DE60012028D1 - Zwischenprodukte für die herstellung von naphthyridin-3-carbonsäure-derivaten - Google Patents
Zwischenprodukte für die herstellung von naphthyridin-3-carbonsäure-derivatenInfo
- Publication number
- DE60012028D1 DE60012028D1 DE60012028T DE60012028T DE60012028D1 DE 60012028 D1 DE60012028 D1 DE 60012028D1 DE 60012028 T DE60012028 T DE 60012028T DE 60012028 T DE60012028 T DE 60012028T DE 60012028 D1 DE60012028 D1 DE 60012028D1
- Authority
- DE
- Germany
- Prior art keywords
- naphthyridine
- production
- acid derivatives
- carbonic acid
- intermediate products
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9920919.9A GB9920919D0 (en) | 1999-09-03 | 1999-09-03 | Novel compound |
| GB9920919 | 1999-09-03 | ||
| PCT/GB2000/003358 WO2001017961A2 (en) | 1999-09-03 | 2000-09-01 | Intermediates for the production of naphthyridine-3-carboxylic acid derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE60012028D1 true DE60012028D1 (de) | 2004-08-12 |
| DE60012028T2 DE60012028T2 (de) | 2005-08-18 |
Family
ID=10860355
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE60012028T Expired - Lifetime DE60012028T2 (de) | 1999-09-03 | 2000-09-01 | Intermediate für die Herstellung von Chinoloncarbonsäurederivaten |
Country Status (30)
| Country | Link |
|---|---|
| US (3) | US6703512B1 (de) |
| EP (1) | EP1212321B1 (de) |
| JP (1) | JP4208463B2 (de) |
| KR (1) | KR100705363B1 (de) |
| CN (1) | CN1255402C (de) |
| AR (1) | AR029452A1 (de) |
| AT (1) | ATE270671T1 (de) |
| AU (1) | AU773698B2 (de) |
| BR (1) | BRPI0013750B8 (de) |
| CA (1) | CA2383751C (de) |
| CO (1) | CO5180620A1 (de) |
| CZ (1) | CZ2002759A3 (de) |
| DE (1) | DE60012028T2 (de) |
| DK (1) | DK1212321T3 (de) |
| ES (1) | ES2223570T3 (de) |
| GB (1) | GB9920919D0 (de) |
| HK (1) | HK1046908B (de) |
| HU (1) | HU229391B1 (de) |
| IL (2) | IL148441A0 (de) |
| MX (1) | MXPA02002356A (de) |
| MY (1) | MY126789A (de) |
| NO (1) | NO322501B1 (de) |
| NZ (1) | NZ517601A (de) |
| PL (1) | PL206491B1 (de) |
| PT (1) | PT1212321E (de) |
| SI (1) | SI1212321T1 (de) |
| TR (1) | TR200200548T2 (de) |
| TW (1) | TWI264435B (de) |
| WO (1) | WO2001017961A2 (de) |
| ZA (1) | ZA200201779B (de) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2281817C (en) * | 1999-06-29 | 2008-07-29 | Smithkline Beecham Corporation | Methods of use of fluoroquinolone compounds against maxillary sinus pathogenic bacteria |
| GB9920919D0 (en) | 1999-09-03 | 1999-11-10 | Sb Pharmco Inc | Novel compound |
| GB9920917D0 (en) | 1999-09-03 | 1999-11-10 | Sb Pharmco Inc | Novel process |
| SI1412078T1 (sl) | 2001-08-02 | 2009-04-30 | Lg Life Sciences Ltd Lg Twin T | Postopki za pripravo amino-zaščitenih derivatov 4-aminometilen-pirolidin-3-ona, gemifloksacina ali njegove soli |
| KR100517638B1 (ko) | 2002-04-08 | 2005-09-28 | 주식회사 엘지생명과학 | 게미플록사신 산염의 새로운 제조방법 |
| EP1521809B1 (de) * | 2002-07-17 | 2005-11-23 | Ciba SC Holding AG | Oxidationsverfahren zur herstellung von chinacridonpigmenten |
| KR100653334B1 (ko) * | 2003-03-07 | 2006-12-04 | 주식회사 엘지생명과학 | 4-아미노메틸-3-알콕시이미노피롤리딘 메탄설폰산염의 신규한 제조 방법 |
