CY1117021T1 - Φαρμακευτικες συνθεσεις οι οποιες περιεχουν νιλοτινιβη ή αλας αυτης - Google Patents

Φαρμακευτικες συνθεσεις οι οποιες περιεχουν νιλοτινιβη ή αλας αυτης

Info

Publication number
CY1117021T1
CY1117021T1 CY20151101150T CY151101150T CY1117021T1 CY 1117021 T1 CY1117021 T1 CY 1117021T1 CY 20151101150 T CY20151101150 T CY 20151101150T CY 151101150 T CY151101150 T CY 151101150T CY 1117021 T1 CY1117021 T1 CY 1117021T1
Authority
CY
Cyprus
Prior art keywords
salt
nilotinibe
pharmaceutical compositions
compositions containing
granules
Prior art date
Application number
CY20151101150T
Other languages
English (en)
Inventor
Nathalie Bruneau
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37684496&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1117021(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CY1117021T1 publication Critical patent/CY1117021T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1641Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • A61K9/1623Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1635Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

Μία φαρμακευτική σύνθεση, ειδικότερα κάψουλες, η οποία περιέχει κοκκία τα οποία περιέχουν νιλοτινίβη ή ένα άλας αυτής, με τουλάχιστον ένα φαρμακευτικά αποδεκτό έκδοχο. Τα κοκκία μπορούν να παράγονται δια μίας υγρής μεθόδου κοκκιοποίησης.
CY20151101150T 2006-09-27 2015-12-16 Φαρμακευτικες συνθεσεις οι οποιες περιεχουν νιλοτινιβη ή αλας αυτης CY1117021T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06121371A EP1923053A1 (en) 2006-09-27 2006-09-27 Pharmaceutical compositions comprising nilotinib or its salt
EP07820560.6A EP2068839B2 (en) 2006-09-27 2007-09-25 Pharmaceutical compositions comprising nilotinib or its salt

Publications (1)

Publication Number Publication Date
CY1117021T1 true CY1117021T1 (el) 2017-04-05

Family

ID=37684496

Family Applications (2)

Application Number Title Priority Date Filing Date
CY20151101150T CY1117021T1 (el) 2006-09-27 2015-12-16 Φαρμακευτικες συνθεσεις οι οποιες περιεχουν νιλοτινιβη ή αλας αυτης
CY20231100367T CY1126116T1 (el) 2006-09-27 2023-07-27 Φαρμακευτικες συνθεσεις αποτελουμενες απο νιλοτινιμπη

Family Applications After (1)

Application Number Title Priority Date Filing Date
CY20231100367T CY1126116T1 (el) 2006-09-27 2023-07-27 Φαρμακευτικες συνθεσεις αποτελουμενες απο νιλοτινιμπη

Country Status (35)

Country Link
US (2) US8293756B2 (el)
EP (4) EP1923053A1 (el)
JP (2) JP5567340B2 (el)
KR (2) KR20090076931A (el)
CN (2) CN101516344A (el)
AR (1) AR062980A1 (el)
AU (1) AU2007301977B2 (el)
BR (1) BRPI0719438B1 (el)
CA (1) CA2662571C (el)
CL (1) CL2007002766A1 (el)
CO (1) CO6160288A2 (el)
CY (2) CY1117021T1 (el)
DK (2) DK3984528T3 (el)
ES (3) ES2957912T3 (el)
FI (2) FI2068839T4 (el)
HK (1) HK1133193A1 (el)
HR (2) HRP20230753T3 (el)
HU (2) HUE028204T2 (el)
IL (1) IL197496A (el)
JO (1) JO3757B1 (el)
LT (1) LT3984528T (el)
MA (1) MA30807B1 (el)
MX (1) MX2009003184A (el)
MY (1) MY148237A (el)
NO (2) NO347404B1 (el)
NZ (1) NZ575317A (el)
PE (2) PE20081379A1 (el)
PL (2) PL3984528T3 (el)
PT (2) PT3984528T (el)
RU (1) RU2469707C2 (el)
SI (2) SI3984528T1 (el)
TN (1) TN2009000093A1 (el)
TW (3) TW201418245A (el)
WO (1) WO2008037716A2 (el)
ZA (1) ZA200901511B (el)

