DE4400464A1 - Endoparasitizide Mittel - Google Patents

Endoparasitizide Mittel

Info

Publication number
DE4400464A1
DE4400464A1 DE4400464A DE4400464A DE4400464A1 DE 4400464 A1 DE4400464 A1 DE 4400464A1 DE 4400464 A DE4400464 A DE 4400464A DE 4400464 A DE4400464 A DE 4400464A DE 4400464 A1 DE4400464 A1 DE 4400464A1
Authority
DE
Germany
Prior art keywords
spp
alkyl
methyl
formula
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
DE4400464A
Other languages
German (de)
English (en)
Inventor
Norbert Dr Mencke
Achim Dr Dr Harder
Peter Dr Jeschke
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Priority to DE4400464A priority Critical patent/DE4400464A1/de
Priority to TW083111751A priority patent/TW364850B/zh
Priority to AU81592/94A priority patent/AU685535B2/en
Priority to ES94120772T priority patent/ES2168285T3/es
Priority to EP94120772A priority patent/EP0662326B1/de
Priority to DE1994509977 priority patent/DE122006000001I2/de
Priority to AT94120772T priority patent/ATE209501T1/de
Priority to PT94120772T priority patent/PT662326E/pt
Priority to DE59409977T priority patent/DE59409977D1/de
Priority to DK94120772T priority patent/DK0662326T5/da
Priority to US08/368,515 priority patent/US5589503A/en
Priority to CA002139725A priority patent/CA2139725C/en
Priority to NZ270300A priority patent/NZ270300A/en
Priority to PL95306709A priority patent/PL180019B1/pl
Priority to JP01633595A priority patent/JP4033920B2/ja
Priority to FI950091A priority patent/FI116885B/fi
Priority to IL11228595A priority patent/IL112285A/xx
Priority to KR1019950000274A priority patent/KR100359618B1/ko
Priority to PH49754A priority patent/PH31462A/en
Priority to SK31-95A priority patent/SK283367B6/sk
Priority to ZA95136A priority patent/ZA95136B/xx
Priority to UA95018024A priority patent/UA41327C2/uk
Priority to HU9500065A priority patent/HU226207B1/hu
Priority to CZ199561A priority patent/CZ290246B6/cs
Priority to NO950093A priority patent/NO307030B1/no
Priority to RU95100759/13A priority patent/RU2124364C1/ru
Priority to CNB951011588A priority patent/CN1165338C/zh
Publication of DE4400464A1 publication Critical patent/DE4400464A1/de
Priority to NL300218C priority patent/NL300218I2/nl
Priority to FR06C0002C priority patent/FR06C0002I2/fr
Priority to NO2006001C priority patent/NO2006001I2/no
Priority to JP2007228858A priority patent/JP2007314580A/ja
Withdrawn legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15—Depsipeptides; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08—Peptides having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N33/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic nitrogen compounds
    • A01N33/02—Amines; Quaternary ammonium compounds
    • A01N33/04—Nitrogen directly attached to aliphatic or cycloaliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Luminescent Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Peptides Or Proteins (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Compositions Of Oxide Ceramics (AREA)
  • Cosmetics (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DE4400464A 1994-01-11 1994-01-11 Endoparasitizide Mittel Withdrawn DE4400464A1 (de)

Priority Applications (31)

Application Number Priority Date Filing Date Title
DE4400464A DE4400464A1 (de) 1994-01-11 1994-01-11 Endoparasitizide Mittel
TW083111751A TW364850B (en) 1994-01-11 1994-12-16 Nematocidal compositions
AU81592/94A AU685535B2 (en) 1994-01-11 1994-12-20 Endoparasiticidal compositions
ES94120772T ES2168285T3 (es) 1994-01-11 1994-12-27 Agentes endoparasiticidas que contienen praziquantel y epsiprantel.
EP94120772A EP0662326B1 (de) 1994-01-11 1994-12-27 Endoparasitizide Mittel die Praziquantel und Epsiprantel enthalten
DE1994509977 DE122006000001I2 (de) 1994-01-11 1994-12-27 Endoparasitizide Mittel die Praziquantel und Epsiprantel enthalten
AT94120772T ATE209501T1 (de) 1994-01-11 1994-12-27 Endoparasitizide mittel die praziquantel und epsiprantel enthalten
PT94120772T PT662326E (pt) 1994-01-11 1994-12-27 Agentes endoparasiticidas que contem praziquantel e epsiprantel
DE59409977T DE59409977D1 (de) 1994-01-11 1994-12-27 Endoparasitizide Mittel die Praziquantel und Epsiprantel enthalten
DK94120772T DK0662326T5 (da) 1994-01-11 1994-12-27 Endoparasiticide midler indeholdende praziquantel og epsiprantel
US08/368,515 US5589503A (en) 1994-01-11 1995-01-04 Endoparasiticidal compositions
CA002139725A CA2139725C (en) 1994-01-11 1995-01-06 Endoparasiticidal compositions
NZ270300A NZ270300A (en) 1994-01-11 1995-01-06 Endoparasiticidal compositions containing praziquantel and epsiprantel together with certain cyclic depsipeptides
FI950091A FI116885B (fi) 1994-01-11 1995-01-09 Endoparasiitteja tappavat aineet
JP01633595A JP4033920B2 (ja) 1994-01-11 1995-01-09 内寄生性生物防除剤である組成物
PL95306709A PL180019B1 (pl) 1994-01-11 1995-01-09 Srodek do zwalczania pasozytów wewnetrznych i sposób wytwarzania srodka do zwalczania pasozytów wewnetrznych PL PL PL PL PL PL PL PL PL PL PL
IL11228595A IL112285A (en) 1994-01-11 1995-01-09 Endoparasiticidal compositions containing praziquantel epsiprantel and cyclic depsipeptides
KR1019950000274A KR100359618B1 (ko) 1994-01-11 1995-01-09 내부기생충구제제조성물
PH49754A PH31462A (en) 1994-01-11 1995-01-09 Endoparasiticidal compositions.
HU9500065A HU226207B1 (en) 1994-01-11 1995-01-10 Endoparaziticide compositions
ZA95136A ZA95136B (en) 1994-01-11 1995-01-10 Endoparasiticidal compositions
UA95018024A UA41327C2 (uk) 1994-01-11 1995-01-10 Ендопаразитицидний засіб
SK31-95A SK283367B6 (sk) 1994-01-11 1995-01-10 Endoparaziticídne prostriedky a ich použitie
CZ199561A CZ290246B6 (cs) 1994-01-11 1995-01-10 Endoparasiticidní prostředky a jejich pouľití
NO950093A NO307030B1 (no) 1994-01-11 1995-01-10 Endoparasittmiddel samt anvendelse av praziquantel eller epsiprantel sammen med cykliske depsipeptider
CNB951011588A CN1165338C (zh) 1994-01-11 1995-01-11 杀体内寄生虫组合物
RU95100759/13A RU2124364C1 (ru) 1994-01-11 1995-01-11 Эндопаразитицидное средство
NL300218C NL300218I2 (nl) 1994-01-11 2006-01-26 Endoparasiticide middelen die prziquantel en spsiprantel bevatten.
FR06C0002C FR06C0002I2 (en:Method) 1994-01-11 2006-01-26
NO2006001C NO2006001I2 (no) 1994-01-11 2006-01-27 Emodepsid/prazikvantel
JP2007228858A JP2007314580A (ja) 1994-01-11 2007-09-04 内寄生性生物防除剤である組成物

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4400464A DE4400464A1 (de) 1994-01-11 1994-01-11 Endoparasitizide Mittel

Publications (1)

Publication Number Publication Date
DE4400464A1 true DE4400464A1 (de) 1995-07-13

Family

ID=6507651

Family Applications (3)

Application Number Title Priority Date Filing Date
DE4400464A Withdrawn DE4400464A1 (de) 1994-01-11 1994-01-11 Endoparasitizide Mittel
DE1994509977 Active DE122006000001I2 (de) 1994-01-11 1994-12-27 Endoparasitizide Mittel die Praziquantel und Epsiprantel enthalten
DE59409977T Expired - Lifetime DE59409977D1 (de) 1994-01-11 1994-12-27 Endoparasitizide Mittel die Praziquantel und Epsiprantel enthalten

