DD132270A5 - Verfahren zur herstellung von depot-steroidestern - Google Patents

Verfahren zur herstellung von depot-steroidestern

Info

Publication number
DD132270A5
DD132270A5 DD7600196384A DD19638476A DD132270A5 DD 132270 A5 DD132270 A5 DD 132270A5 DD 7600196384 A DD7600196384 A DD 7600196384A DD 19638476 A DD19638476 A DD 19638476A DD 132270 A5 DD132270 A5 DD 132270A5
Authority
DD
German Democratic Republic
Prior art keywords
steroidesters
depot
preparing
preparing depot
depot steroidesters
Prior art date
Application number
DD7600196384A
Other languages
German (de)
English (en)
Inventor
Paul-Eberhard Schulze
Ulrich Speck
Dieter Bittler
Rudolf Wiechert
Bernard Acksteiner
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of DD132270A5 publication Critical patent/DD132270A5/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0033Androstane derivatives substituted in position 17 alfa and 17 beta
    • C07J1/004Androstane derivatives substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0048Alkynyl derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0081Substituted in position 17 alfa and 17 beta
    • C07J1/0088Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096Alkynyl derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J11/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J21/00Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005Ketals
    • C07J21/006Ketals at position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J31/00Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C07J5/0046Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
    • C07J5/0053Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa not substituted in position 16
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J53/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002Carbocyclic rings fused
    • C07J53/0043 membered carbocyclic rings
    • C07J53/0053 membered carbocyclic rings in position 12
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J53/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002Carbocyclic rings fused
    • C07J53/0043 membered carbocyclic rings
    • C07J53/0083 membered carbocyclic rings in position 15/16

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DD7600196384A 1975-12-19 1976-12-15 Verfahren zur herstellung von depot-steroidestern DD132270A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2558076A DE2558076C2 (de) 1975-12-19 1975-12-19 Depot-Steroidester, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Präparate

Publications (1)

Publication Number Publication Date
DD132270A5 true DD132270A5 (de) 1978-09-13

Family

ID=5965325

Family Applications (1)

Application Number Title Priority Date Filing Date
DD7600196384A DD132270A5 (de) 1975-12-19 1976-12-15 Verfahren zur herstellung von depot-steroidestern

Country Status (35)

Country Link
US (1) US4119626A (pl)
JP (1) JPS5278860A (pl)
AT (1) AT357704B (pl)
AU (1) AU507111B2 (pl)
BE (1) BE849553A (pl)
BG (2) BG30475A3 (pl)
CA (1) CA1086305A (pl)
CH (1) CH630097A5 (pl)
CS (1) CS194788B2 (pl)
DD (1) DD132270A5 (pl)
DE (1) DE2558076C2 (pl)
DK (1) DK146629C (pl)
EG (1) EG12383A (pl)
ES (1) ES454297A1 (pl)
FI (1) FI57263C (pl)
FR (1) FR2335231A1 (pl)
GB (1) GB1554199A (pl)
GR (1) GR62084B (pl)
HU (1) HU179343B (pl)
IE (1) IE44320B1 (pl)
IL (1) IL50981A (pl)
IT (1) IT1065783B (pl)
LU (1) LU76398A1 (pl)
MX (1) MX3798E (pl)
NL (1) NL7614023A (pl)
NO (2) NO145620C (pl)
NZ (1) NZ182890A (pl)
PH (1) PH13907A (pl)
PL (1) PL105525B1 (pl)
PT (1) PT65973B (pl)
RO (1) RO75383A (pl)
SE (1) SE428930B (pl)
SU (1) SU648105A3 (pl)
YU (1) YU293176A (pl)
ZA (1) ZA767510B (pl)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7613248A (nl) * 1976-11-26 1978-05-30 Akzo Nv Werkwijze voor het bereiden van nieuwe steroid- esters.
DE2848423A1 (de) * 1978-11-08 1980-05-29 Merck Patent Gmbh Hydrocortisonester, diese enthaltende pharmazeutische zubereitungen und verfahren zu ihrer herstellung
US4507290A (en) * 1981-04-07 1985-03-26 World Health Organization Esters of 17 α-ethynyl 19-nor-testosterone and 17 α-ethynyl-18-homo-19-nor-testosterone and pharmaceutical compositions containing the same
DE3133082A1 (de) * 1981-08-18 1983-03-10 Schering Ag, 1000 Berlin Und 4619 Bergkamen Neue hydrocortison-derivate, ihre herstellung und verwendung
JPS59184200A (ja) * 1983-03-31 1984-10-19 Takeda Chem Ind Ltd ステロイド化合物、その製造法及び薬剤
DE3511588A1 (de) * 1985-03-27 1986-10-02 Schering AG, Berlin und Bergkamen, 1000 Berlin Waessrige kristallsuspension von steroidglykoestern
JPH02139518U (pl) * 1989-04-25 1990-11-21
DE4232521A1 (de) * 1992-09-22 1994-03-24 Schering Ag Gestagen wirksame 4,5;11,12-Estradiene, Verfahren zu ihrer Herstellung, diese Estradiene enthaltende Arzneimittel sowie deren Verwendung zur Herstellung von Arzneimitteln

