ATE267167T1 - Verfahren zur herstellung von 7-azabicyclo (4.1.0)-hept-3-ene-3-carbonsäureestern - Google Patents
Verfahren zur herstellung von 7-azabicyclo (4.1.0)-hept-3-ene-3-carbonsäureesternInfo
- Publication number
- ATE267167T1 ATE267167T1 AT00970163T AT00970163T ATE267167T1 AT E267167 T1 ATE267167 T1 AT E267167T1 AT 00970163 T AT00970163 T AT 00970163T AT 00970163 T AT00970163 T AT 00970163T AT E267167 T1 ATE267167 T1 AT E267167T1
- Authority
- AT
- Austria
- Prior art keywords
- ene
- azabicyclohept
- producing
- azabicyclo
- hept
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 1
- 239000002841 Lewis acid Substances 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000002118 epoxides Chemical class 0.000 abstract 1
- 150000007517 lewis acids Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/04—Formation of amino groups in compounds containing carboxyl groups
- C07C227/06—Formation of amino groups in compounds containing carboxyl groups by addition or substitution reactions, without increasing the number of carbon atoms in the carbon skeleton of the acid
- C07C227/08—Formation of amino groups in compounds containing carboxyl groups by addition or substitution reactions, without increasing the number of carbon atoms in the carbon skeleton of the acid by reaction of ammonia or amines with acids containing functional groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/52—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
- C07C229/54—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring
- C07C229/64—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring the carbon skeleton being further substituted by singly-bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D203/00—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
- C07D203/02—Preparation by ring-closure
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D203/00—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
- C07D203/26—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP31261699A JP2001131144A (ja) | 1999-11-02 | 1999-11-02 | ７−アザビシクロ［４．１．０］ヘプト−３−エン−３−カルボン酸エステル類の製造方法 |
| PCT/JP2000/007578 WO2001032617A1 (en) | 1999-11-02 | 2000-10-27 | Process for the preparation of 7-azabicyclo[4.1.0]-hept-3-ene-3-carboxylic acid esters |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE267167T1 true ATE267167T1 (de) | 2004-06-15 |
Family
ID=18031355
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT00970163T ATE267167T1 (de) | 1999-11-02 | 2000-10-27 | Verfahren zur herstellung von 7-azabicyclo (4.1.0)-hept-3-ene-3-carbonsäureestern |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US6790964B1 (de) |
| EP (1) | EP1229022B1 (de) |
| JP (1) | JP2001131144A (de) |
| CN (1) | CN1420866A (de) |
| AT (1) | ATE267167T1 (de) |
| AU (1) | AU7961700A (de) |
| DE (1) | DE60010918T2 (de) |
| WO (1) | WO2001032617A1 (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011021223A2 (en) * | 2009-08-19 | 2011-02-24 | Msn Laboratories Limited | Novel salts of ethyl (3r, 4s, 5r)-4,5-imino-3-(l-ethylpropoxy)-1- cvclohexene-1-carboxylate and its use |
| CN104370762A (zh) * | 2014-11-13 | 2015-02-25 | 中科院广州化学有限公司 | 一种微波合成烷基芳基胺类化合物的方法 |
| CN104557653A (zh) * | 2014-12-31 | 2015-04-29 | 大连联化化学有限公司 | 7-甲基-氮杂-二环[4,1,0]庚烷的制备方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN100409844C (zh) * | 1995-02-27 | 2008-08-13 | 吉里德科学公司 | 神经氨酸苷酶抑制剂 |
| US5866601A (en) | 1995-02-27 | 1999-02-02 | Gilead Sciences, Inc. | Carbocyclic compounds |
| US5763483A (en) | 1995-12-29 | 1998-06-09 | Gilead Sciences, Inc. | Carbocyclic compounds |
| ATE215062T1 (de) | 1996-08-23 | 2002-04-15 | Gilead Sciences Inc | Verfahren zur herstellung von cyclohexen- carboxylatderivate |
| JPH10231280A (ja) | 1996-12-20 | 1998-09-02 | Sagami Chem Res Center | ３−アミノ−２−ヒドロキシ−４−フェニルブチロニトリル誘導体の製造方法 |
| NZ502988A (en) * | 1997-09-17 | 2002-08-28 | Gilead Sciences Inc | 5-Acetamido-4-amino-2-propionyloxy-6-isopropoxy-1-cyclohexene useful for treating influenza |
| DK1059283T3 (da) * | 1999-06-11 | 2003-09-15 | Hoffmann La Roche | Fremgangsmåde til fremstilling af neuraminidase-inhibitor ro-64-0796 |
-
1999
- 1999-11-02 JP JP31261699A patent/JP2001131144A/ja active Pending
-
2000
- 2000-10-27 CN CN00818117A patent/CN1420866A/zh active Pending
- 2000-10-27 AT AT00970163T patent/ATE267167T1/de not_active IP Right Cessation
- 2000-10-27 US US10/111,910 patent/US6790964B1/en not_active Expired - Fee Related
- 2000-10-27 EP EP00970163A patent/EP1229022B1/de not_active Expired - Lifetime
- 2000-10-27 DE DE60010918T patent/DE60010918T2/de not_active Expired - Fee Related
- 2000-10-27 WO PCT/JP2000/007578 patent/WO2001032617A1/ja not_active Ceased
- 2000-10-27 AU AU79617/00A patent/AU7961700A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN1420866A (zh) | 2003-05-28 |
| WO2001032617A1 (en) | 2001-05-10 |
| EP1229022B1 (de) | 2004-05-19 |
| DE60010918D1 (de) | 2004-06-24 |
| US6790964B1 (en) | 2004-09-14 |
| EP1229022A4 (de) | 2002-11-27 |
| EP1229022A1 (de) | 2002-08-07 |
| DE60010918T2 (de) | 2005-05-25 |
| JP2001131144A (ja) | 2001-05-15 |
| AU7961700A (en) | 2001-05-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |