DE1593057A1 - Steroid-Pyrazole und Verfahren zu ihrer Herstellung - Google Patents

Steroid-Pyrazole und Verfahren zu ihrer Herstellung

Info

Publication number
DE1593057A1
DE1593057A1 DE19661593057 DE1593057A DE1593057A1 DE 1593057 A1 DE1593057 A1 DE 1593057A1 DE 19661593057 DE19661593057 DE 19661593057 DE 1593057 A DE1593057 A DE 1593057A DE 1593057 A1 DE1593057 A1 DE 1593057A1
Authority
DE
Germany
Prior art keywords
compounds
oxo
hydroxy
pregneno
dihydroxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19661593057
Other languages
German (de)
English (en)
Inventor
Hirschmann Ralph Franz
John Fried
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of DE1593057A1 publication Critical patent/DE1593057A1/de
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J75/00Processes for the preparation of steroids in general
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE19661593057 1965-07-30 1966-07-29 Steroid-Pyrazole und Verfahren zu ihrer Herstellung Pending DE1593057A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US47616065A 1965-07-30 1965-07-30

Publications (1)

Publication Number Publication Date
DE1593057A1 true DE1593057A1 (de) 1970-04-23

Family

ID=23890732

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19661593057 Pending DE1593057A1 (de) 1965-07-30 1966-07-29 Steroid-Pyrazole und Verfahren zu ihrer Herstellung

Country Status (8)

Country Link
BE (1) BE684857A (ru)
BR (1) BR6681630D0 (ru)
CH (1) CH566350A5 (ru)
DE (1) DE1593057A1 (ru)
ES (1) ES329985A1 (ru)
GB (1) GB1141070A (ru)
IL (1) IL26185A (ru)
NL (1) NL6610736A (ru)

Also Published As

Publication number Publication date
CH566350A5 (en) 1975-09-15
BE684857A (ru) 1967-01-30
GB1141070A (en) 1969-01-22
NL6610736A (ru) 1967-01-31
BR6681630D0 (pt) 1973-12-04
IL26185A (en) 1970-03-22
ES329985A1 (es) 1967-06-01

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