CY1108843T1 - 3,11β cis διϋδροτετραβεναζινη για την θεραπεια της σχιζοφρενιας και αλλων ψυχωσεων - Google Patents
3,11β cis διϋδροτετραβεναζινη για την θεραπεια της σχιζοφρενιας και αλλων ψυχωσεωνInfo
- Publication number
- CY1108843T1 CY1108843T1 CY20091100221T CY091100221T CY1108843T1 CY 1108843 T1 CY1108843 T1 CY 1108843T1 CY 20091100221 T CY20091100221 T CY 20091100221T CY 091100221 T CY091100221 T CY 091100221T CY 1108843 T1 CY1108843 T1 CY 1108843T1
- Authority
- CY
- Cyprus
- Prior art keywords
- schizophrenia
- cis
- treatment
- dimrodetretravenasine
- psychologies
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/473—Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- General Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Organic Chemistry (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Saccharide Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Η εφεύρεση παρέχει την χρήση της 3,11b-cis-διϋδροτετραβεναζίνης ή ενός φαρμακευτικώς αποδεκτού άλατος αυτής για την κατασκευή ενός φαρμάκου για την προφύλαξη ή την θεραπεία της σχιζοφρένιας και άλλων ψυχώσεων.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0516167.4A GB0516167D0 (en) | 2005-08-06 | 2005-08-06 | Pharmaceutical compounds |
GB0516790A GB0516790D0 (en) | 2005-08-16 | 2005-08-16 | Pharmaceutical compounds |
EP06765238A EP1855677B1 (en) | 2005-08-06 | 2006-08-04 | 3,11b cis dihydrotetrabanezine for the treatment of schizophrenia and other psychoses |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1108843T1 true CY1108843T1 (el) | 2014-07-02 |
Family
ID=37400949
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20091100221T CY1108843T1 (el) | 2005-08-06 | 2009-02-26 | 3,11β cis διϋδροτετραβεναζινη για την θεραπεια της σχιζοφρενιας και αλλων ψυχωσεων |
Country Status (21)
Country | Link |
---|---|
US (1) | US20110257220A1 (el) |
EP (2) | EP1855677B1 (el) |
JP (1) | JP2009504622A (el) |
KR (1) | KR20080033500A (el) |
AT (2) | ATE534391T1 (el) |
AU (1) | AU2006277753B2 (el) |
CA (1) | CA2620960A1 (el) |
CY (1) | CY1108843T1 (el) |
DE (1) | DE602006004009D1 (el) |
DK (1) | DK1855677T3 (el) |
ES (1) | ES2318771T3 (el) |
HK (1) | HK1111083A1 (el) |
HR (1) | HRP20090074T3 (el) |
MX (1) | MX2008001549A (el) |
NZ (1) | NZ566011A (el) |
PL (1) | PL1855677T3 (el) |
PT (1) | PT1855677E (el) |
RS (1) | RS50807B (el) |
RU (1) | RU2407743C2 (el) |
SI (1) | SI1855677T1 (el) |
WO (1) | WO2007017654A1 (el) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK2081929T3 (da) | 2006-11-08 | 2013-04-15 | Neurocrine Biosciences Inc | Substituerede 3-isobutyl-9,10-dimethoxy-1,3,4,6,7,11B-hexahydro-2H-pyrido[2,1-A]isoquinolin-2-ol-forbindelser og fremgangsmåder angående disse |
US8008500B2 (en) | 2007-06-08 | 2011-08-30 | General Electric Company | Intermediates useful for making tetrabenazine compounds |
