DE3360589D1 - 4"-epi erythromycin a and derivatives thereof as useful antibacterial agents - Google Patents

4"-epi erythromycin a and derivatives thereof as useful antibacterial agents

Info

Publication number
DE3360589D1
DE3360589D1 DE8383300905T DE3360589T DE3360589D1 DE 3360589 D1 DE3360589 D1 DE 3360589D1 DE 8383300905 T DE8383300905 T DE 8383300905T DE 3360589 T DE3360589 T DE 3360589T DE 3360589 D1 DE3360589 D1 DE 3360589D1
Authority
DE
Germany
Prior art keywords
derivatives
antibacterial agents
hydrogen
useful antibacterial
considered
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE8383300905T
Other languages
English (en)
Inventor
Frank C Sciavolino
Mark A Guadliana
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Application granted granted Critical
Publication of DE3360589D1 publication Critical patent/DE3360589D1/de
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DE8383300905T 1982-03-01 1983-02-22 4"-epi erythromycin a and derivatives thereof as useful antibacterial agents Expired DE3360589D1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/353,547 US4382085A (en) 1982-03-01 1982-03-01 4"-Epi erythromycin A and derivatives thereof as useful antibacterial agents

Publications (1)

Publication Number Publication Date
DE3360589D1 true DE3360589D1 (en) 1985-09-26

Family

ID=23389603

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8383300905T Expired DE3360589D1 (en) 1982-03-01 1983-02-22 4"-epi erythromycin a and derivatives thereof as useful antibacterial agents

Country Status (26)

Country Link
US (1) US4382085A (de)
EP (1) EP0087905B1 (de)
JP (1) JPS58159499A (de)
KR (1) KR850000965B1 (de)
AT (1) ATE15048T1 (de)
AU (1) AU555208B2 (de)
CA (1) CA1178596A (de)
CS (3) CS235036B2 (de)
DD (1) DD211565A5 (de)
DE (1) DE3360589D1 (de)
DK (1) DK157495C (de)
EG (1) EG16630A (de)
ES (2) ES8403928A1 (de)
FI (1) FI74287C (de)
GR (1) GR78094B (de)
GT (1) GT198301599A (de)
HU (1) HU193157B (de)
IE (1) IE56056B1 (de)
IL (1) IL68004A (de)
NO (1) NO155932C (de)
NZ (1) NZ203417A (de)
PH (1) PH17908A (de)
PL (1) PL138758B1 (de)
PT (1) PT76298B (de)
RO (1) RO86647B (de)
ZA (1) ZA831356B (de)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4526889A (en) * 1982-11-15 1985-07-02 Pfizer Inc. Epimeric azahomoerythromycin A derivative, intermediates and method of use
PH19293A (en) * 1982-11-15 1986-03-04 Pfizer Epimeric azahomoerythromycin,pharmaceutical composition containing the same and method of use thereof
GR80277B (en) * 1983-09-06 1985-01-04 Pfizer Azahomoerythromycin b derivatives and intermediates therefor
JPS60120895A (ja) * 1983-12-02 1985-06-28 Taisho Pharmaceut Co Ltd 6−0−メチル−2′−0,ν−ビス(ベンジルオキシカルボニル)−ν−デメチルエリスロマイシンaの製法
JPS60214796A (ja) * 1984-04-06 1985-10-28 Taisho Pharmaceut Co Ltd 6−0−メチルエリスロマイシン類の製法
EP0184921A3 (de) * 1984-12-08 1986-10-29 Beecham Group Plc Erythromycinderivate
US4783811A (en) * 1984-12-27 1988-11-08 Texas Instruments Incorporated Method and apparatus for determining syllable boundaries
US4681872A (en) * 1985-11-12 1987-07-21 Abbott Laboratories Erythromycin A 11,12-carbonate and method of use
US4640910A (en) * 1985-11-12 1987-02-03 Abbott Laboratories Erythromycin A silylated compounds and method of use
US4833236A (en) * 1986-05-02 1989-05-23 Taisho Pharmaceutical Co., Ltd. Erythromycin derivatives
DK0699207T3 (da) * 1993-05-19 1997-12-08 Pfizer Mellemprodukt til azithromycin
US5441939A (en) * 1994-03-04 1995-08-15 Pfizer Inc. 3"-desmethoxy derivatives of erythromycin and azithromycin
US5605889A (en) * 1994-04-29 1997-02-25 Pfizer Inc. Method of administering azithromycin
CA2492846C (en) * 2002-08-29 2012-09-25 Kosan Biosciences, Inc. Motilide compounds
WO2004101592A1 (ja) * 2003-05-19 2004-11-25 Taisho Pharmaceutical Co., Ltd. エリスロマイシンa誘導体の製造方法
US7211568B2 (en) * 2003-12-18 2007-05-01 Kosan Biosciences Incorporated 9-Desoxoerythromycin compounds as prokinetic agents

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3417077A (en) * 1966-05-16 1968-12-17 Lilly Co Eli Erythromycin derivative and process for the preparation thereof
US3884904A (en) * 1973-06-21 1975-05-20 Abbott Lab 11-Substituted erythromycin B derivatives
US3884903A (en) * 1973-06-21 1975-05-20 Abbott Lab 4{41 -Deoxy-4{41 -oxoerythromycin B derivatives
SE445223B (sv) * 1977-02-04 1986-06-09 Pfizer Sett att framstella 4"-amino-erytomylin-a-derivat
US4150220A (en) * 1977-02-04 1979-04-17 Pfizer Inc. Semi-synthetic 4"-erythromycin A derivatives

Also Published As

Publication number Publication date
KR840003647A (ko) 1984-09-15
AU555208B2 (en) 1986-09-18
US4382085A (en) 1983-05-03
RO86647A (ro) 1985-04-17
ES520177A0 (es) 1984-04-01
DK96783D0 (da) 1983-02-28
CS235036B2 (en) 1985-04-16
DD211565A5 (de) 1984-07-18
CS235048B2 (en) 1985-04-16
IE56056B1 (en) 1991-04-10
DK96783A (da) 1983-09-02
GT198301599A (es) 1984-09-13
PL240764A1 (en) 1985-01-02
ATE15048T1 (de) 1985-09-15
RO86647B (ro) 1985-05-01
PL138758B1 (en) 1986-10-31
IL68004A0 (en) 1983-06-15
ZA831356B (en) 1983-11-30
PH17908A (en) 1985-01-25
GR78094B (de) 1984-09-26
DK157495C (da) 1990-06-11
FI74287C (fi) 1988-01-11
CS235049B2 (en) 1985-04-16
PT76298A (en) 1983-03-01
EP0087905B1 (de) 1985-08-21
EG16630A (en) 1991-03-30
ES526323A0 (es) 1985-11-16
IE830411L (en) 1983-09-01
CA1178596A (en) 1984-11-27
ES8602837A1 (es) 1985-11-16
ES8403928A1 (es) 1984-04-01
EP0087905A1 (de) 1983-09-07
NO830686L (no) 1983-09-02
AU1189883A (en) 1983-09-08
IL68004A (en) 1986-11-30
FI830654A0 (fi) 1983-02-28
FI74287B (fi) 1987-09-30
PT76298B (en) 1986-01-27
JPS58159499A (ja) 1983-09-21
NZ203417A (en) 1985-10-11
FI830654L (fi) 1983-09-02
NO155932C (no) 1987-06-24
DK157495B (da) 1990-01-15
KR850000965B1 (ko) 1985-07-02
HU193157B (en) 1987-08-28
NO155932B (no) 1987-03-16
JPH0140039B2 (de) 1989-08-24

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition