DD279882A5 - 6-beta-(substituierte)-(s)-hydroxymethyl-penicillan-saeuren und derivate derselben - Google Patents

6-beta-(substituierte)-(s)-hydroxymethyl-penicillan-saeuren und derivate derselben Download PDF

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Publication number
DD279882A5
DD279882A5 DD88312469A DD31246988A DD279882A5 DD 279882 A5 DD279882 A5 DD 279882A5 DD 88312469 A DD88312469 A DD 88312469A DD 31246988 A DD31246988 A DD 31246988A DD 279882 A5 DD279882 A5 DD 279882A5
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DD
German Democratic Republic
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product
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allyl
reaction
group
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DD88312469A
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German (de)
English (en)
Inventor
Yuhpyung L Chen
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Publication of DD279882A5 publication Critical patent/DD279882A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/86—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with only atoms other than nitrogen atoms directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DD88312469A 1987-01-27 1988-01-27 6-beta-(substituierte)-(s)-hydroxymethyl-penicillan-saeuren und derivate derselben DD279882A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US731987A 1987-01-27 1987-01-27

Publications (1)

Publication Number Publication Date
DD279882A5 true DD279882A5 (de) 1990-06-20

Family

ID=21725481

Family Applications (1)

Application Number Title Priority Date Filing Date
DD88312469A DD279882A5 (de) 1987-01-27 1988-01-27 6-beta-(substituierte)-(s)-hydroxymethyl-penicillan-saeuren und derivate derselben

Country Status (25)

Country Link
EP (1) EP0276942B1 (pt)
JP (1) JPS63246384A (pt)
KR (1) KR900005050B1 (pt)
CN (1) CN1014710B (pt)
AT (1) ATE74359T1 (pt)
AU (2) AU590142B2 (pt)
CA (1) CA1288091C (pt)
DD (1) DD279882A5 (pt)
DE (1) DE3869630D1 (pt)
DK (1) DK36788A (pt)
ES (1) ES2031589T3 (pt)
FI (1) FI880334A (pt)
GR (1) GR3004460T3 (pt)
HU (1) HU205765B (pt)
IE (1) IE60348B1 (pt)
IL (1) IL85167A (pt)
MY (1) MY102312A (pt)
NO (1) NO172493C (pt)
NZ (1) NZ223296A (pt)
PH (1) PH24478A (pt)
PL (2) PL159842B1 (pt)
PT (1) PT86613B (pt)
SU (2) SU1591812A3 (pt)
YU (2) YU46436B (pt)
ZA (1) ZA88514B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0276942B1 (en) * 1987-01-27 1992-04-01 Pfizer Inc. 6-beta(substituted)-(s)-hydroxymethylpenicillanic acids and derivatives thereof
AU5617398A (en) * 1996-12-30 1998-07-31 Beacon Laboratories L.L.C. Tricarboxylic acid-containing oxyalkyl esters and uses thereof
GB0128052D0 (en) * 2001-11-22 2002-01-16 Drug Discovery Lab As Compounds
US8187727B2 (en) 2005-07-22 2012-05-29 Lg Chem, Ltd. Imidazole derivatives, preparation method thereof and organic electronic device using the same

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4272439A (en) * 1978-06-02 1981-06-09 Schering Corporation 6-(Substituted-hydroxymethylene penams)
US4304779A (en) * 1979-05-09 1981-12-08 Schering Corporation 6-(Nitrogen-containing heterocyclic)hydroxymethylpenicillanic acids, compounds related thereto and processes for their preparation
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
GR77151B (pt) * 1982-01-11 1984-09-07 Prizer
DD234015A5 (de) * 1984-01-30 1986-03-19 Pfizer Verfahren zur herstellung von 6-(subst.)-methylen-penicillan-und 6-(subst.)-hydroxymethyl-penicillansaeure und deren derivaten
EP0150984B1 (en) * 1984-01-30 1991-09-11 Pfizer Inc. 6-(substituted) methylenepenicillanic and 6-(substituted) hydroxymethylpenicillanic acids and derivatives thereof
EP0276942B1 (en) * 1987-01-27 1992-04-01 Pfizer Inc. 6-beta(substituted)-(s)-hydroxymethylpenicillanic acids and derivatives thereof

Also Published As

Publication number Publication date
YU14488A (en) 1990-02-28
MY102312A (en) 1992-05-28
NO880297L (no) 1988-07-28
PH24478A (en) 1990-07-18
PL159842B1 (pl) 1993-01-29
EP0276942B1 (en) 1992-04-01
KR880009030A (ko) 1988-09-13
HU205765B (en) 1992-06-29
AU1074388A (en) 1988-07-28
IL85167A0 (en) 1988-07-31
FI880334A0 (fi) 1988-01-26
PL161601B1 (pl) 1993-07-30
GR3004460T3 (pt) 1993-03-31
PT86613B (pt) 1991-12-31
FI880334A (fi) 1988-07-28
ES2031589T3 (es) 1992-12-16
IE60348B1 (en) 1994-06-29
DK36788A (da) 1988-09-23
SU1681730A3 (ru) 1991-09-30
AU4883290A (en) 1990-05-17
CN88100588A (zh) 1988-08-10
PT86613A (pt) 1988-02-01
NZ223296A (en) 1989-10-27
ATE74359T1 (de) 1992-04-15
NO172493C (no) 1993-07-28
YU46436B (sh) 1993-10-20
HUT47118A (en) 1989-01-30
EP0276942A1 (en) 1988-08-03
CN1014710B (zh) 1991-11-13
YU124389A (en) 1990-12-31
CA1288091C (en) 1991-08-27
NO172493B (no) 1993-04-19
NO880297D0 (no) 1988-01-25
YU47020B (sh) 1994-11-15
DE3869630D1 (de) 1992-05-07
JPS63246384A (ja) 1988-10-13
DK36788D0 (da) 1988-01-26
IL85167A (en) 1994-01-25
IE880197L (en) 1988-07-27
KR900005050B1 (en) 1990-07-19
PL270301A1 (en) 1988-12-08
SU1591812A3 (ru) 1990-09-07
AU613821B2 (en) 1991-08-08
AU590142B2 (en) 1989-10-26
ZA88514B (en) 1989-09-27

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Legal Events

Date Code Title Description
NPV Change in the person, the name or the address of the representative (addendum to changes before extension act)
ENJ Ceased due to non-payment of renewal fee