DE60018833D1 - Verfahren zur Synthese von Nukleosidanaloga - Google Patents

Verfahren zur Synthese von Nukleosidanaloga

Info

Publication number
DE60018833D1
DE60018833D1 DE60018833T DE60018833T DE60018833D1 DE 60018833 D1 DE60018833 D1 DE 60018833D1 DE 60018833 T DE60018833 T DE 60018833T DE 60018833 T DE60018833 T DE 60018833T DE 60018833 D1 DE60018833 D1 DE 60018833D1
Authority
DE
Germany
Prior art keywords
synthesis
nucleoside analogues
nucleoside
analogues
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60018833T
Other languages
German (de)
English (en)
Inventor
Robert William Scott
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Products Inc
Original Assignee
Pfizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Application granted granted Critical
Publication of DE60018833D1 publication Critical patent/DE60018833D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/14—Pyrrolo-pyrimidine radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • General Health & Medical Sciences (AREA)
  • Biotechnology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE60018833T 1999-05-11 2000-05-09 Verfahren zur Synthese von Nukleosidanaloga Expired - Lifetime DE60018833D1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13365199P 1999-05-11 1999-05-11

Publications (1)

Publication Number Publication Date
DE60018833D1 true DE60018833D1 (de) 2005-04-28

Family

ID=22459680

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60018833T Expired - Lifetime DE60018833D1 (de) 1999-05-11 2000-05-09 Verfahren zur Synthese von Nukleosidanaloga

Country Status (22)

Country Link
US (1) US6271370B1 (enExample)
EP (1) EP1052264B1 (enExample)
JP (1) JP2001011092A (enExample)
KR (1) KR100403900B1 (enExample)
CN (1) CN1275575A (enExample)
AR (1) AR028991A1 (enExample)
AT (1) ATE291582T1 (enExample)
AU (1) AU3401100A (enExample)
BR (1) BR0002089A (enExample)
CA (1) CA2307951A1 (enExample)
CZ (1) CZ20001710A3 (enExample)
DE (1) DE60018833D1 (enExample)
HU (1) HUP0001843A3 (enExample)
ID (1) ID25992A (enExample)
IL (1) IL136027A0 (enExample)
IN (1) IN186850B (enExample)
MX (1) MXPA00004532A (enExample)
PL (1) PL340109A1 (enExample)
RU (1) RU2200738C2 (enExample)
TR (1) TR200001340A2 (enExample)
YU (1) YU25500A (enExample)
ZA (1) ZA200002263B (enExample)

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Also Published As

Publication number Publication date
AU3401100A (en) 2000-11-16
YU25500A (sh) 2003-08-29
CZ20001710A3 (cs) 2001-09-12
EP1052264A2 (en) 2000-11-15
HUP0001843A2 (hu) 2001-06-28
ID25992A (id) 2000-11-16
BR0002089A (pt) 2001-01-02
EP1052264B1 (en) 2005-03-23
HU0001843D0 (en) 2000-07-28
MXPA00004532A (es) 2002-03-08
US6271370B1 (en) 2001-08-07
PL340109A1 (en) 2000-11-20
IN186850B (enExample) 2001-11-24
EP1052264A3 (en) 2001-06-13
CN1275575A (zh) 2000-12-06
HUP0001843A3 (en) 2001-09-28
ZA200002263B (en) 2001-12-24
IL136027A0 (en) 2001-05-20
AR028991A1 (es) 2003-06-04
KR20010069193A (ko) 2001-07-23
ATE291582T1 (de) 2005-04-15
CA2307951A1 (en) 2000-11-11
RU2200738C2 (ru) 2003-03-20
TR200001340A2 (tr) 2000-12-21
KR100403900B1 (ko) 2003-11-01
JP2001011092A (ja) 2001-01-16

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