CY2360B1 - Hiv protease inhibitor combination. - Google Patents

Hiv protease inhibitor combination.

Info

Publication number
CY2360B1
CY2360B1 CY0300040A CY0300040A CY2360B1 CY 2360 B1 CY2360 B1 CY 2360B1 CY 0300040 A CY0300040 A CY 0300040A CY 0300040 A CY0300040 A CY 0300040A CY 2360 B1 CY2360 B1 CY 2360B1
Authority
CY
Cyprus
Prior art keywords
hiv protease
hiv
protease inhibitor
combination
inhibitor combination
Prior art date
Application number
CY0300040A
Other languages
English (en)
Inventor
Paul J Deutsch
Emilio A Emini
Joseph P Vacca
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of CY2360B1 publication Critical patent/CY2360B1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Peptides Or Proteins (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
CY0300040A 1994-08-11 2003-05-07 Hiv protease inhibitor combination. CY2360B1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US28947494A 1994-08-11 1994-08-11
US33936994A 1994-11-14 1994-11-14
US49246195A 1995-07-20 1995-07-20

Publications (1)

Publication Number Publication Date
CY2360B1 true CY2360B1 (en) 2004-06-04

Family

ID=27403895

Family Applications (1)

Application Number Title Priority Date Filing Date
CY0300040A CY2360B1 (en) 1994-08-11 2003-05-07 Hiv protease inhibitor combination.

Country Status (20)

Country Link
EP (1) EP0774969B8 (no)
JP (1) JPH10504036A (no)
KR (1) KR970704441A (no)
CN (1) CN1101190C (no)
AT (1) ATE232727T1 (no)
AU (1) AU698664B2 (no)
CA (1) CA2197207C (no)
CY (1) CY2360B1 (no)
CZ (1) CZ292577B6 (no)
DE (1) DE69529678T2 (no)
DK (1) DK0774969T3 (no)
ES (1) ES2190456T3 (no)
FI (1) FI970565A0 (no)
HU (1) HUT76540A (no)
IL (1) IL114808A (no)
MX (1) MX9701121A (no)
NO (1) NO314168B1 (no)
PL (1) PL181578B1 (no)
SK (1) SK18197A3 (no)
WO (1) WO1996004913A1 (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA49803C2 (uk) * 1994-06-03 2002-10-15 Дж.Д. Сьорль Енд Ко Спосіб лікування ретровірусних інфекцій
US6037157A (en) * 1995-06-29 2000-03-14 Abbott Laboratories Method for improving pharmacokinetics
EP0955054A4 (en) * 1996-11-08 2003-01-29 Japan Energy Corp AIDS CURE

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US517041A (en) * 1894-03-27 Fruit-picker
CA1340588C (en) * 1988-06-13 1999-06-08 Balraj Krishan Handa Amino acid derivatives
EP0731088B1 (en) * 1990-11-19 2000-10-04 Monsanto Company Retroviral protease inhibitors
EP0554400B1 (en) * 1990-11-19 1997-07-23 Monsanto Company Retroviral protease inhibitors
IE913840A1 (en) * 1990-11-20 1992-05-20 Abbott Lab Retroviral protease inhibiting compounds
ATE163926T1 (de) * 1991-11-08 1998-03-15 Merck & Co Inc Hiv-protease-inhibitoren verwendbar in der aids- behandlung
KR100333016B1 (ko) * 1992-12-29 2002-11-22 아보트 러보러터리즈 레트로바이러스성프로테아제억제화합물,이의제조방법및이를함유하는약제학적조성물

Also Published As

Publication number Publication date
CN1160350A (zh) 1997-09-24
PL181578B1 (pl) 2001-08-31
CA2197207A1 (en) 1996-02-22
FI970565A (fi) 1997-02-10
EP0774969B1 (en) 2003-02-19
CN1101190C (zh) 2003-02-12
AU698664B2 (en) 1998-11-05
EP0774969B8 (en) 2003-07-02
MX9701121A (es) 1997-05-31
WO1996004913A1 (en) 1996-02-22
DE69529678T2 (de) 2003-09-25
EP0774969A1 (en) 1997-05-28
PL318506A1 (en) 1997-06-23
KR970704441A (ko) 1997-09-06
AU3361195A (en) 1996-03-07
NO314168B1 (no) 2003-02-10
CZ292577B6 (cs) 2003-10-15
SK18197A3 (en) 1997-09-10
IL114808A (en) 1999-10-28
CA2197207C (en) 2006-10-17
FI970565A0 (fi) 1997-02-10
NO970632D0 (no) 1997-02-11
JPH10504036A (ja) 1998-04-14
NO970632L (no) 1997-04-10
HUT76540A (en) 1997-09-29
IL114808A0 (en) 1995-12-08
CZ38997A3 (en) 1997-11-12
ES2190456T3 (es) 2003-08-01
DE69529678D1 (de) 2003-03-27
ATE232727T1 (de) 2003-03-15
DK0774969T3 (da) 2003-03-31

Similar Documents

Publication Publication Date Title
AU2725392A (en) Hiv protease inhibitors
MY109834A (en) Benzoxazinones as inhibitors of hiv reverse transcriptase
DE60036961D1 (de) Gamma-hydroxy-2-(fluoralkylaminocarbonyl)-1-piperazinpentanamide als hiv-proteasehemmer
EP0766674A4 (en) NOVEL HIV PROTEASE INHIBITORS
PL314984A1 (en) Hiv protease inhibitors
MX9705916A (es) Terapia de combinacion para infeccion por vih usando el inhibidor de proteasa de vih indinavir y el inhibidor de transcriptasa inversa 3tc, opcionalmente junto con azt, ddi, o ddc.
MX9700036A (es) Combinacion de compuestos, uso en la preparacion de composiciones para tratar infeccion por el vir s de inmunodeficiencia humana, y composiciones obtenidas.
EP0774969B8 (en) Hiv protease inhibitor combination
WO2002096359A3 (en) Piperazine pentanamide hiv protease inhibitors