Family Applications After (2)

Application Number Title Priority Date Filing Date
DE1994509977 Active DE122006000001I2 (de) 1994-01-11 1994-12-27 Endoparasitizide Mittel die Praziquantel und Epsiprantel enthalten
DE59409977T Expired - Lifetime DE59409977D1 (de) 1994-01-11 1994-12-27 Endoparasitizide Mittel die Praziquantel und Epsiprantel enthalten

Country Status (27)

Country Link
US (1) US5589503A (en:Method)
EP (1) EP0662326B1 (en:Method)
JP (2) JP4033920B2 (en:Method)
KR (1) KR100359618B1 (en:Method)
CN (1) CN1165338C (en:Method)
AT (1) ATE209501T1 (en:Method)
AU (1) AU685535B2 (en:Method)
CA (1) CA2139725C (en:Method)
CZ (1) CZ290246B6 (en:Method)
DE (3) DE4400464A1 (en:Method)
DK (1) DK0662326T5 (en:Method)
ES (1) ES2168285T3 (en:Method)
FI (1) FI116885B (en:Method)
FR (1) FR06C0002I2 (en:Method)
HU (1) HU226207B1 (en:Method)
IL (1) IL112285A (en:Method)
NL (1) NL300218I2 (en:Method)
NO (2) NO307030B1 (en:Method)
NZ (1) NZ270300A (en:Method)
PH (1) PH31462A (en:Method)
PL (1) PL180019B1 (en:Method)
PT (1) PT662326E (en:Method)
RU (1) RU2124364C1 (en:Method)
SK (1) SK283367B6 (en:Method)
TW (1) TW364850B (en:Method)
UA (1) UA41327C2 (en:Method)
ZA (1) ZA95136B (en:Method)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005055973A3 (de) * 2003-12-13 2005-08-11 Bayer Healthcare Ag Endoparasitizide mittel zur topischen applikation

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
DE19520275A1 (de) * 1995-06-02 1996-12-05 Bayer Ag Endoparasitizide Mittel
HUP0004132A3 (en) * 1997-10-20 2006-06-28 Dainippon Sumitomo Pharma Co Rapidly soluble drug composition
DE19921887A1 (de) * 1999-05-12 2000-11-16 Bayer Ag Endoparasitizide Mittel
DE10008128A1 (de) * 2000-02-22 2001-08-23 Bayer Ag Endoparasitizide Mittel
KR100358084B1 (ko) * 2000-10-04 2002-10-25 주식회사대성미생물연구소 프라지콴텔과 시메티딘 합제를 이용한 어류의아가미흡충증 치료방법
DE10104362A1 (de) * 2001-02-01 2002-08-08 Bayer Ag Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit
CN100509734C (zh) * 2001-06-28 2009-07-08 日本瑞翁株式会社 含环烷基烷基醚的溶剂及其制备方法
ES2439725T3 (es) * 2001-10-05 2014-01-24 Rubicon Scientific Llc Piensos para animales que incluyen principios activos
DE10359798A1 (de) 2003-12-19 2005-07-21 Bayer Healthcare Ag Cyclohexadepsipeptide zur Bekämpfung von Endoparasiten und ein Verfahren zu ihrer Herstellung
DE102004055316A1 (de) * 2004-11-16 2006-05-18 Bayer Healthcare Ag Verhinderung vertikaler Endoparasiten-Infektionen
DE102005011779A1 (de) * 2005-03-11 2006-09-14 Bayer Healthcare Ag Endoparasitizide Mittel
BRPI0918841B8 (pt) * 2008-08-28 2021-05-25 Pfizer derivados de dioxa-biciclo[3.2.1]octano-2,3,4-triol, seus cristais, composições farmacêuticas e usos
DE102009012423A1 (de) 2009-03-10 2010-09-16 Bayer Animal Health Gmbh Zubereitung auf Ölbasis
CN108524480A (zh) 2011-03-02 2018-09-14 国立大学法人东京大学 体内寄生虫防除剂
RU2638830C2 (ru) * 2011-11-25 2017-12-18 Байер Интеллектуэль Проперти Гмбх Применение арильных и гетарильных карбоксамидов в качестве эндопаразитицидов
TWI749509B (zh) * 2015-05-20 2021-12-11 美商百靈佳殷格翰動物保健美國有限公司 驅蟲酯肽化合物
BR112018013369A2 (pt) * 2015-12-28 2019-02-19 Merial, Inc. compostos depsipeptídicos anti-helmínticos
JP2020504710A (ja) 2016-11-16 2020-02-13 ベーリンガー インゲルハイム アニマル ヘルス ユーエスエイ インコーポレイテッド 駆虫性デプシペプチド化合物
EP4013388A1 (en) 2019-08-14 2022-06-22 Vetoquinol SA Compositions comprising tigolaner for controlling parasites
CN113943350B (zh) * 2021-11-02 2023-08-15 海南大学三亚南繁研究院 一种环肽化合物或其药学上可接受的盐及其制备方法和应用、药物及其应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO176766C (no) * 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
GB9024924D0 (en) * 1990-11-16 1991-01-02 Beecham Group Plc Novel compositions
NZ247278A (en) * 1991-02-12 1995-03-28 Ancare Distributors Veterinary anthelmintic drench comprising a suspension of praziquantel in a liquid carrier
PT634408E (pt) * 1992-03-17 2002-05-31 Fujisawa Pharmaceutical Co Derivado de depsipeptido sua producao e utilizacao
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
CN1073560C (zh) * 1993-02-19 2001-10-24 明治制果株式会社 环缩酚酸肽pf1022衍生物
DE4317457A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4317432A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005055973A3 (de) * 2003-12-13 2005-08-11 Bayer Healthcare Ag Endoparasitizide mittel zur topischen applikation

Also Published As

Publication number Publication date
ES2168285T3 (es) 2002-06-16
JP2007314580A (ja) 2007-12-06
RU95100759A (ru) 1997-03-20
TW364850B (en) 1999-07-21
CA2139725A1 (en) 1995-07-12
PL180019B1 (pl) 2000-12-29
FR06C0002I1 (en:Method) 2006-03-10
NO2006001I1 (no) 2006-02-13
US5589503A (en) 1996-12-31
DK0662326T5 (da) 2008-11-03
HUT69180A (en) 1995-08-28
FR06C0002I2 (en:Method) 2006-12-29
CA2139725C (en) 2005-01-04
IL112285A0 (en) 1995-03-30
DK0662326T3 (da) 2002-03-18
DE122006000001I2 (de) 2007-05-24
CZ290246B6 (cs) 2002-06-12
EP0662326B1 (de) 2001-11-28
NZ270300A (en) 1995-09-26
EP0662326A2 (de) 1995-07-12
FI950091A0 (fi) 1995-01-09
UA41327C2 (uk) 2001-09-17
DE122006000001I1 (de) 2006-05-04
CN1165338C (zh) 2004-09-08
NL300218I1 (nl) 2006-04-03
CZ6195A3 (en) 1995-07-12
CN1121429A (zh) 1996-05-01
JPH07223951A (ja) 1995-08-22
NL300218I2 (nl) 2006-07-03
PL306709A1 (en) 1995-07-24
PH31462A (en) 1998-11-03
NO2006001I2 (no) 2008-02-04
NO307030B1 (no) 2000-01-31
FI950091L (fi) 1995-07-12
NO950093D0 (no) 1995-01-10
RU2124364C1 (ru) 1999-01-10
KR950031104A (ko) 1995-12-18
EP0662326A3 (de) 1997-12-17
SK283367B6 (sk) 2003-06-03
PT662326E (pt) 2002-05-31
ZA95136B (en) 1995-09-07
IL112285A (en) 1999-06-20
HU226207B1 (en) 2008-06-30
NO950093L (no) 1995-07-12
SK3195A3 (en) 1995-08-09
DE59409977D1 (de) 2002-01-10
AU8159294A (en) 1995-07-20
JP4033920B2 (ja) 2008-01-16
KR100359618B1 (ko) 2003-01-29
AU685535B2 (en) 1998-01-22
FI116885B (fi) 2006-03-31
ATE209501T1 (de) 2001-12-15

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Legal Events

Date Code Title Description
8139 Disposal/non-payment of the annual fee