CS277411B6 - Novel esters of beta-carboline-3-carboxylic acids being substituted in position 5 or 6 - Google Patents

Novel esters of beta-carboline-3-carboxylic acids being substituted in position 5 or 6 Download PDF

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Publication number
CS277411B6
CS277411B6 CS869386A CS938686A CS277411B6 CS 277411 B6 CS277411 B6 CS 277411B6 CS 869386 A CS869386 A CS 869386A CS 938686 A CS938686 A CS 938686A CS 277411 B6 CS277411 B6 CS 277411B6
Authority
CS
Czechoslovakia
Prior art keywords
carboline
substituted
formula
group
carboxylic acid
Prior art date
Application number
CS869386A
Other languages
Czech (cs)
English (en)
Other versions
CS938686A3 (en
Inventor
Helmut Dr Biere
Andreas Dr Huth
Dieter Dr Rahtz
Ralph Dr Schmiechen
Dieter Dr Seidelmann
Wolfgang Dr Kehr
Herbert Hans Dr Schneider
Mogens Dr Engelstoft
Bondo John Dr Hansen
Frank Dr Watjen
Tage Dr Honore
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of CS938686A3 publication Critical patent/CS938686A3/cs
Publication of CS277411B6 publication Critical patent/CS277411B6/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Psychiatry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Heat Sensitive Colour Forming Recording (AREA)
  • Polyesters Or Polycarbonates (AREA)
  • Fats And Perfumes (AREA)
  • Carbon And Carbon Compounds (AREA)
  • Non-Alcoholic Beverages (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CS869386A 1986-03-20 1986-12-16 Novel esters of beta-carboline-3-carboxylic acids being substituted in position 5 or 6 CS277411B6 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19863609699 DE3609699A1 (de) 1986-03-20 1986-03-20 5- oder 6-substituierte-(beta)-carbolin-3-carbonsaeureester

Publications (2)

Publication Number Publication Date
CS938686A3 CS938686A3 (en) 1992-11-18
CS277411B6 true CS277411B6 (en) 1993-03-17

Family

ID=6297016

Family Applications (2)

Application Number Title Priority Date Filing Date
CS869386A CS277411B6 (en) 1986-03-20 1986-12-16 Novel esters of beta-carboline-3-carboxylic acids being substituted in position 5 or 6
CS903634A CS277498B6 (en) 1986-03-20 1986-12-16 Process for preparing esters of beta-carboline-3-carboxylic acids being substituted in position 5 or 6

Family Applications After (1)

Application Number Title Priority Date Filing Date
CS903634A CS277498B6 (en) 1986-03-20 1986-12-16 Process for preparing esters of beta-carboline-3-carboxylic acids being substituted in position 5 or 6

Country Status (24)

Country Link
US (2) US5414002A (fi)
EP (1) EP0239667B1 (fi)
JP (1) JPH0670053B2 (fi)
AT (1) ATE63119T1 (fi)
AU (1) AU596385B2 (fi)
CA (1) CA1332837C (fi)
CS (2) CS277411B6 (fi)
DD (1) DD260068A5 (fi)
DE (2) DE3609699A1 (fi)
DK (1) DK168953B1 (fi)
ES (1) ES2039346T3 (fi)
FI (2) FI864498A0 (fi)
GR (1) GR3002085T3 (fi)
HU (1) HU195218B (fi)
IE (1) IE59344B1 (fi)
IL (1) IL80667A (fi)
MX (1) MX9203701A (fi)
NO (2) NO864362D0 (fi)
NZ (1) NZ218482A (fi)
PH (1) PH25100A (fi)
PT (1) PT83763B (fi)
RU (2) RU1771475C (fi)
UA (2) UA13475A (fi)
ZA (1) ZA872072B (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4122722A1 (de) * 1991-07-06 1993-01-07 Schering Ag Verfahren zur herstellung von indol-derivaten
DE19502753A1 (de) * 1995-01-23 1996-07-25 Schering Ag Neue 9H-Pyrido[3,4-b]indol-Derivate
DE10136842A1 (de) * 2001-07-23 2003-02-13 Schering Ag GABA¶A¶-Rezeptor-Modulatoren mit NMDA-antagonistischer Aktivität
US20030045541A1 (en) * 2001-07-23 2003-03-06 Christopher Bruckner GABA-Receptor modulators with NMDA-Antagonistic activity