US8053578B2 (en) | 2007-11-29 | 2011-11-08 | General Electric Company | Alpha-fluoroalkyl dihydrotetrabenazine imaging agents and probes |
GB0810857D0 (en) * | 2008-06-13 | 2008-07-23 | Cambridge Lab Ireland Ltd | Pharmaceutical compounds |
GB2463451A (en) | 2008-09-08 | 2010-03-17 | Cambridge Lab | 3, 11b cis-dihydrotetrabenazine compounds for use in the treatment of dementia |
GB2463283A (en) * | 2008-09-08 | 2010-03-10 | Cambridge Lab | 3,11b-cis-dihydrotetrabenazine for use in treating asthma |
CA2801061A1 (en) | 2010-06-01 | 2011-12-08 | Auspex Pharmaceuticals, Inc. | Benzoquinolone inhibitors of vmat2 |
KR101882044B1 (ko) | 2011-04-01 | 2018-07-25 | 쓰리엠 이노베이티브 프로퍼티즈 캄파니 | 트라이아진계 자외선 흡수제를 포함하는 필름 |
US20160346270A1 (en) | 2014-01-27 | 2016-12-01 | Auspex Pharmaceuticals, Inc. | Benzoquinoline inhibitors of vesicular monoamine transporter 2 |
JP6718376B2 (ja) * | 2014-02-07 | 2020-07-08 | ニューロクライン バイオサイエンシーズ,インコーポレイテッド | 抗精神病薬物およびvmat2阻害剤を含む医薬組成物およびその使用 |
EP3368534B1 (en) | 2015-10-30 | 2021-01-27 | Neurocrine Biosciences, Inc. | Valbenazine ditosylate and polymorphs thereof |
HRP20220621T1 (hr) | 2015-12-23 | 2022-06-24 | Neurocrine Biosciences, Inc. | Postupak sinteze za proizvodnju (s)-(2r,3r,11br)-3-izobutil-9,10-dimetoksi-2,3,4,6,7,11b-heksahidro-1h-pirido[2,1-a]izokinolin-2-il 2-amino-3-metilbutanoat di(4-metilbenzensulfonata) |
JP2020500875A (ja) * | 2016-12-02 | 2020-01-16 | ニューロクライン バイオサイエンシーズ,インコーポレイテッド | 統合失調症または統合失調感情障害を処置するためのバルベナジンの使用 |
CA3051832A1 (en) | 2017-01-27 | 2018-08-02 | Neurocrine Bioscienes, Inc. | Methods for the administration of certain vmat2 inhibitors |
GB201705304D0 (en) | 2017-04-01 | 2017-05-17 | Adeptio Pharmaceuticals Ltd | Pharmaceutical compositions |
GB201705302D0 (en) * | 2017-04-01 | 2017-05-17 | Adeptio Pharmaceuticals Ltd | Pharmaceutical compositions |
GB201705303D0 (en) | 2017-04-01 | 2017-05-17 | Adeptio Pharmaceuticals Ltd | Pharmaceutical compositions |
GB201705306D0 (en) | 2017-04-01 | 2017-05-17 | Adeptio Pharmaceuticals Ltd | Pharmaceutical compositions |
EP3684333A2 (en) | 2017-09-21 | 2020-07-29 | Neurocrine Biosciences, Inc. | High dosage valbenazine formulation and compositions, methods, and kits related thereto |
US10993941B2 (en) | 2017-10-10 | 2021-05-04 | Neurocrine Biosciences, Inc. | Methods for the administration of certain VMAT2 inhibitors |
CN111836543A (zh) | 2017-10-10 | 2020-10-27 | 纽罗克里生物科学有限公司 | 施用某些vmat2抑制剂的方法 |
WO2020037022A1 (en) | 2018-08-15 | 2020-02-20 | Neurocrine Biosciences, Inc. | Methods for the administration of certain vmat2 inhibitors |
US10940141B1 (en) | 2019-08-23 | 2021-03-09 | Neurocrine Biosciences, Inc. | Methods for the administration of certain VMAT2 inhibitors |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2830993A (en) | 1958-04-15 | Quinolizine derivatives | ||
US2843591A (en) * | 1958-07-15 | Method for preparing same | ||
