DE2362816A1 - Mit heterocyclischer acylgruppe substituierte cephalosporinderivate - Google Patents

Mit heterocyclischer acylgruppe substituierte cephalosporinderivate

Info

Publication number
DE2362816A1
DE2362816A1 DE19732362816 DE2362816A DE2362816A1 DE 2362816 A1 DE2362816 A1 DE 2362816A1 DE 19732362816 DE19732362816 DE 19732362816 DE 2362816 A DE2362816 A DE 2362816A DE 2362816 A1 DE2362816 A1 DE 2362816A1
Authority
DE
Germany
Prior art keywords
group
solution
atom
formula
added
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19732362816
Other languages
German (de)
English (en)
Inventor
Ichiro Isaka
Teruya Kashiwagi
Norio Kawahara
Akio Koda
Tetsuya Maeda
Masuo Murakami
Yukiyasu Murakami
Isao Souzu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Astellas Pharma Inc
Original Assignee
Yamanouchi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP12843172A external-priority patent/JPS551273B2/ja
Priority claimed from JP2684073A external-priority patent/JPS49110686A/ja
Priority claimed from JP5644173A external-priority patent/JPS504090A/ja
Priority claimed from JP8940873A external-priority patent/JPS5036487A/ja
Application filed by Yamanouchi Pharmaceutical Co Ltd filed Critical Yamanouchi Pharmaceutical Co Ltd
Publication of DE2362816A1 publication Critical patent/DE2362816A1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
DE19732362816 1972-12-21 1973-12-18 Mit heterocyclischer acylgruppe substituierte cephalosporinderivate Pending DE2362816A1 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP12843172A JPS551273B2 (enExample) 1972-12-21 1972-12-21
JP2684073A JPS49110686A (enExample) 1973-03-07 1973-03-07
JP5644173A JPS504090A (enExample) 1973-05-21 1973-05-21
JP8940873A JPS5036487A (enExample) 1973-08-09 1973-08-09

Publications (1)

Publication Number Publication Date
DE2362816A1 true DE2362816A1 (de) 1974-06-27

Family

ID=27458582

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19732362816 Pending DE2362816A1 (de) 1972-12-21 1973-12-18 Mit heterocyclischer acylgruppe substituierte cephalosporinderivate

Country Status (5)

Country Link
AT (1) AT328081B (enExample)
CA (1) CA1022544A (enExample)
DE (1) DE2362816A1 (enExample)
FR (1) FR2211214B1 (enExample)
GB (1) GB1449256A (enExample)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2539664A1 (de) * 1974-09-06 1976-03-18 Sumitomo Chemical Co Cephalosporin-derivate
JPS5188988A (enExample) * 1975-01-31 1976-08-04
US4015000A (en) * 1972-09-29 1977-03-29 Ciba-Geigy Corporation 6-Acylamino-penam-3-carboxylic and 7-acylamino-3-cephem-4-carboxylic acids
DE2657652A1 (de) * 1976-01-15 1977-07-21 Cusi Lab Acyl-cephalosporine
DE2737066A1 (de) * 1976-08-17 1978-02-23 Fujisawa Pharmaceutical Co 7-(n-substituierte-2-phenylglycinamido)-3-substituierte-3-cephem-4-carbonsaeure-verbindungen, verfahren zu ihrer herstellung und sie enthaltende arzneimittel

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS51115491A (en) * 1975-04-03 1976-10-12 Sumitomo Chem Co Ltd Method for preparing 77* *44hydroxyy1*5 naphthyridinee33carboxyamino ** phenylacetamido*cephalosporins
US4302454A (en) 1976-03-03 1981-11-24 Sumitomo Chemical Company, Limited Cephalosporins
US4041162A (en) * 1976-03-11 1977-08-09 Smithkline Corporation 7-Acyl-3-(sulfoalkyl substituted oxadiazolylthiomethyl) cephalosporins
EP0003115A1 (en) * 1978-01-16 1979-07-25 Sandoz Ag Penicillins, per se and for use as antibacterially active antibiotics and their production
GB2045238B (en) * 1978-11-28 1982-12-01 Mitsui Toatsu Chemicals Cephalosporins
JPS5764698A (en) * 1980-10-07 1982-04-19 Eisai Co Ltd Cephem derivative, its preparation, and antibacterial agent composed of said derivative
US4468394A (en) * 1981-04-02 1984-08-28 Eisai Co., Ltd. Cephalosporin compounds
AU2006326662B2 (en) 2005-12-09 2011-07-28 Amgen Inc. Quinolone based compounds exhibiting prolyl hydroxylase inhibitory activity, and compositions, and uses thereof
US8048892B2 (en) 2006-12-18 2011-11-01 Amgen Inc. Azaquinolone based compounds exhibiting prolyl hydroxylase inhibitory activity, compositions, and uses thereof
WO2008076427A2 (en) 2006-12-18 2008-06-26 Amgen Inc. Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory activity, compositions, and uses thereof
EP2142509B1 (en) 2007-04-18 2013-12-04 Amgen, Inc Quinolones and azaquinolones that inhibit prolyl hydroxylase
ES2446418T3 (es) 2007-04-18 2014-03-07 Amgen, Inc Derivados de indanona que inhiben la prolil hidroxilasa
CA2685219C (en) 2007-05-04 2012-06-19 Amgen Inc. Diazaquinolones that inhibit prolyl hydroxylase activity
US8030346B2 (en) 2007-05-04 2011-10-04 Amgen Inc. Heterocyclic quinolone derivatives that inhibit prolyl hydroxylase activity

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL38099A (en) * 1970-12-17 1976-01-30 Smith Kline French Lab 3-heterocyclyl thiomethylcephalosporins

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4015000A (en) * 1972-09-29 1977-03-29 Ciba-Geigy Corporation 6-Acylamino-penam-3-carboxylic and 7-acylamino-3-cephem-4-carboxylic acids
DE2539664A1 (de) * 1974-09-06 1976-03-18 Sumitomo Chemical Co Cephalosporin-derivate
DK157246B (da) * 1974-09-06 1989-11-27 Sumitomo Chemical Co Analogifremgangsmaade til fremstilling af n-acylamino-alfa-phenylacetamidocephalosporiner eller farmaceutisk acceptable salte heraf.
JPS5188988A (enExample) * 1975-01-31 1976-08-04
DE2657652A1 (de) * 1976-01-15 1977-07-21 Cusi Lab Acyl-cephalosporine
DE2737066A1 (de) * 1976-08-17 1978-02-23 Fujisawa Pharmaceutical Co 7-(n-substituierte-2-phenylglycinamido)-3-substituierte-3-cephem-4-carbonsaeure-verbindungen, verfahren zu ihrer herstellung und sie enthaltende arzneimittel

Also Published As

Publication number Publication date
CA1022544A (en) 1977-12-13
FR2211214B1 (enExample) 1978-01-13
FR2211214A1 (enExample) 1974-07-19
ATA1075673A (de) 1975-05-15
GB1449256A (en) 1976-09-15
AT328081B (de) 1976-03-10

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