ATE288891T1 - Verfahren zur herstellung von amid-derivaten und ihren zwischenverbindungen - Google Patents

Verfahren zur herstellung von amid-derivaten und ihren zwischenverbindungen

Info

Publication number
ATE288891T1
ATE288891T1 AT96931296T AT96931296T ATE288891T1 AT E288891 T1 ATE288891 T1 AT E288891T1 AT 96931296 T AT96931296 T AT 96931296T AT 96931296 T AT96931296 T AT 96931296T AT E288891 T1 ATE288891 T1 AT E288891T1
Authority
AT
Austria
Prior art keywords
producing
compound
äxvü
äxviü
intermediate compounds
Prior art date
Application number
AT96931296T
Other languages
English (en)
Inventor
Takashi Inaba
Yasuki Yamada
Original Assignee
Japan Tobacco Inc
Agouron Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Japan Tobacco Inc, Agouron Pharma filed Critical Japan Tobacco Inc
Application granted granted Critical
Publication of ATE288891T1 publication Critical patent/ATE288891T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/10—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D263/14—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D321/00—Heterocyclic compounds containing rings having two oxygen atoms as the only ring hetero atoms, not provided for by groups C07D317/00 - C07D319/00
    • C07D321/02—Seven-membered rings
    • C07D321/04—Seven-membered rings not condensed with other rings
    • C07D321/06—1,3-Dioxepines; Hydrogenated 1,3-dioxepines
AT96931296T 1995-09-26 1996-09-24 Verfahren zur herstellung von amid-derivaten und ihren zwischenverbindungen ATE288891T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP24818395 1995-09-26
PCT/JP1996/002756 WO1997011937A1 (fr) 1995-09-26 1996-09-24 Procede de production de derives amides et de leurs intermediaires

Publications (1)

Publication Number Publication Date
ATE288891T1 true ATE288891T1 (de) 2005-02-15

Family

ID=17174443

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96931296T ATE288891T1 (de) 1995-09-26 1996-09-24 Verfahren zur herstellung von amid-derivaten und ihren zwischenverbindungen

Country Status (9)

Country Link
US (5) US6133461A (de)
EP (1) EP0983999B8 (de)
JP (1) JP3566968B2 (de)
AT (1) ATE288891T1 (de)
AU (1) AU717637B2 (de)
DE (1) DE69634345T2 (de)
ES (1) ES2233976T3 (de)
PT (1) PT983999E (de)
WO (1) WO1997011937A1 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5962725A (en) * 1996-09-05 1999-10-05 Agouron Pharmaceuticals, Inc. Intermediate compounds useful for making HIV protease inhibitors such as nelfinavir
US5925759A (en) * 1996-09-05 1999-07-20 Agouron Pharmaceuticals, Inc. Methods of making HIV-protease inhibitors and intermediates for making HIV-protease inhibitors
UA67727C2 (uk) * 1996-09-05 2004-07-15 Агурон Фармасевтікелс, Інк. Проміжні сполуки для одержання інгібіторів віл-протеази і способи одержання інгібіторів віл-протеази
DE19730602A1 (de) * 1997-07-17 1999-01-21 Clariant Gmbh 3-Acetoxy-2-methylbenzoesäurechlorid und ein Verfahren zu seiner Herstellung
US6084107A (en) * 1997-09-05 2000-07-04 Agouron Pharmaceuticals, Inc. Intermediates for making HIV-protease inhibitors
IN188157B (de) 1998-01-16 2002-08-24 Japan Tobacco Inc
US6403799B1 (en) 1999-10-21 2002-06-11 Agouron Pharmaceuticals, Inc. Methods for the preparation of intermediates in the synthesis of HIV-protease inhibitors
JP2006525307A (ja) 2003-05-08 2006-11-09 ファイザー インコーポレイテッド Ｈｉｖ−プロテアーゼ阻害剤の合成に有用な中間体及びその製造法
JPWO2005040099A1 (ja) * 2003-10-23 2007-03-08 小野薬品工業株式会社 ３−置換−（２ｒ，３ｒ）−２−保護されたアミノ−３−ヒドロキシプロピオン酸誘導体の製造方法およびその中間体
CN112409370B (zh) * 2020-12-10 2021-12-24 四川新迪医药化工有限公司 环氧侧链中间体的制备方法及环氧侧链中间体、钆布醇
CN115724849A (zh) * 2022-11-28 2023-03-03 安庆朗坤药业有限公司 一种4,4-二甲基-3,5,8-三氧杂双环[5.1.0]辛烷的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4110101A (en) * 1977-04-06 1978-08-29 Velsicol Chemical Corporation Dioxepane substituted amides
US4341756A (en) * 1980-01-31 1982-07-27 The Regents Of The University Of California Novel amino-dioxepane intermediates for the synthesis of new non-ionic contrast media
JPS56127373A (en) * 1980-01-31 1981-10-06 Univ California Novel amino-dioxepane intermediate for synthesizing novel nonionic contrast agent
MX9308016A (es) * 1992-12-22 1994-08-31 Lilly Co Eli Compuestos inhibidores de la proteasa del virus de la inmunodeficiencia humana, procedimiento para su preparacion y formulacion farmaceutica que los contiene.
US5484926A (en) * 1993-10-07 1996-01-16 Agouron Pharmaceuticals, Inc. HIV protease inhibitors

Also Published As

Publication number Publication date
JP3566968B2 (ja) 2004-09-15
EP0983999A1 (de) 2000-03-08
US20010021782A1 (en) 2001-09-13
ES2233976T3 (es) 2005-06-16
US6133461A (en) 2000-10-17
US6596903B2 (en) 2003-07-22
US6252085B1 (en) 2001-06-26
AU717637B2 (en) 2000-03-30
US6476232B2 (en) 2002-11-05
US6333416B2 (en) 2001-12-25
EP0983999B1 (de) 2005-02-09
US20030040633A1 (en) 2003-02-27
AU7002096A (en) 1997-04-17
US20020049337A1 (en) 2002-04-25
EP0983999A4 (de) 2002-09-11
PT983999E (pt) 2005-05-31
EP0983999B8 (de) 2005-06-08
DE69634345D1 (de) 2005-03-17
DE69634345T2 (de) 2006-03-02
WO1997011937A1 (fr) 1997-04-03

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