DE1291337B - Verfahren zur Herstellung von neuen 3-Oxo-17ª‰-hydroxy-4, 9, 11-gonatrienderivaten und 17ª‰-Acylaten derselben - Google Patents

Verfahren zur Herstellung von neuen 3-Oxo-17ª‰-hydroxy-4, 9, 11-gonatrienderivaten und 17ª‰-Acylaten derselben

Info

Publication number
DE1291337B
DE1291337B DER37266A DER0037266A DE1291337B DE 1291337 B DE1291337 B DE 1291337B DE R37266 A DER37266 A DE R37266A DE R0037266 A DER0037266 A DE R0037266A DE 1291337 B DE1291337 B DE 1291337B
Authority
DE
Germany
Prior art keywords
hydroxy
oxo
oximino
ecm
water
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DER37266A
Other languages
German (de)
English (en)
Inventor
Nomine
Dr-Ing Gerard
Bucourt
Dr-Ing Robert
Pierdet Andre
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Priority claimed from FR974762A external-priority patent/FR1514075A/fr
Publication of DE1291337B publication Critical patent/DE1291337B/de
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23K—FODDER
    • A23K20/00—Accessory food factors for animal feeding-stuffs
    • A23K20/10—Organic substances
    • A23K20/168—Steroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/566—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol having an oxo group in position 17, e.g. estrone
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J75/00—Processes for the preparation of steroids in general
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/16—Benz[e]indenes; Hydrogenated benz[e]indenes
DER37266A 1963-02-20 1964-02-20 Verfahren zur Herstellung von neuen 3-Oxo-17ª‰-hydroxy-4, 9, 11-gonatrienderivaten und 17ª‰-Acylaten derselben Pending DE1291337B (de)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
FR925431A FR1426077A (fr) 1963-02-20 1963-02-20 Nouveau dérivé estratriénique et procédé de préparation
FR940549A FR1453214A (fr) 1963-02-20 1963-07-05 Nouveaux dérivés stéroïdes insaturés et procédés de préparation
FR949609A FR3060M (fr) 1963-02-20 1963-10-04 Nouveau médicament doué notamment d'activité hypocholestérolémiante.
FR949608A FR3069M (fr) 1963-02-20 1963-10-04 Nouveau médicament notamment pour le traitement des troubles de l'anabolisme protidique.
BE644138A BE644138A (xx) 1963-02-20 1964-02-20
FR974762A FR1514075A (fr) 1964-02-17 1964-05-15 Nouveau dérivé stéroïde triénique et procédé de préparation
FR985285A FR3804M (fr) 1963-02-20 1964-08-14 Nouveau médicament notamment pour le traitement des troubles dus a une insuffisance de sécrétion du corps jaune.
FR19090A FR1492782A (fr) 1963-02-20 1965-06-01 Nouveau dérivé stéroïde insaturé et procédé de préparation
FR29732A FR5235M (xx) 1963-02-20 1965-08-27

Publications (1)

Publication Number Publication Date
DE1291337B true DE1291337B (de) 1969-03-27

Family

ID=27575680

Family Applications (2)

Application Number Title Priority Date Filing Date
DER37266A Pending DE1291337B (de) 1963-02-20 1964-02-20 Verfahren zur Herstellung von neuen 3-Oxo-17ª‰-hydroxy-4, 9, 11-gonatrienderivaten und 17ª‰-Acylaten derselben
DE19661593307 Withdrawn DE1593307A1 (de) 1963-02-20 1966-06-01 Neues Verfahren zur Herstellung von Gonatrienderivaten

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE19661593307 Withdrawn DE1593307A1 (de) 1963-02-20 1966-06-01 Neues Verfahren zur Herstellung von Gonatrienderivaten

Country Status (11)

Country Link
US (2) US3248294A (xx)
BE (1) BE644138A (xx)
BR (2) BR6456982D0 (xx)
CH (2) CH429713A (xx)
DE (2) DE1291337B (xx)
DK (1) DK117957B (xx)
FR (8) FR1426077A (xx)
GB (2) GB1048232A (xx)
NL (6) NL6401555A (xx)
OA (2) OA01429A (xx)
SE (3) SE323073B (xx)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3424745A (en) * 1964-05-27 1969-01-28 Roussel Uclaf Novel process for the preparation of trienic steroid derivatives
US3346454A (en) * 1964-11-04 1967-10-10 Roussel Uclaf 17-alkyl-19-nor-delta4, 9, 11-pregnatriene-3, 20-diones, process and intermediates for preparing same and therapeutic compositions thereof
US3422121A (en) * 1965-08-13 1969-01-14 Merck & Co Inc Process for the preparation of 13-lower alkyl-gona-4,8(14),9-triene-3,17-dione
US3424769A (en) * 1966-04-04 1969-01-28 Syntex Corp Process for the preparation of novel 6alpha-methyl-delta4,9(10)- diene steroids
NL129638C (xx) * 1966-08-12
US3461118A (en) * 1966-10-17 1969-08-12 Syntex Corp 3beta-tetrahydrofuranyloxy - and 3beta-tetrahydropyranyloxyestra - 4,9(10) - dienes and -4,9(10),11-trienes,their preparation and intermediates thereof
US3760073A (en) * 1971-06-09 1973-09-18 Roussel Uclaf Treatment of wounds
FR2162268A1 (en) * 1971-12-08 1973-07-20 Roussel Uclaf 6-alpha, 17-beta-dihydroxy-13-beta-ethyl-17-alpha - -ethynylgona-4,9,11-triene-3-one - with anti oesterogenic anti-lh and
FR2407940A1 (fr) * 1977-11-08 1979-06-01 Roussel Uclaf Nouveaux derives steroides 17 a-aryle, ou 17 a-heteroaryle, leur procede de preparation et leur application comme medicament
HU201091B (en) * 1985-12-26 1990-09-28 Mitsubishi Chem Ind Process for producing gonatriene derivatives and pharmaceutical compositions comprising same
HU203667B (en) * 1986-12-11 1991-09-30 Roussel Uclaf Process for producing synergetic zootechnical compositions containing three components
DE4232521A1 (de) * 1992-09-22 1994-03-24 Schering Ag Gestagen wirksame 4,5;11,12-Estradiene, Verfahren zu ihrer Herstellung, diese Estradiene enthaltende Arzneimittel sowie deren Verwendung zur Herstellung von Arzneimitteln
FR2696641B1 (fr) * 1992-10-13 1997-07-04 Roussel Uclaf Nouvelle utilisation de l'altrenogest.
US6498153B1 (en) 1998-12-31 2002-12-24 Akzo Nobel N.V. Extended release growth promoting two component composition
CN101704871B (zh) * 2009-12-01 2012-05-23 北京紫竹药业有限公司 甾体化合物及其用途

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
None *

Also Published As

Publication number Publication date
FR3069M (fr) 1965-01-18
FR1492782A (fr) 1967-08-25
US3248294A (en) 1966-04-26
OA01428A (fr) 1969-07-04
NL124135C (xx)
NL127247C (xx)
FR3804M (fr) 1966-01-03
BE644138A (xx) 1964-08-20
FR1426077A (fr) 1966-01-28
DK117957B (da) 1970-06-22
CH467255A (fr) 1969-01-15
FR5235M (xx) 1967-07-17
OA01429A (fr) 1969-07-04
FR3060M (fr) 1965-01-11
GB1048232A (en) 1966-11-16
DE1593307A1 (de) 1970-07-23
BR6456982D0 (pt) 1973-08-14
NL6615432A (xx) 1967-01-25
US3257278A (en) 1966-06-21
SE323073B (xx) 1970-04-27
SE319173B (xx) 1970-01-12
GB1048231A (en) 1966-11-16
NL6401555A (xx) 1964-08-21
FR1453214A (fr) 1966-06-03
CH429713A (fr) 1967-02-15
FR2713M (fr) 1964-08-10
SE323071B (xx) 1970-04-27
NL6607609A (xx) 1966-12-02
NL126190C (xx)
BR6680069D0 (pt) 1973-12-26

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