DE60001835D1 - Mesalazine enthaltende pharmazeutische zusammensetzungen mit gesteuerte freisetzung - Google Patents

Mesalazine enthaltende pharmazeutische zusammensetzungen mit gesteuerte freisetzung

Info

Publication number
DE60001835D1
DE60001835D1 DE60001835T DE60001835T DE60001835D1 DE 60001835 D1 DE60001835 D1 DE 60001835D1 DE 60001835 T DE60001835 T DE 60001835T DE 60001835 T DE60001835 T DE 60001835T DE 60001835 D1 DE60001835 D1 DE 60001835D1
Authority
DE
Germany
Prior art keywords
pharmaceutical compositions
mesalazine
controlled release
containing pharmaceutical
active ingredient
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60001835T
Other languages
English (en)
Other versions
DE60001835T2 (de
Inventor
Roberto Villa
Massimo Pedrani
Mauro Ajani
Lorenzo Fossati
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Cosmo Technologies Ltd
Original Assignee
Cosmo SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=11383159&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE60001835(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Cosmo SpA filed Critical Cosmo SpA
Application granted granted Critical
Publication of DE60001835D1 publication Critical patent/DE60001835D1/de
Publication of DE60001835T2 publication Critical patent/DE60001835T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/60—Salicylic acid; Derivatives thereof
    • A61K31/606—Salicylic acid; Derivatives thereof having amino groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846—Poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE60001835T 1999-06-14 2000-06-08 Mesalazine enthaltende pharmazeutische zusammensetzungen mit gesteuerte freisetzung Expired - Lifetime DE60001835T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT1999MI001316A ITMI991316A1 (it) 1999-06-14 1999-06-14 Composizioni farmaceutiche orali a rilascio modificato di mesalazina
PCT/EP2000/005321 WO2000076481A1 (en) 1999-06-14 2000-06-08 Mesalazine controlled release oral pharmaceutical compositions

Publications (2)

Publication Number Publication Date
DE60001835D1 true DE60001835D1 (de) 2003-04-30
DE60001835T2 DE60001835T2 (de) 2003-11-13

Family

ID=11383159

Family Applications (2)

Application Number Title Priority Date Filing Date
DE60001835T Expired - Lifetime DE60001835T2 (de) 1999-06-14 2000-06-08 Mesalazine enthaltende pharmazeutische zusammensetzungen mit gesteuerte freisetzung
DE60027608T Expired - Lifetime DE60027608T2 (de) 1999-06-14 2000-06-08 Mesalazine enthaltende pharmazeutische Zusammensetzungen mit gesteuerter Freisetzung

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE60027608T Expired - Lifetime DE60027608T2 (de) 1999-06-14 2000-06-08 Mesalazine enthaltende pharmazeutische Zusammensetzungen mit gesteuerter Freisetzung

Country Status (18)

Country Link
US (1) US6773720B1 (de)
EP (2) EP1287822B1 (de)
JP (2) JP4727875B2 (de)
CN (2) CN100448448C (de)
AT (2) ATE235234T1 (de)
AU (1) AU5077200A (de)
CA (1) CA2377299C (de)
DE (2) DE60001835T2 (de)
DK (2) DK1198226T3 (de)
ES (2) ES2194732T3 (de)
HK (2) HK1046247B (de)
IT (1) ITMI991316A1 (de)
MX (1) MXPA01012888A (de)
NO (1) NO329402B1 (de)
PT (2) PT1198226E (de)
RU (1) RU2245148C2 (de)
TR (1) TR200200561T2 (de)
WO (1) WO2000076481A1 (de)

