CY1112107T1 - Νεα ενωση πυριδαζινης και χρηση αυτης - Google Patents

Νεα ενωση πυριδαζινης και χρηση αυτης

Info

Publication number
CY1112107T1
CY1112107T1 CY20101100287T CY101100287T CY1112107T1 CY 1112107 T1 CY1112107 T1 CY 1112107T1 CY 20101100287 T CY20101100287 T CY 20101100287T CY 101100287 T CY101100287 T CY 101100287T CY 1112107 T1 CY1112107 T1 CY 1112107T1
Authority
CY
Cyprus
Prior art keywords
union
pyridazin
new
new pyridazin
compound
Prior art date
Application number
CY20101100287T
Other languages
English (en)
Inventor
Steven S Bondy
Terrence C Dahl
David A Oare
Reza Oliyai
Winston C Tse
Vahid Zia
Original Assignee
Gilead Sciences, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences, Inc. filed Critical Gilead Sciences, Inc.
Publication of CY1112107T1 publication Critical patent/CY1112107T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Ένωση του τύπου (1) και άλατα και διαλυτώματα αυτής παρέχονται για τη θεραπεία ή την προφύλαξη μολύνσεων ιού ηπατίτιδας C. Παρέχονται μέθοδοι κατασκευής και τυποποίησης της ένωσης (1).
CY20101100287T 2006-07-07 2010-03-29 Νεα ενωση πυριδαζινης και χρηση αυτης CY1112107T1 (el)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US81928906P 2006-07-07 2006-07-07
US83240306P 2006-07-21 2006-07-21
US83276906P 2006-07-24 2006-07-24
EP07796714A EP2038275B1 (en) 2006-07-07 2007-07-06 Novel pyridazine compound and use thereof

Publications (1)

Publication Number Publication Date
CY1112107T1 true CY1112107T1 (el) 2015-11-04

Family

ID=38814329

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20101100287T CY1112107T1 (el) 2006-07-07 2010-03-29 Νεα ενωση πυριδαζινης και χρηση αυτης

Country Status (28)

Country Link
US (3) US8569487B2 (el)
EP (1) EP2038275B1 (el)
JP (1) JP4958974B2 (el)
KR (1) KR101143596B1 (el)
CN (1) CN102617571B (el)
AP (1) AP3430A (el)
AR (1) AR061969A1 (el)
AT (1) ATE454384T1 (el)
AU (1) AU2007269614B2 (el)
CA (1) CA2656415C (el)
CY (1) CY1112107T1 (el)
DE (1) DE602007004220D1 (el)
DK (1) DK2038275T3 (el)
EA (1) EA019452B1 (el)
ES (1) ES2339298T3 (el)
HK (1) HK1123803A1 (el)
HR (2) HRP20090078A2 (el)
IL (1) IL195528A (el)
MX (1) MX2009000235A (el)
NO (1) NO20090595L (el)
NZ (1) NZ574312A (el)
PL (1) PL2038275T3 (el)
PT (1) PT2038275E (el)
RS (1) RS51336B (el)
SG (1) SG175604A1 (el)
SI (1) SI2038275T1 (el)
TW (1) TWI360549B (el)
WO (1) WO2008005519A2 (el)

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JP5639762B2 (ja) 2006-12-14 2014-12-10 ギリアード サイエンシーズ， インコーポレイテッド ウイルス阻害剤
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TW201105323A (en) 2009-06-23 2011-02-16 Gilead Sciences Inc Pharmaceutical compositions useful for treating HCV
TW201113279A (en) 2009-06-23 2011-04-16 Gilead Sciences Inc Pharmaceutical compositions useful for treating HCV
WO2011053617A1 (en) 2009-10-30 2011-05-05 Boehringer Ingelheim International Gmbh Dosage regimens for hcv combination therapy comprising bi201335, interferon alpha and ribavirin
MX2012007076A (es) * 2009-12-18 2012-07-20 Boehringer Ingelheim Int Terapia combinada de hcv.
EP2571882A1 (en) 2010-05-21 2013-03-27 Gilead Sciences, Inc. Heterocyclic flaviviridae virus inhibitors
TW201211047A (en) * 2010-06-10 2012-03-16 Gilead Sciences Inc Methods for treating HCV
NZ613370A (en) 2010-12-20 2015-05-29 Gilead Sciences Inc Combinations for treating hcv
JP6042412B2 (ja) 2011-04-28 2016-12-14 オンコペプティデス エービーＯｎｃｏｐｅｐｔｉｄｅｓ ＡＢ 細胞毒性ジペプチドの凍結乾燥調製物
SI2709613T2 (sl) 2011-09-16 2020-12-31 Gilead Pharmasset LLC c/o Gilead Sciences, Inc. Postopki za zdravljenje HCV
EP2928463B1 (en) * 2012-10-26 2019-11-20 Oncopeptides AB Lyophilized preparations of melphalan flufenamide
SG11201506021XA (en) 2013-01-31 2015-08-28 Gilead Pharmasset Llc Combination formulation of two antiviral compounds
RS62434B1 (sr) 2014-12-26 2021-11-30 Univ Emory Antivirusni n4-hidroksicitidin derivati
KR102626210B1 (ko) 2017-12-07 2024-01-18 에모리 유니버시티 N4-하이드록시사이티딘 및 유도체 및 이와 관련된 항-바이러스 용도

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