BR0312619A - Composição farmacêutica, método para formular uma composição de modafinil, unidade de dosagem farmacêutica, e, métodos para alterar o estado sonolento de um mamìfero, intensificar a condição de atividade ou aumentar a regularidade da periodicidade do sono - Google Patents

Composição farmacêutica, método para formular uma composição de modafinil, unidade de dosagem farmacêutica, e, métodos para alterar o estado sonolento de um mamìfero, intensificar a condição de atividade ou aumentar a regularidade da periodicidade do sono

Info

Publication number
BR0312619A
BR0312619A BR0312619-6A BR0312619A BR0312619A BR 0312619 A BR0312619 A BR 0312619A BR 0312619 A BR0312619 A BR 0312619A BR 0312619 A BR0312619 A BR 0312619A
Authority
BR
Brazil
Prior art keywords
composition
methods
regularity
formulating
altering
Prior art date
Application number
BR0312619-6A
Other languages
English (en)
Inventor
Craig Heacock
Alpa Parikh
Piyush R Patel
Original Assignee
Cephalon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=30118520&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR0312619(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Cephalon Inc filed Critical Cephalon Inc
Publication of BR0312619A publication Critical patent/BR0312619A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Pulmonology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

"COMPOSIçãO FARMACêUTICA, MéTODO PARA FORMULAR UMA COMPOSIçãO DE, MODAFINIL, UNIDADE DE DOSAGEM FARMACêUTICA, E MéTODOS PARA ALTERAR O ESTADO SONOLENTO DE UM MAMìFERO, INTENSIFICAR A CONDIçãO DE ATIVIDADE OU AUMENTAR A REGULARIDADE DA PERIODICIDADE DO SONO". Expõem-se composições farmacêuticas que compreendem modafinil na forma de partículas de dimensão definida. A dimensão de partícula de modafinil pode ter um efeito significativo no perfil de potência e segurança da droga.
BR0312619-6A 2002-07-12 2003-07-11 Composição farmacêutica, método para formular uma composição de modafinil, unidade de dosagem farmacêutica, e, métodos para alterar o estado sonolento de um mamìfero, intensificar a condição de atividade ou aumentar a regularidade da periodicidade do sono BR0312619A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US39553702P 2002-07-12 2002-07-12
US10/616,776 US20040048931A1 (en) 2002-07-12 2003-07-10 Modafinil pharmaceutical compositions
PCT/US2003/021969 WO2004006905A1 (en) 2002-07-12 2003-07-11 Modafinil pharmaceutical compositions

Publications (1)

Publication Number Publication Date
BR0312619A true BR0312619A (pt) 2005-04-19

Family

ID=30118520

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0312619-6A BR0312619A (pt) 2002-07-12 2003-07-11 Composição farmacêutica, método para formular uma composição de modafinil, unidade de dosagem farmacêutica, e, métodos para alterar o estado sonolento de um mamìfero, intensificar a condição de atividade ou aumentar a regularidade da periodicidade do sono

Country Status (24)

Country Link
US (2) US20040048931A1 (pt)
EP (1) EP1542666B1 (pt)
JP (1) JP4902959B2 (pt)
KR (2) KR101163768B1 (pt)
CN (1) CN100423716C (pt)
AT (1) ATE363899T1 (pt)
AU (1) AU2003259128B2 (pt)
BR (1) BR0312619A (pt)
CA (1) CA2491317C (pt)
CY (1) CY1107714T1 (pt)
DE (1) DE60314265T2 (pt)
DK (1) DK1542666T3 (pt)
EA (2) EA200600968A1 (pt)
ES (1) ES2285189T3 (pt)
HK (1) HK1077195A1 (pt)
IL (1) IL165835A0 (pt)
IS (1) IS2516B (pt)
MX (1) MXPA05000373A (pt)
NO (1) NO334450B1 (pt)
NZ (1) NZ537627A (pt)
PL (1) PL216994B1 (pt)
PT (1) PT1542666E (pt)
TW (1) TW200407111A (pt)
WO (1) WO2004006905A1 (pt)