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US8895064B2 (en) 1999-06-14 2014-11-25 Cosmo Technologies Limited Controlled release and taste masking oral pharmaceutical composition
DK1183014T3 (da) 1999-06-14 2004-02-09 Cosmo Spa Smagsmaskerede orale farmaceutiske sammensætninger med kontrolleret frigivelse
CA2359812C (en) 2000-11-20 2004-02-10 The Procter & Gamble Company Pharmaceutical dosage form with multiple coatings for reduced impact of coating fractures
AR036797A1 (es) 2001-10-15 2004-10-06 Ferring Bv Un metodo para preparar una composicion farmaceutica que comprende acido 5-aminosalicilico para utilizar en el tratamiento de colitis ulcerosa y enfermedades de crohn
ITMI20012599A1 (it) * 2001-12-11 2003-06-11 Cosmo Spa Composizioni farmaceutiche per la somministrazione orale di eparina osuoi derivati, utili per la terapia di malattie infiammatorie dell'int
US9308220B2 (en) 2001-12-11 2016-04-12 Cosmo Technologies Limited Pharmaceutical compositions for the oral administration of heparin or derivatives thereof
US20030118329A1 (en) * 2001-12-21 2003-06-26 Pere Obrador Video indexing using high resolution still images
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FR2852843B1 (fr) 2003-03-24 2008-05-23 Karim Ioualalen Systeme galenique permettant le masquage du gout
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US7825106B2 (en) 2003-09-03 2010-11-02 Agi Therapeutics Ltd. Modified release formulations and methods of treating inflammatory bowel disease
US7737133B2 (en) 2003-09-03 2010-06-15 Agi Therapeutics Ltd. Formulations and methods of treating inflammatory bowel disease
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US8497258B2 (en) 2005-11-12 2013-07-30 The Regents Of The University Of California Viscous budesonide for the treatment of inflammatory diseases of the gastrointestinal tract
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WO2011045775A1 (en) 2009-10-16 2011-04-21 Ranbaxy Laboratories Limited A delayed release pharmaceutical composition of mesalamine
IT1398643B1 (it) 2010-03-04 2013-03-08 Cosmo Technologies Ltd Composizione solida per la somministrazione orale di coloranti, e utilizzo diagnostico della stessa
EP2425826A1 (de) * 2010-09-01 2012-03-07 Disphar International B.V. Mesalazin-Tablette mit verbesserter Auflösung
IT1402047B1 (it) * 2010-10-19 2013-08-28 Cross Pharma Sa Uso del mexiprostil nel trattamento delle malattie infiammatorie intestinali
EP2468264A1 (de) 2010-12-27 2012-06-27 Laboratorios Liconsa, S.A. Orale pharmazeutische Tablette zur gesteuerten Abgabe von Mesalazin und Verfahren zu deren Erhalt
SG10201607085WA (en) 2011-01-07 2016-10-28 Elcelyx Therapeutics Inc Chemosensory Receptor Ligand-Based Therapies
US9795792B2 (en) 2011-02-25 2017-10-24 Medtronic, Inc. Emergency mode switching for non-pacing modes
US10154964B2 (en) 2011-09-07 2018-12-18 Cosmo Technologies Limited Controlled release and taste masking oral pharmaceutical composition
JP6175074B2 (ja) 2012-01-06 2017-08-02 エルセリクス セラピューティクス インコーポレイテッド 代謝障害を治療するための組成物および方法
BR112014016808B1 (pt) 2012-01-06 2022-01-11 Anji Pharma (Us) Llc Uso de um composto de biguanida para a fabricação de um medicamento para baixar os níveis de glicose no sangue e para o tratamento de um distúrbio do metabolismo de glicose
EP2822542A1 (de) * 2012-03-07 2015-01-14 Santarus, Inc. Gesteuerte freisetzung fester dosierungsformen von mesalamin
US20150164920A1 (en) 2012-03-30 2015-06-18 Laboratorios Del Dr. Esteve S.A. Controlled release formulation comprising mesalamine
WO2013158928A2 (en) 2012-04-18 2013-10-24 Elcelyx Therapeutics, Inc. Chemosensory receptor ligand-based therapies
EP2872127A1 (de) 2012-07-11 2015-05-20 Elcelyx Therapeutics, Inc. Zusammensetzungen mit statinen, biguaniden und weiteren mitteln zur verringerung des herz-kreislauf-risikos
EP2722058A1 (de) 2012-10-19 2014-04-23 Cosmo Technologies Ltd Orale Feststoffzusammensetzung mit Farbstoffen für die Verwendung bei der endoskopischen Diagnose
CA2896864C (en) 2013-01-05 2021-04-20 Elcelyx Therapeutics, Inc. Delayed-release composition comprising biguanide
LT2959892T (lt) * 2013-02-22 2020-12-10 Zeria Pharmaceutical Co., Ltd. Enterine danga padengta tabletė
US9539265B2 (en) 2013-03-15 2017-01-10 Aihol Corporation Pharmaceutical formulation containing glycosaminoglycan
EP2953619A1 (de) 2013-03-15 2015-12-16 Warner Chilcott Company, LLC Pharmazeutische mesalaminzusammensetzung mit mehrfachdosierungselemente für reduzierte abgabevariabilität
CN104922090B (zh) * 2015-07-03 2017-11-14 湖南方盛制药股份有限公司 美沙拉秦肠溶缓释微丸
EP3162362A1 (de) 2015-10-30 2017-05-03 Dr. Falk Pharma Gmbh Optimierte mesalazinhaltige hochdosistablette
ITUA20162293A1 (it) 2016-04-05 2017-10-05 Sofar Spa Processo per formulazioni solide di mesalazina
US20180147301A1 (en) 2016-11-28 2018-05-31 Cosmo Technologies Ltd. Solid oral composition containing dyes
US10098898B1 (en) 2017-12-04 2018-10-16 Handa Pharmaceuticals, Llc Release stable mesalamine dosage forms
EP3501503A1 (de) * 2017-12-22 2019-06-26 Cosmo Technologies Ltd. Feste verabreichungszusammensetzung
EP3662895A1 (de) 2018-12-07 2020-06-10 Tillotts Pharma AG Verfahren zur herstellung von reduzierenden zuckerfreien 5-asa-tablettenkernen
IT201800011120A1 (it) 2018-12-14 2020-06-14 Dpl Pharma S P A Composizioni farmaceutiche orali solide per la somministrazione di mesalazina o suoi derivati
CN112587506A (zh) * 2020-12-09 2021-04-02 南京森博医药研发有限公司 一种用于制备美沙拉嗪肠溶缓释胶囊的方法

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Also Published As

Publication number Publication date
EP1198226A1 (de) 2002-04-24
DK1287822T3 (da) 2006-08-28
ITMI991316A1 (it) 2000-12-14
HK1085669A1 (en) 2006-09-01
HK1046247B (zh) 2006-04-07
ATE235234T1 (de) 2003-04-15
DE60001835T2 (de) 2003-11-13
PT1198226E (pt) 2003-07-31
JP5235839B2 (ja) 2013-07-10
DE60027608T2 (de) 2007-04-26
ES2262749T3 (es) 2006-12-01
NO20016107D0 (no) 2001-12-14
DK1198226T3 (da) 2003-07-21
CN1355694A (zh) 2002-06-26
CN1720919A (zh) 2006-01-18
ES2194732T3 (es) 2003-12-01
HK1046247A1 (en) 2003-01-03
DE60027608D1 (de) 2006-06-01
NO20016107L (no) 2002-02-11
CA2377299C (en) 2009-05-12
EP1198226B1 (de) 2003-03-26
JP2010024241A (ja) 2010-02-04
CN100448448C (zh) 2009-01-07
WO2000076481A1 (en) 2000-12-21
US6773720B1 (en) 2004-08-10
TR200200561T2 (tr) 2002-06-21
JP2003501458A (ja) 2003-01-14
CA2377299A1 (en) 2000-12-21
EP1287822A2 (de) 2003-03-05
EP1287822B1 (de) 2006-04-26
MXPA01012888A (es) 2002-07-30
CN1217665C (zh) 2005-09-07
JP4727875B2 (ja) 2011-07-20
PT1287822E (pt) 2006-07-31
RU2245148C2 (ru) 2005-01-27
NO329402B1 (no) 2010-10-11
ATE324104T1 (de) 2006-05-15
ITMI991316A0 (it) 1999-06-14
EP1287822A3 (de) 2003-03-19
AU5077200A (en) 2001-01-02

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Legal Events

Date Code Title Description
8327 Change in the person/name/address of the patent owner

Owner name: COSMO S.P.A., LAINATE, MILANO, IT

8364 No opposition during term of opposition
8327 Change in the person/name/address of the patent owner

Owner name: COSMO TECHNOLOGIES LIMITED, BRAY, WICKLOW, IE