisch aktiven sulfonamiden und zwischenprodukte zur deren synthese

Country Status (9)

Country Link
US (1) US6982344B2 (de)
EP (1) EP1334966B1 (de)
JP (1) JP4012389B2 (de)
KR (1) KR100821546B1 (de)
AT (1) ATE508109T1 (de)
AU (1) AU2001295949A1 (de)
CA (1) CA2426277C (de)
DE (1) DE60144570D1 (de)
WO (1) WO2002032859A1 (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008004673A1 (fr) * 2006-07-07 2008-01-10 Takeda Pharmaceutical Company Limited Dérives de cycloalkène, procédé de production des dérivés et utilisation de ceux-ci
JPWO2008114831A1 (ja) * 2007-03-20 2010-07-08 国立大学法人 岡山大学 スルホンアミド基を有する抗菌剤
MY163936A (en) 2010-01-27 2017-11-15 Takeda Pharmaceuticals Co Compounds for suppressing a peripheral nerve disorder induced by an anti-cancer agent
CN107406450B (zh) * 2015-03-10 2019-06-04 泸州东方农化有限公司 一种制备高纯度磺胺化合物的方法及其中间体

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0726194A (ja) 1993-07-12 1995-01-27 Japan Synthetic Rubber Co Ltd コーティング用水分散体
EP0721451A1 (de) 1993-09-28 1996-07-17 Novartis AG Acylierte sulfonamide als insektizide und akarizide
JP3799580B2 (ja) * 1995-01-20 2006-07-19 日本曹達株式会社 Ｎ−置換−ｎ−スルホニルアミド類の製造方法
JPH11147873A (ja) 1997-11-13 1999-06-02 Yamanouchi Pharmaceut Co Ltd 新規スルホンアミド誘導体及び医薬
PT1063228E (pt) 1998-03-09 2005-05-31 Takeda Pharmaceutical Derivados de cicloalcenos processo para a sua preparacao e utilizacao
AU1553001A (en) * 1999-11-29 2001-06-12 Takeda Chemical Industries Ltd. Process for the production of optically active cyclohexene derivatives and intermediates therefor

Also Published As

Publication number Publication date
WO2002032859A1 (fr) 2002-04-25
KR100821546B1 (ko) 2008-04-11
CA2426277C (en) 2010-11-30
EP1334966A4 (de) 2007-04-18
EP1334966B1 (de) 2011-05-04
US6982344B2 (en) 2006-01-03
JP2002193916A (ja) 2002-07-10
US20040049041A1 (en) 2004-03-11
CA2426277A1 (en) 2003-04-17
ATE508109T1 (de) 2011-05-15
JP4012389B2 (ja) 2007-11-21
KR20030048440A (ko) 2003-06-19
EP1334966A1 (de) 2003-08-13
AU2001295949A1 (en) 2002-04-29

Similar Documents

Publication Publication Date Title
ATE346062T1 (de) Verfahren zur herstellung von optisch-aktiven sulfoxid-derivaten
DE60100238D1 (de) Synthese von 3,6-Dialkyl-5,6-Dihydro-4-Hydroxy-2H-Pyran-2-one
ATE190614T1 (de) Dihydrat des n-(4-amino-6,7-dimethoxychinazol-2- yl)-n-methyl-n'-(tetrahydrofuroyl-2)- propylendiamin hydrochlorids(=alfuzosin hydrochlorid dihydrat) und ein verfahren zur herstellung
DE60228724D1 (de) Verfahren zur herstellung von beraprost und dessen salzen
DE60235365D1 (de) Verfahren zur herstellung von 7-amino-syn-3,5-dihydroxyheptansäurederivaten und zwischenverbindungen diesesverfahrens und deren herestellung
DE69637770D1 (de) Verfahren zur herstellung von amidderivaten und ihren zwischenverbindungen
HUP9901526A2 (hu) Atorvastatin szintézis, közbenső termékei és eljárás ezek előállítására
DE3767993D1 (de) Verfahren zur herstellung von thienylaethylaminen, und mittels des verfahrens hergestellte dithienylaethylamine.
ATE288891T1 (de) Verfahren zur herstellung von amid-derivaten und ihren zwischenverbindungen
ATE277915T1 (de) Verfahren sowie neue zwischenprodukte zur herstellung von isoxazolin-3-yl-acylbenzolen
DE60144570D1 (de) Verfahren zur herstellung von optisch aktiven sulfonamiden und zwischenprodukte zur deren synthese
DE69521012T2 (de) Verfahren zur Herstellung von 1-(4,5-Dihydro)2-thiazolyl-3-Azetidinthiolderivaten
DE60136566D1 (de) Verfahren zur herstellung von optisch aktiven 2,4-dihydrobenzofuranverbindungen
DE602004003737D1 (de) Verfahren zur Herstellung von disubstituierten 9-Alkylidenfluorenen und deren Derivaten.
ATE282594T1 (de) Verfahren zur herstellung von (+)-trans-4-p- fluorophenyl-3-hydroxymethyl-1-methylpiperidin
DE69529958D1 (de) Aminoalkyloxime, Verfahren zur dessen Herstellung, ihre Verwendung als Medikamente und Zwischenprodukte
ATE150453T1 (de) Verfahren zur herstellung von trans-piperidin-2,5-dicarboxylaten
ATE300534T1 (de) Verfahren und zwischenverbindungen zur herstellung von imidazopyridinen
DE69127960D1 (de) Verfahren zur Herstellung von (S)-vinyl- und (S)-allenyl-Gaba
DE602005002750D1 (de) Chirale heptinderivate zur herstellung von epothilonen und verfahren zu deren herstellung
DE60019619D1 (de) Dihydrobenzofuranderivate, verfahren zu ihrer herstellung und mittel
DE69928610D1 (de) Verfahren zur Herstellung von 2-Carbamoyl-Pyridinen
ATE265421T1 (de) Verfahren zur herstellung von midodrin
DE69731090D1 (de) Thienylcyclohexan-derivte zur herstellung von thienylcyclohexylen
DE602004006896D1 (de) Bis-dicarbonsäuresalze von benazepril und herstellung von benazepril über diese salze