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Also Published As

Publication number Publication date
IL197496A (en) 2016-04-21
HRP20151383T4 (hr) 2023-03-03
US20130023549A1 (en) 2013-01-24
EP3984528A1 (en) 2022-04-20
SI3984528T1 (sl) 2023-09-29
DK2068839T3 (da) 2016-01-11
BRPI0719438B1 (pt) 2022-04-19
CY1126116T1 (el) 2023-11-15
MY148237A (en) 2013-03-29
BRPI0719438A2 (pt) 2013-12-10
ES2957912T3 (es) 2024-01-29
EP3009128A1 (en) 2016-04-20
JO3757B1 (ar) 2021-01-31
ES2556625T5 (es) 2023-03-02
EP2068839B2 (en) 2022-10-12
JP2010504942A (ja) 2010-02-18
AU2007301977B2 (en) 2011-09-08
SI2068839T2 (sl) 2023-01-31
CA2662571A1 (en) 2008-04-03
LT3984528T (lt) 2023-08-10
RU2469707C2 (ru) 2012-12-20
FI2068839T4 (fi) 2023-01-31
HUE063083T2 (hu) 2023-12-28
KR20140121903A (ko) 2014-10-16
CA2662571C (en) 2016-09-27
NO20220946A1 (no) 2009-04-24
AU2007301977A1 (en) 2008-04-03
CO6160288A2 (es) 2010-05-20
KR101598747B1 (ko) 2016-03-02
PL3984528T3 (pl) 2023-08-28
EP2068839A2 (en) 2009-06-17
RU2009115782A (ru) 2010-11-10
MA30807B1 (fr) 2009-10-01
CN104306350A (zh) 2015-01-28
ES2556625T3 (es) 2016-01-19
TW200821298A (en) 2008-05-16
HRP20151383T1 (hr) 2016-01-15
ZA200901511B (en) 2010-02-24
US20100087463A1 (en) 2010-04-08
NO20091501L (no) 2009-04-24
PE20081379A1 (es) 2008-11-27
JP5567340B2 (ja) 2014-08-06
HUE028204T2 (en) 2016-12-28
CL2007002766A1 (es) 2008-08-08
TWI540128B (zh) 2016-07-01
IL197496A0 (en) 2009-12-24
US8501760B2 (en) 2013-08-06
KR20090076931A (ko) 2009-07-13
ES2951547T3 (es) 2023-10-23
TWI428333B (zh) 2014-03-01
EP2068839B1 (en) 2015-09-23
TW201418245A (zh) 2014-05-16
PL2068839T3 (pl) 2016-06-30
MX2009003184A (es) 2009-04-03
PT2068839E (pt) 2015-12-30
EP1923053A1 (en) 2008-05-21
WO2008037716A3 (en) 2008-07-17
NO346639B1 (no) 2022-11-07
PT3984528T (pt) 2023-08-07
EP3984528B1 (en) 2023-07-05
JP2014065715A (ja) 2014-04-17
NZ575317A (en) 2011-12-22
AR062980A1 (es) 2008-12-17
DK3984528T3 (da) 2023-07-31
HK1133193A1 (en) 2010-03-19
EP3009128B1 (en) 2023-07-05
TN2009000093A1 (en) 2010-08-19
US8293756B2 (en) 2012-10-23
HRP20230753T3 (hr) 2023-10-27
PE20120626A1 (es) 2012-06-07
NO347404B1 (no) 2023-10-16
SI2068839T1 (sl) 2016-02-29
TW201418244A (zh) 2014-05-16
WO2008037716A2 (en) 2008-04-03
FI3984528T3 (fi) 2023-07-27
CN101516344A (zh) 2009-08-26
PL2068839T5 (pl) 2023-01-30

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