DE60010918D1 - Verfahren zur herstellung von 7-azabicyclo (4.1.0)-hept-3-ene-3-carbonsäureestern - Google Patents

Verfahren zur herstellung von 7-azabicyclo (4.1.0)-hept-3-ene-3-carbonsäureestern

Info

Publication number
DE60010918D1
DE60010918D1 DE60010918T DE60010918T DE60010918D1 DE 60010918 D1 DE60010918 D1 DE 60010918D1 DE 60010918 T DE60010918 T DE 60010918T DE 60010918 T DE60010918 T DE 60010918T DE 60010918 D1 DE60010918 D1 DE 60010918D1
Authority
DE
Germany
Prior art keywords
ene
azabicyclohept
producing
azabicyclo
hept
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60010918T
Other languages
English (en)
Other versions
DE60010918T2 (de
Inventor
Shiro Terashima
Katsuji Ujita
Akihiro Ishiwata
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kuraray Co Ltd
Sagami Chemical Research Institute
Original Assignee
Kuraray Co Ltd
Sagami Chemical Research Institute
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kuraray Co Ltd, Sagami Chemical Research Institute filed Critical Kuraray Co Ltd
Publication of DE60010918D1 publication Critical patent/DE60010918D1/de
Application granted granted Critical
Publication of DE60010918T2 publication Critical patent/DE60010918T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/04Formation of amino groups in compounds containing carboxyl groups
    • C07C227/06Formation of amino groups in compounds containing carboxyl groups by addition or substitution reactions, without increasing the number of carbon atoms in the carbon skeleton of the acid
    • C07C227/08Formation of amino groups in compounds containing carboxyl groups by addition or substitution reactions, without increasing the number of carbon atoms in the carbon skeleton of the acid by reaction of ammonia or amines with acids containing functional groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/52Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
    • C07C229/54Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C229/64Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring the carbon skeleton being further substituted by singly-bound oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D203/00Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D203/02Preparation by ring-closure
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D203/00Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D203/26Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Indole Compounds (AREA)
DE60010918T 1999-11-02 2000-10-27 Verfahren zur herstellung von 7-azabicyclo (4.1.0)-hept-3-ene-3-carbonsäureestern Expired - Fee Related DE60010918T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP31261699A JP2001131144A (ja) 1999-11-02 1999-11-02 7−アザビシクロ[4.1.0]ヘプト−3−エン−3−カルボン酸エステル類の製造方法
JP31261699 1999-11-02
PCT/JP2000/007578 WO2001032617A1 (fr) 1999-11-02 2000-10-27 Elaboration d'esters d'acide 7-azabicyclo[4.1.0]-hept-3-ene-3-carboxylique

Publications (2)

Publication Number Publication Date
DE60010918D1 true DE60010918D1 (de) 2004-06-24
DE60010918T2 DE60010918T2 (de) 2005-05-25

Family

ID=18031355

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60010918T Expired - Fee Related DE60010918T2 (de) 1999-11-02 2000-10-27 Verfahren zur herstellung von 7-azabicyclo (4.1.0)-hept-3-ene-3-carbonsäureestern

Country Status (8)

Country Link
US (1) US6790964B1 (de)
EP (1) EP1229022B1 (de)
JP (1) JP2001131144A (de)
CN (1) CN1420866A (de)
AT (1) ATE267167T1 (de)
AU (1) AU7961700A (de)
DE (1) DE60010918T2 (de)
WO (1) WO2001032617A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011021223A2 (en) * 2009-08-19 2011-02-24 Msn Laboratories Limited Novel salts of ethyl (3r, 4s, 5r)-4,5-imino-3-(l-ethylpropoxy)-1- cvclohexene-1-carboxylate and its use
CN104370762A (zh) * 2014-11-13 2015-02-25 中科院广州化学有限公司 一种微波合成烷基芳基胺类化合物的方法
CN104557653A (zh) * 2014-12-31 2015-04-29 大连联化化学有限公司 7-甲基-氮杂-二环[4,1,0]庚烷的制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE759917T1 (de) * 1995-02-27 1998-10-22 Gilead Sciences Inc Neue selektive inhibitoren viraler oder bakterieller neuraminidasen
US5866601A (en) 1995-02-27 1999-02-02 Gilead Sciences, Inc. Carbocyclic compounds
US5763483A (en) * 1995-12-29 1998-06-09 Gilead Sciences, Inc. Carbocyclic compounds
EP0920410B1 (de) 1996-08-23 2002-03-27 Gilead Sciences, Inc. Verfahren zur herstellung von cyclohexen-carboxylatderivate
JPH10231280A (ja) 1996-12-20 1998-09-02 Sagami Chem Res Center 3−アミノ−2−ヒドロキシ−4−フェニルブチロニトリル誘導体の製造方法
TR200000723T2 (tr) * 1997-09-17 2001-06-21 Gilead Sciences, Inc. Altı elemanlı halkalar ihtiva eden bileşikler ve ilaç olarak kullanımları.
DE60002949T2 (de) * 1999-06-11 2004-05-19 F. Hoffmann-La Roche Ag Verfahren zur Herstellung des Neuraminidase-Inhibitoren ro-64-0796

Also Published As

Publication number Publication date
EP1229022B1 (de) 2004-05-19
US6790964B1 (en) 2004-09-14
CN1420866A (zh) 2003-05-28
EP1229022A4 (de) 2002-11-27
EP1229022A1 (de) 2002-08-07
JP2001131144A (ja) 2001-05-15
AU7961700A (en) 2001-05-14
WO2001032617A1 (fr) 2001-05-10
ATE267167T1 (de) 2004-06-15
DE60010918T2 (de) 2005-05-25

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee