DE3116890A1 - "2-guanidinothiazolderivate" - Google Patents
"2-guanidinothiazolderivate"Info
- Publication number
- DE3116890A1 DE3116890A1 DE19813116890 DE3116890A DE3116890A1 DE 3116890 A1 DE3116890 A1 DE 3116890A1 DE 19813116890 DE19813116890 DE 19813116890 DE 3116890 A DE3116890 A DE 3116890A DE 3116890 A1 DE3116890 A1 DE 3116890A1
- Authority
- DE
- Germany
- Prior art keywords
- guanidino
- thiazole
- general formula
- group
- radical
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US14494680A | 1980-04-29 | 1980-04-29 |
Publications (1)
Publication Number | Publication Date |
---|---|
DE3116890A1 true DE3116890A1 (de) | 1982-03-04 |
Family
ID=22510873
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE19813116890 Ceased DE3116890A1 (de) | 1980-04-29 | 1981-04-28 | "2-guanidinothiazolderivate" |
Country Status (16)
Country | Link |
---|---|
JP (1) | JPS574977A (fr) |
AR (1) | AR231538A1 (fr) |
AU (1) | AU540239B2 (fr) |
BE (1) | BE888602A (fr) |
CH (1) | CH646964A5 (fr) |
DE (1) | DE3116890A1 (fr) |
DK (1) | DK188881A (fr) |
ES (1) | ES501736A0 (fr) |
FR (1) | FR2481280A1 (fr) |
GB (1) | GB2076397B (fr) |
IE (1) | IE51151B1 (fr) |
IL (1) | IL62747A (fr) |
IT (1) | IT1146750B (fr) |
NL (1) | NL8102099A (fr) |
NZ (1) | NZ196923A (fr) |
SE (1) | SE452462B (fr) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3332138A1 (de) * | 1982-12-03 | 1984-06-07 | Kotobuki Seiyaku Co. Ltd., Nagano | 2,4-substituierte thiazolderivate, verfahren zu deren herstellung und diese enthaltende arzneimittel |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4501747A (en) * | 1982-05-10 | 1985-02-26 | Sanofi | Certain amide derivatives of 2-guanidino-thiazoles and compositions containing same |
FR2531705B1 (fr) * | 1982-08-13 | 1986-12-05 | Sanofi Sa | Amidobenzamides, leurs sels, procede pour leur preparation et compositions pharmaceutiques les renfermant |
EP0123741A1 (fr) * | 1983-04-26 | 1984-11-07 | Shionogi & Co., Ltd. | 2-Guanidino-4-hydroxyméthylthiazoles et leurs dérivés |
US4680300A (en) * | 1985-01-10 | 1987-07-14 | Syntex (U.S.A.) Inc. | Anti-inflammatory guanidines |
US4837316A (en) * | 1985-08-29 | 1989-06-06 | Fujirebio Kabushiki Kaisha | Alkylamide derivatives with H2 -receptor antagonistic and cytoprotective action |
EP0385525B1 (fr) * | 1989-03-03 | 1994-04-13 | Akzo Nv | Dérivés d'aminoéthylthiazole et d'aminoéthyloxazole. |
Citations (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4165377A (en) * | 1977-04-20 | 1979-08-21 | Ici Americas Inc. | Guanidino imidazoles and thiazoles |
US4165378A (en) * | 1977-04-20 | 1979-08-21 | Ici Americas Inc. | Guanidine derivatives of imidazoles and thiazoles |
JPS5555174A (en) | 1978-10-16 | 1980-04-22 | Ici Ltd | Branched chain heterocyclic derivative*its manufacture and pharmaceutic composition containing it and having secretion controlling activity |
DE3008056A1 (de) * | 1979-03-06 | 1980-09-18 | Yamanouchi Pharma Co Ltd | Guanidinothiazolverbindungen, verfahren zu ihrer herstellung und arzneimittel |
EP0030092A1 (fr) * | 1979-11-13 | 1981-06-10 | Imperial Chemical Industries Plc | Dérivés de la guanidine, procédés pour leur préparation et compositions pharmaceutiques les contenant |
DE3150334A1 (de) * | 1980-12-19 | 1982-07-15 | Shionogi & Co., Ltd., Osaka | "bis-(carboxamid)-derivate" |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS54132566A (en) * | 1978-01-18 | 1979-10-15 | Ici Ltd | Guanidine derivative*its manufacture and secretion controlling pharmaceutical composition containing it |
US4309435A (en) * | 1978-10-16 | 1982-01-05 | Imperial Chemical Industries Ltd. | Antisecretory guanidine derivatives and pharmaceutical compositions containing them |
