CY1107714T1 - Φαρμακευτικες συνθεσεις μοδαφινιλιου - Google Patents

Φαρμακευτικες συνθεσεις μοδαφινιλιου

Info

Publication number
CY1107714T1
CY1107714T1 CY20071101071T CY071101071T CY1107714T1 CY 1107714 T1 CY1107714 T1 CY 1107714T1 CY 20071101071 T CY20071101071 T CY 20071101071T CY 071101071 T CY071101071 T CY 071101071T CY 1107714 T1 CY1107714 T1 CY 1107714T1
Authority
CY
Cyprus
Prior art keywords
pharmaceutical compositions
modufinilium
modafinil
potency
drug
Prior art date
Application number
CY20071101071T
Other languages
English (en)
Inventor
Craig Heacock
Alpa Parikh
Piyush R Patel
Original Assignee
Cephalon, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=30118520&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1107714(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Cephalon, Inc. filed Critical Cephalon, Inc.
Publication of CY1107714T1 publication Critical patent/CY1107714T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Φαρμακευτικές συνθέσεις περιλαμβάνουν μοδαφινίλιο σε μορφή σωματιδίων καθορισμένου μεγέθους. Το μέγεθος των σωματιδίων του μοδαφινιλίου μπορεί να έχει σημαντική επίδραση στη δραστικότητα και το ασφαλές προφίλ του φαρμάκου.
CY20071101071T 2002-07-12 2007-08-09 Φαρμακευτικες συνθεσεις μοδαφινιλιου CY1107714T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US39553702P 2002-07-12 2002-07-12
US10/616,776 US20040048931A1 (en) 2002-07-12 2003-07-10 Modafinil pharmaceutical compositions
EP03764620A EP1542666B1 (en) 2002-07-12 2003-07-11 Modafinil pharmaceutical compositions

Publications (1)

Publication Number Publication Date
CY1107714T1 true CY1107714T1 (el) 2013-04-18

Family

ID=30118520

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20071101071T CY1107714T1 (el) 2002-07-12 2007-08-09 Φαρμακευτικες συνθεσεις μοδαφινιλιου

Country Status (24)

Country Link
US (2) US20040048931A1 (el)
EP (1) EP1542666B1 (el)
JP (1) JP4902959B2 (el)
KR (2) KR101163768B1 (el)
CN (1) CN100423716C (el)
AT (1) ATE363899T1 (el)
AU (1) AU2003259128B2 (el)
BR (1) BR0312619A (el)
CA (1) CA2491317C (el)
CY (1) CY1107714T1 (el)
DE (1) DE60314265T2 (el)
DK (1) DK1542666T3 (el)
EA (2) EA200600968A1 (el)
ES (1) ES2285189T3 (el)
HK (1) HK1077195A1 (el)
IL (1) IL165835A0 (el)
IS (1) IS2516B (el)
MX (1) MXPA05000373A (el)
NO (1) NO334450B1 (el)
NZ (1) NZ537627A (el)
PL (1) PL216994B1 (el)
PT (1) PT1542666E (el)
TW (1) TW200407111A (el)
WO (1) WO2004006905A1 (el)

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US7368591B2 (en) 2003-09-19 2008-05-06 Cephalon France Process for enantioselective synthesis of single enantiomers of modafinil by asymmetric oxidation
EP1516869A1 (en) 2003-09-19 2005-03-23 Cephalon France Process for enantioselective synthesis of single enantiomers of modafinil by asymmetric oxidation
US20050137264A1 (en) * 2003-12-22 2005-06-23 Patel Ashish A. Modafinil compositions
US20060024370A1 (en) 2004-07-29 2006-02-02 Cephalon France Modafinil oral lyophilizate
WO2007013962A2 (en) * 2005-07-21 2007-02-01 Neurohealing Pharmaceuticals, Inc. Rapid onset and short term modafinil compositions and methods of use thereof
BRPI0614701A2 (pt) * 2005-07-29 2011-04-12 Vanda Pharmaceuticals Inc usos de um composto para melhorar a vigìlia e composições farmacêuticas
WO2007098446A2 (en) * 2006-02-21 2007-08-30 Accu-Break Pharmaceuticals, Inc. Method for minimizing variation in dosage forms
AU2007272501A1 (en) * 2006-07-12 2008-01-17 Elan Pharma International Limited Nanoparticulate formulations of modafinil
EP2056811B8 (en) * 2006-08-14 2018-03-21 Neurohealing Pharmaceuticals, Inc. Modafinil-based treatment for premature ejaculation
US8173169B2 (en) * 2007-07-11 2012-05-08 Hikma Pharmaceuticals Formulation and process for the preparation of modafinil
ES2451540T3 (es) * 2008-12-03 2014-03-27 Astellas Deutschland Gmbh Formas de dosificación oral de bendamustina
EP2517704B1 (en) * 2009-12-25 2019-05-01 Innopharmax, Inc. Pharmaceutical composition for treating parkinson's disease and preparation method thereof
FR2987266B1 (fr) 2012-02-28 2014-12-19 Debregeas Et Associes Pharma Procede d'obtention d'une composition pharmaceutique a base de modafinil, composition pharmaceutique ainsi obtenue et son application
US10058542B1 (en) 2014-09-12 2018-08-28 Thioredoxin Systems Ab Composition comprising selenazol or thiazolone derivatives and silver and method of treatment therewith
WO2022007578A1 (zh) * 2020-07-10 2022-01-13 广州新创忆药物临床研究有限公司 治疗阿尔茨海默病的组合及其应用

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Also Published As

Publication number Publication date
NO20045533L (no) 2005-02-11
EA007562B1 (ru) 2006-12-29
NZ537627A (en) 2006-11-30
US20040048931A1 (en) 2004-03-11
KR101163768B1 (ko) 2012-07-06
EA200500190A1 (ru) 2005-06-30
CA2491317A1 (en) 2004-01-22
BR0312619A (pt) 2005-04-19
IS7595A (is) 2004-12-13
HK1077195A1 (en) 2006-02-10
JP4902959B2 (ja) 2012-03-21
PT1542666E (pt) 2007-07-18
US8580308B2 (en) 2013-11-12
PL372615A1 (en) 2005-07-25
EP1542666A1 (en) 2005-06-22
KR20110092361A (ko) 2011-08-17
WO2004006905A1 (en) 2004-01-22
CA2491317C (en) 2011-12-06
AU2003259128A1 (en) 2004-02-02
ATE363899T1 (de) 2007-06-15
PL216994B1 (pl) 2014-06-30
MXPA05000373A (es) 2005-03-31
TW200407111A (en) 2004-05-16
JP2005533114A (ja) 2005-11-04
DE60314265T2 (de) 2008-01-31
IL165835A0 (en) 2006-01-15
DK1542666T3 (da) 2007-09-17
IS2516B (is) 2009-06-15
NO334450B1 (no) 2014-03-03
EP1542666B1 (en) 2007-06-06
KR20050026475A (ko) 2005-03-15
ES2285189T3 (es) 2007-11-16
EA200600968A1 (ru) 2007-02-27
DE60314265D1 (de) 2007-07-19
US20070065517A1 (en) 2007-03-22
CN100423716C (zh) 2008-10-08
CN1668289A (zh) 2005-09-14
AU2003259128B2 (en) 2008-12-04

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