| US8822934B2 (en) * | 2006-11-03 | 2014-09-02 | Accuray Incorporated | Collimator changer |
| CN104693088B (zh) * | 2013-12-06 | 2018-01-05 | 常州市勇毅生物药业有限公司 | 一种吉米沙星侧链的制备方法 |
Family Cites Families (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS57134482A (en) | 1981-02-13 | 1982-08-19 | Dainippon Pharmaceut Co Ltd | 1-ethyl-6-fluoro-1,4-dihydro-4-oxo-7-(1-piperazinyl)-1,8- naphthyridine-3-carboxylic acid-3/2 hydrate and its preparation |
| IN162769B (de) | 1984-11-13 | 1988-07-09 | Kyorin Seiyaku Kk | |
| NZ222047A (en) | 1986-10-08 | 1991-01-29 | Bristol Myers Co | Quinoline - or naphthyridine - carboxylic acid anti-bacterial agents |
| JPH01100165A (ja) | 1987-10-13 | 1989-04-18 | Shionogi & Co Ltd | オキシムまたはヒドロキシアミン誘導体系抗菌剤 |
| US4920120A (en) | 1988-01-25 | 1990-04-24 | Warner-Lambert Company | Antibacterial agents |
| JPH0356479A (ja) | 1989-07-24 | 1991-03-12 | Takeshi Yokota | 水溶性キノロン誘導体のｐ‐トルエンスルホン酸塩 |
| RU2049777C1 (ru) | 1989-08-16 | 1995-12-10 | Пфайзер Инк. | Азабицикло-хинолон-карбоновые кислоты или их фармацевтически приемлемые кислотно-аддитивные соли и промежуточные продукты для их получения |
| US5137892A (en) | 1990-12-12 | 1992-08-11 | Abbott Laboratories | Quinoline, naphthyridine and pyridobenzoxazine derivatives |
| EP0541086A1 (de) | 1991-11-08 | 1993-05-12 | Kaken Pharmaceutical Co., Ltd. | Antibakterielle 6-Fluoro-Chinolone mit einer Oximegruppe an dem Substituent in Position 7 |
| JPH0673056A (ja) | 1992-08-26 | 1994-03-15 | Kaken Pharmaceut Co Ltd | キノリンカルボン酸誘導体およびその塩 |
| US5776944A (en) | 1994-06-16 | 1998-07-07 | Lg Chemical Ltd. | 7-(4-aminomethyl-3-methyloxyiminopyrroplidin-1-yl)-1-cyclopropyl-6-flu oro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid and the process for the preparation thereof |
| DE69509442T2 (de) | 1994-06-16 | 1999-09-02 | Lg Chemical Ltd | Chinolincarbonsäurederivate mit 7-(4-Amino-methyl-3-oxim)-pyrrolidin-Substituenten und Verfahren zu ihrer Herstellung |
| JP3449658B2 (ja) | 1994-12-21 | 2003-09-22 | 杏林製薬株式会社 | 安定性に優れた８−アルコキシキノロンカルボン酸水和物並びにその製造方法 |
| DK0789697T3 (da) | 1995-06-06 | 1998-10-19 | Pfizer | Krystalform af vandfrit 7-([1alfa, 5alfa, 6alfa,]-6-amino-3-azabicyclo[3.1.0]hex-3-yl)-6-fluor-1-(2,4-difluorphenyl)-1,4-d |
| UA59341C2 (uk) | 1995-08-11 | 2003-09-15 | Пфайзер, Інк. | (1s,2s)-1-(4-гідроксифеніл)-2-(4-гідрокси-4-фенілпіперидин-1-іл)-1-пропанолметансульфонат тригідрат |
| UA49880C2 (uk) | 1996-03-29 | 2002-10-15 | Смітклайн Бічам Корпорейшн | Дигідрат ерпоcартану, фармацевтична композиція, спосіб отримання твердої дозованої форми, спосіб блокування рецепторів ангіотензину іі |
| MA24500A1 (fr) * | 1997-03-21 | 1998-10-01 | Lg Life Sciences Ltd | Derive du sel d'acide carboxylique de naphthyridine . |
| KR100286874B1 (ko) | 1998-03-04 | 2001-04-16 | 성재갑 | 보호된 4-아미노메틸-피롤리딘-3-온의 제조방법 |
| AU4211799A (en) | 1998-05-29 | 1999-12-13 | Pharmacia & Upjohn Company | 3-[(1--n-methylamino)ethyl-n-benzyl] pyrrolidine monomethanesulfonate |
| GB9820405D0 (en) | 1998-09-18 | 1998-11-11 | Smithkline Beecham Plc | Process |
| DK1223935T3 (da) | 1999-06-29 | 2008-02-04 | Lg Life Sciences Ltd | Anvendelse af gemifloxacinforbindelser mod bakterier |