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KR20060024028A (ko) 2000-07-27 2006-03-15 테바 파마슈티컬 인더스트리즈 리미티드 결정질의 순수한 모다피닐 및 이의 제조 방법
US6919378B2 (en) 2000-10-11 2005-07-19 Cephalon, Inc. Pharmaceutical solutions of modafinil compounds
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FR2849029B1 (fr) 2002-12-20 2005-03-18 Lafon Labor Procede de preparation et formes cristallines des enantiomeres optiques du modafinil.
CA2420180A1 (en) * 2003-02-28 2004-08-28 Bernard Charles Sherman Tablets comprising modafinil
US20070066996A1 (en) * 2003-03-17 2007-03-22 Katzman Daniel E Modafinil-based neurorehabilitation of impaired neurological function associated with brian injury
US20040253308A1 (en) * 2003-04-29 2004-12-16 Barr Laboratories, Inc. Surface-treated modafinil particles
EP1516869A1 (en) 2003-09-19 2005-03-23 Cephalon France Process for enantioselective synthesis of single enantiomers of modafinil by asymmetric oxidation
US7368591B2 (en) 2003-09-19 2008-05-06 Cephalon France Process for enantioselective synthesis of single enantiomers of modafinil by asymmetric oxidation
US20050137264A1 (en) * 2003-12-22 2005-06-23 Patel Ashish A. Modafinil compositions
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EP1909573A4 (en) * 2005-07-21 2010-09-22 Neurohealing Pharmaceuticals I SHORT-TERM EFFECTIVE MODAFINIL COMPOSITIONS WITH A RAPID INITIAL EFFECT, AND METHOD FOR THEIR USE
EP1919477B1 (en) * 2005-07-29 2012-07-11 Vanda Pharmaceuticals Inc. Use of [2-(2-methylimidazol-1-yl)methyl]pyridine for treating sleep disorders
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US8173169B2 (en) * 2007-07-11 2012-05-08 Hikma Pharmaceuticals Formulation and process for the preparation of modafinil
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JP5718937B2 (ja) * 2009-12-25 2015-05-13 イノファーマックス インコーポレイテッド パーキンソン病を治療するための医薬組成物及びその調製方法
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Also Published As

Publication number Publication date
KR20110092361A (ko) 2011-08-17
PL372615A1 (en) 2005-07-25
EA200500190A1 (ru) 2005-06-30
ATE363899T1 (de) 2007-06-15
WO2004006905A1 (en) 2004-01-22
NO20045533L (no) 2005-02-11
EA007562B1 (ru) 2006-12-29
IS2516B (is) 2009-06-15
PL216994B1 (pl) 2014-06-30
JP4902959B2 (ja) 2012-03-21
AU2003259128B2 (en) 2008-12-04
JP2005533114A (ja) 2005-11-04
DK1542666T3 (da) 2007-09-17
KR101163768B1 (ko) 2012-07-06
EP1542666A1 (en) 2005-06-22
DE60314265T2 (de) 2008-01-31
CY1107714T1 (el) 2013-04-18
HK1077195A1 (en) 2006-02-10
KR20050026475A (ko) 2005-03-15
CN1668289A (zh) 2005-09-14
MXPA05000373A (es) 2005-03-31
DE60314265D1 (de) 2007-07-19
TW200407111A (en) 2004-05-16
AU2003259128A1 (en) 2004-02-02
CA2491317A1 (en) 2004-01-22
ES2285189T3 (es) 2007-11-16
EP1542666B1 (en) 2007-06-06
IS7595A (is) 2004-12-13
CA2491317C (en) 2011-12-06
US20070065517A1 (en) 2007-03-22
NO334450B1 (no) 2014-03-03
US20040048931A1 (en) 2004-03-11
PT1542666E (pt) 2007-07-18
CN100423716C (zh) 2008-10-08
NZ537627A (en) 2006-11-30
IL165835A0 (en) 2006-01-15
US8580308B2 (en) 2013-11-12
EA200600968A1 (ru) 2007-02-27

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B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

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