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB660199A (en) * 1947-09-13 1951-10-31 Sterling Drug Inc Acyloxyalkanoates of hydroxylated hormones
GB817735A (en) * 1955-08-26 1959-08-06 Lab Francais Chimiotherapie Improvements in or relating to steroidal compounds
US3082222A (en) * 1958-03-26 1963-03-19 Ott Erwin Steroid acid-esters and salts thereof, and method of making the same
FR1326329A (fr) * 1959-10-28 1963-05-10 Préparation de sels d'hormones solubles dans l'eau et dans les lipides
US3629245A (en) * 1965-05-14 1971-12-21 Roussel Uclaf 16 17-isoxazolino-delta-1 3 5(10)-gonatrienes
US3856956A (en) * 1967-02-02 1974-12-24 Boots Pure Drug Co Ltd 17-acyloxysteroids and their manufacture
GB1253828A (en) * 1967-10-25 1971-11-17 Shionogi & Co 2,3-EPITHIO-5alpha-ANDROST-6-ENE STEROIDS
US3916002A (en) * 1973-12-17 1975-10-28 Taubert Hans Dieter Oligomeric steroid esters, process for their production, and therapeutic compositions containing the same

Also Published As

Publication number Publication date
FI57263C (fi) 1980-07-10
YU293176A (en) 1982-08-31
HU179343B (en) 1982-10-28
NO145620B (no) 1982-01-18
NO145620C (no) 1982-04-28
FR2335231B1 (pl) 1980-03-14
IE44320B1 (en) 1981-10-21
PH13907A (en) 1980-10-27
PT65973B (en) 1978-06-16
US4119626A (en) 1978-10-10
SE428930B (sv) 1983-08-01
IL50981A0 (en) 1977-01-31
DK566076A (da) 1977-06-20
NO147717C (no) 1983-06-01
DK146629C (da) 1984-04-30
BE849553A (fr) 1977-06-17
FR2335231A1 (fr) 1977-07-15
FI763544A (pl) 1977-06-20
IT1065783B (it) 1985-03-04
ES454297A1 (es) 1977-12-16
FI57263B (fi) 1980-03-31
CA1086305A (en) 1980-09-23
DK146629B (da) 1983-11-21
NZ182890A (en) 1980-05-08
GB1554199A (en) 1979-10-17
DE2558076C2 (de) 1983-12-15
PL105525B1 (pl) 1979-10-31
JPS5278860A (en) 1977-07-02
CH630097A5 (de) 1982-05-28
SE7614107L (sv) 1977-06-20
SU648105A3 (ru) 1979-02-15
IE44320L (en) 1977-06-19
ZA767510B (en) 1977-11-30
NO764284L (pl) 1977-06-21
EG12383A (en) 1979-06-30
NO803670L (no) 1977-06-21
AT357704B (de) 1980-07-25
JPS6131115B2 (pl) 1986-07-17
GR62084B (en) 1979-02-21
NL7614023A (nl) 1977-06-21
MX3798E (es) 1981-07-22
AU2073776A (en) 1978-06-29
DE2558076A1 (de) 1977-06-30
AU507111B2 (en) 1980-02-07
PT65973A (en) 1977-01-01
BG30475A3 (en) 1981-06-15
NO147717B (no) 1983-02-21
BG31504A3 (en) 1982-01-15
LU76398A1 (pl) 1977-06-10
ATA935576A (de) 1979-12-15
IL50981A (en) 1980-09-16
CS194788B2 (en) 1979-12-31
RO75383A (ro) 1980-11-30

Similar Documents

Publication Publication Date Title
DD130857A5 (de) Verfahren zur herstellung von n-phosphonomethylglycintriestern
DD129103A5 (de) Verfahren zur herstellung von n-phosphonomethylglycin
DD128681A5 (de) Verfahren zur herstellung von n hoch 2-arylsulfonyl-l-argininamiden
DD129330A5 (de) Verfahren zur herstellung von antitumorsubstanzen
DD128782A5 (de) Verfahren zur herstellung von n-alkyldiphenylaminen
AT344147B (de) Verfahren zur herstellung von acylcyaniden
DD130036A5 (de) Verfahren zur herstellung von optisch aktiven 11-desoxy-16-aryloxy-omega-tetranorprostaglandinen
ATA691376A (de) Verfahren zur herstellung von ueberzuegen
DD129326A5 (de) Verfahren zur herstellung von 1,4-diphenyl-3-pyrazolin-5-onen
ATA314576A (de) Verfahren zur herstellung von 4-nideralkyl-5- cyano-oxazolen
DD132270A5 (de) Verfahren zur herstellung von depot-steroidestern
DD131556A5 (de) Verfahren zur herstellung von 5-m-tolyoxyuracil
AT348499B (de) Verfahren zur herstellung von aethylchlorthioformiat
AT349032B (de) Verfahren zur herstellung von 4-alkyl-thiosemicarbaziden
DD132435A5 (de) Verfahren zur herstellung von indolochinolizinen
DD131562A5 (de) Verfahren zur herstellung von 5-pregnen-derivaten
DD122961A5 (de) Verfahren zur herstellung von diphenylaether-derivaten
DD132431A5 (de) Verfahren zur herstellung von aryloxy-1-amino-3-propanolen-2
AT350582B (de) Verfahren zur herstellung von n-mehtyl-harn- stoffen
AT352914B (de) Verfahren zur herstellung von polyen- verbindungen
DD131088A5 (de) Verfahren zur herstellung von diaminoalkoxybenzolen
AT376633B (de) Verfahren zur herstellung von phosphornitriden
DD128709A5 (de) Verfahren zur herstellung von dekahydrochinolinderivaten
DD128099A1 (de) Verfahren zur herstellung von allantoin
DD130416A4 (de) Verfahren zur herstellung von o-nitrobenzylbromid