DE3069889D1 (en) * | 1979-01-18 | 1985-02-14 | Ici Plc | Guanidine derivatives, processes for their manufacture and pharmaceutical compositions containing them |
JPS5754177A (ja) * | 1980-09-19 | 1982-03-31 | Teikoku Hormone Mfg Co Ltd | Chikanchiazoorujudotai |
-
1981
- 1981-04-24 NZ NZ196923A patent/NZ196923A/xx unknown
- 1981-04-28 SE SE8102683A patent/SE452462B/sv not_active IP Right Cessation
- 1981-04-28 JP JP6473981A patent/JPS574977A/ja active Granted
- 1981-04-28 ES ES501736A patent/ES501736A0/es active Granted
- 1981-04-28 DK DK188881A patent/DK188881A/da not_active Application Discontinuation
- 1981-04-28 FR FR8108468A patent/FR2481280A1/fr active Granted
- 1981-04-28 BE BE0/204631A patent/BE888602A/fr not_active IP Right Cessation
- 1981-04-28 DE DE19813116890 patent/DE3116890A1/de not_active Ceased
- 1981-04-28 NL NL8102099A patent/NL8102099A/nl not_active Application Discontinuation
- 1981-04-29 GB GB8113289A patent/GB2076397B/en not_active Expired
- 1981-04-29 IL IL62747A patent/IL62747A/xx unknown
- 1981-04-29 AU AU69966/81A patent/AU540239B2/en not_active Ceased
- 1981-04-29 IE IE956/81A patent/IE51151B1/en unknown
- 1981-04-29 CH CH279381A patent/CH646964A5/de not_active IP Right Cessation
- 1981-04-29 IT IT67585/81A patent/IT1146750B/it active
-
1984
- 1984-01-01 AR AR23153884D patent/AR231538A1/es active
Patent Citations (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4165377A (en) * | 1977-04-20 | 1979-08-21 | Ici Americas Inc. | Guanidino imidazoles and thiazoles |
US4165378A (en) * | 1977-04-20 | 1979-08-21 | Ici Americas Inc. | Guanidine derivatives of imidazoles and thiazoles |
JPS5555174A (en) | 1978-10-16 | 1980-04-22 | Ici Ltd | Branched chain heterocyclic derivative*its manufacture and pharmaceutic composition containing it and having secretion controlling activity |
EP0010893A1 (fr) * | 1978-10-16 | 1980-05-14 | Imperial Chemical Industries Plc | Dérivés antisécrétoires hétérocycliques de la guanidine comprenant des chaînes ramifiées, procédés pour leur préparation, produits intermédiaires et compositions pharmaceutiques contenant lesdits dérivés |
DE3008056A1 (de) * | 1979-03-06 | 1980-09-18 | Yamanouchi Pharma Co Ltd | Guanidinothiazolverbindungen, verfahren zu ihrer herstellung und arzneimittel |
EP0030092A1 (fr) * | 1979-11-13 | 1981-06-10 | Imperial Chemical Industries Plc | Dérivés de la guanidine, procédés pour leur préparation et compositions pharmaceutiques les contenant |
DE3150334A1 (de) * | 1980-12-19 | 1982-07-15 | Shionogi & Co., Ltd., Osaka | "bis-(carboxamid)-derivate" |
Non-Patent Citations (1)
Title |
---|
JP-Kokai 55-55 174 * |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3332138A1 (de) * | 1982-12-03 | 1984-06-07 | Kotobuki Seiyaku Co. Ltd., Nagano | 2,4-substituierte thiazolderivate, verfahren zu deren herstellung und diese enthaltende arzneimittel |
Also Published As
Publication number | Publication date |
---|---|
CH646964A5 (de) | 1984-12-28 |
ES8206501A1 (es) | 1982-08-16 |
AR231538A1 (es) | 1984-12-28 |
IE810956L (en) | 1981-10-29 |
IL62747A0 (en) | 1981-06-29 |
SE8102683L (sv) | 1981-10-30 |
DK188881A (da) | 1981-10-30 |
GB2076397B (en) | 1984-02-08 |
NZ196923A (en) | 1983-12-16 |
BE888602A (fr) | 1981-10-28 |
ES501736A0 (es) | 1982-08-16 |
IT1146750B (it) | 1986-11-19 |
GB2076397A (en) | 1981-12-02 |
IT8167585A0 (it) | 1981-04-29 |
AU540239B2 (en) | 1984-11-08 |
AU6996681A (en) | 1981-11-05 |
FR2481280B1 (fr) | 1983-10-28 |
FR2481280A1 (fr) | 1981-10-30 |
NL8102099A (nl) | 1981-11-16 |
IL62747A (en) | 1984-10-31 |
IE51151B1 (en) | 1986-10-15 |
JPS574977A (en) | 1982-01-11 |
JPH027952B2 (fr) | 1990-02-21 |
SE452462B (sv) | 1987-11-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8110 | Request for examination paragraph 44 | ||
8131 | Rejection |