US6087376A (en) * | 1997-02-05 | 2000-07-11 | University Of Kentucky Research Foundation | Use of lobeline compounds in the treatment of central nervous system diseases and pathologies |
GB2410947B (en) * | 2004-02-11 | 2008-09-17 | Cambridge Lab Ltd | Pharmaceutical compounds |
-
2006
- 2006-08-04 KR KR1020087005308A patent/KR20080033500A/ko not_active Application Discontinuation
- 2006-08-04 RS RSP-2009/0055A patent/RS50807B/sr unknown
- 2006-08-04 AT AT08170385T patent/ATE534391T1/de active
- 2006-08-04 WO PCT/GB2006/002936 patent/WO2007017654A1/en active Application Filing
- 2006-08-04 CA CA002620960A patent/CA2620960A1/en not_active Abandoned
- 2006-08-04 MX MX2008001549A patent/MX2008001549A/es active IP Right Grant
- 2006-08-04 PL PL06765238T patent/PL1855677T3/pl unknown
- 2006-08-04 EP EP06765238A patent/EP1855677B1/en active Active
- 2006-08-04 DE DE602006004009T patent/DE602006004009D1/de active Active
- 2006-08-04 EP EP08170385A patent/EP2050451B1/en active Active
- 2006-08-04 DK DK06765238T patent/DK1855677T3/da active
- 2006-08-04 PT PT06765238T patent/PT1855677E/pt unknown
- 2006-08-04 AT AT06765238T patent/ATE415968T1/de active
- 2006-08-04 AU AU2006277753A patent/AU2006277753B2/en not_active Expired - Fee Related
- 2006-08-04 RU RU2008108623/04A patent/RU2407743C2/ru not_active IP Right Cessation
- 2006-08-04 JP JP2008525620A patent/JP2009504622A/ja not_active Ceased
- 2006-08-04 US US11/997,591 patent/US20110257220A1/en not_active Abandoned
- 2006-08-04 NZ NZ566011A patent/NZ566011A/en not_active IP Right Cessation
- 2006-08-04 SI SI200630210T patent/SI1855677T1/sl unknown
- 2006-08-04 ES ES06765238T patent/ES2318771T3/es active Active
-
2008
- 2008-05-20 HK HK08105580.7A patent/HK1111083A1/xx not_active IP Right Cessation
-
2009
- 2009-02-06 HR HR20090074T patent/HRP20090074T3/xx unknown
- 2009-02-26 CY CY20091100221T patent/CY1108843T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
EP2050451B1 (en) | 2011-11-23 |
KR20080033500A (ko) | 2008-04-16 |
MX2008001549A (es) | 2008-04-04 |
US20110257220A1 (en) | 2011-10-20 |
AU2006277753A1 (en) | 2007-02-15 |
NZ566011A (en) | 2011-01-28 |
EP1855677B1 (en) | 2008-12-03 |
ATE415968T1 (de) | 2008-12-15 |
JP2009504622A (ja) | 2009-02-05 |
EP2050451A1 (en) | 2009-04-22 |
RS50807B (sr) | 2010-08-31 |
RU2008108623A (ru) | 2009-09-20 |
HRP20090074T3 (en) | 2009-04-30 |
HK1111083A1 (en) | 2008-08-01 |
EP1855677A1 (en) | 2007-11-21 |
WO2007017654A1 (en) | 2007-02-15 |
PL1855677T3 (pl) | 2009-07-31 |
CA2620960A1 (en) | 2007-02-15 |
SI1855677T1 (sl) | 2009-04-30 |
AU2006277753B2 (en) | 2011-11-10 |
PT1855677E (pt) | 2009-01-13 |
ATE534391T1 (de) | 2011-12-15 |
ES2318771T3 (es) | 2009-05-01 |
DK1855677T3 (da) | 2009-02-09 |
RU2407743C2 (ru) | 2010-12-27 |
DE602006004009D1 (de) | 2009-01-15 |
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