| AU6947900A (en) | 1999-09-01 | 2001-03-26 | Smithkline Beecham Corporation | Methods of use of fluoroquinolone compounds against bacteria |
| GB9920917D0 (en) * | 1999-09-03 | 1999-11-10 | Sb Pharmco Inc | Novel process |
| GB9920919D0 (en) | 1999-09-03 | 1999-11-10 | Sb Pharmco Inc | Novel compound |
| WO2001021176A1 (en) | 1999-09-22 | 2001-03-29 | Smithkline Beecham Corporation | Methods of use of fluoroquinolone compounds against bacteria |
| KR20010091379A (ko) | 2000-03-15 | 2001-10-23 | 성재갑 | 7-(4-아미노메틸-3-옥심)피롤리딘 치환체를 갖는 퀴놀린카르복실산 유도체의 신규 제조방법 |
| KR20020018560A (ko) | 2000-09-01 | 2002-03-08 | 성재갑 | 3-아미노메틸-4-ｚ-메톡시이미노피롤리딘의 신규 제조방법 |
-
1999
- 1999-09-03 GB GBGB9920919.9A patent/GB9920919D0/en not_active Ceased
-
2000
- 2000-09-01 BR BRPI0013750A patent/BRPI0013750B8/pt not_active IP Right Cessation
- 2000-09-01 AU AU68573/00A patent/AU773698B2/en not_active Ceased
- 2000-09-01 CA CA2383751A patent/CA2383751C/en not_active Expired - Lifetime
- 2000-09-01 MY MYPI20004053 patent/MY126789A/en unknown
- 2000-09-01 CN CNB008123292A patent/CN1255402C/zh not_active Expired - Lifetime
- 2000-09-01 HU HU0202733A patent/HU229391B1/hu not_active IP Right Cessation
- 2000-09-01 TR TR2002/00548T patent/TR200200548T2/xx unknown
- 2000-09-01 PT PT00956706T patent/PT1212321E/pt unknown
- 2000-09-01 AR ARP000104596A patent/AR029452A1/es active IP Right Grant
- 2000-09-01 MX MXPA02002356A patent/MXPA02002356A/es active IP Right Grant
- 2000-09-01 DE DE60012028T patent/DE60012028T2/de not_active Expired - Lifetime
- 2000-09-01 EP EP00956706A patent/EP1212321B1/de not_active Expired - Lifetime
- 2000-09-01 WO PCT/GB2000/003358 patent/WO2001017961A2/en active IP Right Grant
- 2000-09-01 US US10/088,149 patent/US6703512B1/en not_active Expired - Lifetime
- 2000-09-01 IL IL14844100A patent/IL148441A0/xx active IP Right Grant
- 2000-09-01 NZ NZ517601A patent/NZ517601A/en not_active IP Right Cessation
- 2000-09-01 AT AT00956706T patent/ATE270671T1/de active
- 2000-09-01 CZ CZ2002759A patent/CZ2002759A3/cs unknown
- 2000-09-01 ES ES00956706T patent/ES2223570T3/es not_active Expired - Lifetime
- 2000-09-01 PL PL354725A patent/PL206491B1/pl not_active IP Right Cessation
- 2000-09-01 CO CO00065923A patent/CO5180620A1/es active IP Right Grant
- 2000-09-01 SI SI200030481T patent/SI1212321T1/xx unknown
- 2000-09-01 JP JP2001521708A patent/JP4208463B2/ja not_active Expired - Fee Related
- 2000-09-01 KR KR1020027002876A patent/KR100705363B1/ko active IP Right Grant
- 2000-09-01 DK DK00956706T patent/DK1212321T3/da active
- 2000-09-29 TW TW089120154A patent/TWI264435B/zh not_active IP Right Cessation
-
2002
- 2002-02-28 IL IL148441A patent/IL148441A/en unknown
- 2002-03-01 NO NO20021043A patent/NO322501B1/no not_active IP Right Cessation
- 2002-03-04 ZA ZA200201779A patent/ZA200201779B/xx unknown
- 2002-11-21 HK HK02108460.2A patent/HK1046908B/zh not_active IP Right Cessation
-
2003
- 2003-12-23 US US10/742,797 patent/US6803467B2/en not_active Expired - Lifetime
-
2004
- 2004-09-08 US US10/935,357 patent/US20050033064A1/en not_active Abandoned
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition |