DD200799A5 - Verfahren zur herstellung von peptiden - Google Patents

Verfahren zur herstellung von peptiden Download PDF

Info

Publication number
DD200799A5
DD200799A5 DD81234210A DD23421081A DD200799A5 DD 200799 A5 DD200799 A5 DD 200799A5 DD 81234210 A DD81234210 A DD 81234210A DD 23421081 A DD23421081 A DD 23421081A DD 200799 A5 DD200799 A5 DD 200799A5
Authority
DD
German Democratic Republic
Prior art keywords
gly
tyr
phe
met
cys
Prior art date
Application number
DD81234210A
Other languages
German (de)
English (en)
Inventor
Paul D Gesellchen
Robert T Shuman
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of DD200799A5 publication Critical patent/DD200799A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/70Enkephalins
    • C07K14/702Enkephalins with at least 1 amino acid in D-form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Analytical Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Veterinary Medicine (AREA)
  • Neurosurgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Plant Substances (AREA)
DD81234210A 1980-10-20 1981-10-19 Verfahren zur herstellung von peptiden DD200799A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/198,896 US4322339A (en) 1980-10-20 1980-10-20 Pharmacologically active peptides

Publications (1)

Publication Number Publication Date
DD200799A5 true DD200799A5 (de) 1983-06-15

Family

ID=22735325

Family Applications (1)

Application Number Title Priority Date Filing Date
DD81234210A DD200799A5 (de) 1980-10-20 1981-10-19 Verfahren zur herstellung von peptiden

Country Status (22)

Country Link
US (1) US4322339A (fr)
EP (1) EP0050503B1 (fr)
JP (1) JPS57108051A (fr)
KR (1) KR830007517A (fr)
AT (1) ATE8252T1 (fr)
AU (1) AU7657581A (fr)
CA (1) CA1187872A (fr)
DD (1) DD200799A5 (fr)
DE (1) DE3164594D1 (fr)
DK (1) DK461581A (fr)
ES (1) ES506315A0 (fr)
FI (1) FI813199L (fr)
GB (1) GB2085892B (fr)
GR (1) GR75824B (fr)
HU (1) HU185321B (fr)
IL (1) IL64084A0 (fr)
NZ (1) NZ198626A (fr)
PL (1) PL131156B1 (fr)
PT (1) PT73840B (fr)
RO (1) RO83297B (fr)
YU (1) YU249181A (fr)
ZA (1) ZA817062B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK28377A (da) 1976-02-02 1977-08-03 Sandoz Ag Fremgangsmade til fremstilling af polypeptidderivater
DE3163199D1 (en) * 1980-07-17 1984-05-24 Sandoz Ag Novel pentapeptides, processes for their production, pharmaceutical compositions comprising said pentapeptides and their use
FR2488253A1 (fr) * 1980-08-08 1982-02-12 Roques Bernard Nouveaux peptides et leur application en therapeutique
DK134784A (da) * 1983-03-07 1984-09-08 Lilly Co Eli Farmakologisk virksomme tripeptid-derivater og fremgangsmaade til fremstilling deraf
GB8314646D0 (en) * 1983-05-26 1983-06-29 Wellcome Found Pharmaceutical amides
US4495178A (en) * 1983-10-06 1985-01-22 G. D. Searle & Co. Enkephalin analogs
US4599325A (en) * 1984-02-16 1986-07-08 G. D. Searle & Co. Substituted tyrosyl alanine dipeptide amides
US6028168A (en) 1991-08-09 2000-02-22 Winfried Kolbeck Lanthionine bridged peptides
US5952465A (en) * 1993-04-23 1999-09-14 Virginia Commonwealth University Polypeptides that include conformation-constraining groups which flank a protein-protein interaction site
WO1994025482A1 (fr) * 1993-04-23 1994-11-10 Evans Herbert J Polypeptides comprenant des groupes contraignant la conformation qui sont adjacents a un site d'interaction proteine-proteine
US5965698A (en) * 1993-04-23 1999-10-12 Virginia Commonwealth University Polypeptides that include conformation-constraining groups which flank a protein--protein interaction site
US6258550B1 (en) 1993-04-23 2001-07-10 Virginia Commonwealth University Polypeptides that include conformation-constraining groups which flank a protein-protein interaction site
US5928896A (en) * 1993-04-23 1999-07-27 Virginia Commonwealth University Polypeptides that include conformation-constraining groups which flank a protein--protein interaction site
US6084066A (en) * 1993-10-29 2000-07-04 Virginia Commonwealth University Polypetides that include conformation-constraining groups which flank a protein-protein interaction site

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1577115A (en) * 1976-07-27 1980-10-22 Reckitt & Colmann Prod Ltd Container closure units
CH619686A5 (en) * 1976-02-02 1980-10-15 Sandoz Ag Process for the preparation of novel peptides or peptide derivatives
DK28377A (da) * 1976-02-02 1977-08-03 Sandoz Ag Fremgangsmade til fremstilling af polypeptidderivater
US4259234A (en) * 1976-09-27 1981-03-31 Eli Lilly And Company Analgesic compounds
US4283329A (en) * 1979-12-17 1981-08-11 Eli Lilly And Company Pharmacologically active peptides

Also Published As

Publication number Publication date
GB2085892A (en) 1982-05-06
DE3164594D1 (en) 1984-08-09
IL64084A0 (en) 1982-01-31
EP0050503B1 (fr) 1984-07-04
KR830007517A (ko) 1983-10-21
US4322339A (en) 1982-03-30
AU7657581A (en) 1982-04-29
PT73840A (en) 1981-11-01
GB2085892B (en) 1984-03-07
CA1187872A (fr) 1985-05-28
FI813199L (fi) 1982-04-21
GR75824B (fr) 1984-08-02
RO83297B (ro) 1984-02-28
HU185321B (en) 1985-01-28
YU249181A (en) 1983-12-31
PL233499A1 (fr) 1982-05-24
ES8301203A1 (es) 1982-12-01
JPS57108051A (en) 1982-07-05
PL131156B1 (en) 1984-10-31
ES506315A0 (es) 1982-12-01
EP0050503A1 (fr) 1982-04-28
ZA817062B (en) 1983-05-25
ATE8252T1 (de) 1984-07-15
DK461581A (da) 1982-05-19
RO83297A (fr) 1984-02-21
PT73840B (en) 1983-01-17
NZ198626A (en) 1984-02-03

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