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ194747A (en) * 1979-08-29 1988-11-29 Schering Ag 9h-pyrido(3,4-b)indol-3-ylcarboxylic acid derivatives
JPS57123180A (en) * 1980-12-17 1982-07-31 Schering Ag 3-substituted beta-carboline, manufacture and psychotropic drug containing same
DE3240511A1 (de) * 1982-10-29 1984-05-03 Schering AG, 1000 Berlin und 4709 Bergkamen Verfahren zur herstellung von ss-carbolinderivaten
DE3322895A1 (de) * 1983-06-23 1985-01-03 Schering AG, 1000 Berlin und 4709 Bergkamen Neue ss-carboline, verfahren zur ihrer herstellung und ihre verwendung als arzneimittel (s)
DE3335323A1 (de) * 1983-09-27 1985-04-04 Schering AG, 1000 Berlin und 4709 Bergkamen Substituierte ss-carboline, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
DK240184D0 (da) * 1984-05-15 1984-05-15 Ferrosan As Beta-carboline-3-carboxylic acid derivatives and method of preparing the same
DK704488D0 (da) * 1988-12-19 1988-12-19 Novo Industri As Nye n-substituerede azaheterocykliske carboxylsyrer
DE3504045A1 (de) * 1985-02-04 1986-08-07 Schering AG, 1000 Berlin und 4709 Bergkamen Verfahren zur herstellung von ss-carbolinen durch dehydrierung
DE3540653A1 (de) * 1985-11-13 1987-05-14 Schering Ag Neue 3-oxadiazol- und 3-carbonsaeure-ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel
DE3545776A1 (de) * 1985-12-20 1987-06-25 Schering Ag 5-aminoalkyl-ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel

Also Published As

Publication number Publication date
PT83763B (pt) 1989-07-31
DE3679059D1 (de) 1991-06-06
NO163737B (no) 1990-04-02
DE3609699A1 (de) 1987-09-24
FI83321C (fi) 1991-06-25
CS938686A3 (en) 1992-11-18
EP0239667B1 (de) 1991-05-02
IL80667A0 (en) 1987-02-27
DK168953B1 (da) 1994-07-18
NO865121L (no) 1987-09-21
ES2039346T3 (es) 1993-10-01
US5700808A (en) 1997-12-23
JPS62221684A (ja) 1987-09-29
NZ218482A (en) 1990-01-29
NO865121D0 (no) 1986-12-17
UA13475A (uk) 1997-04-25
NO864362D0 (no) 1986-10-31
IL80667A (en) 1991-04-15
RU1771475C (ru) 1992-10-23
ATE63119T1 (de) 1991-05-15
AU596385B2 (en) 1990-05-03
UA26390A (uk) 1999-08-30
PH25100A (en) 1991-02-19
DD260068A5 (de) 1988-09-14
FI83321B (fi) 1991-03-15
CS277498B6 (en) 1993-02-17
US5414002A (en) 1995-05-09
RU2034845C1 (ru) 1995-05-10
CA1332837C (en) 1994-11-01
EP0239667A1 (de) 1987-10-07
NO163737C (no) 1990-07-11
HU195218B (en) 1988-04-28
DK536386D0 (da) 1986-11-10
ZA872072B (en) 1987-09-14
GR3002085T3 (en) 1992-12-30
FI865058A (fi) 1987-09-21
HUT41787A (en) 1987-05-28
IE59344B1 (en) 1994-02-09
IE863094L (en) 1987-09-20
JPH0670053B2 (ja) 1994-09-07
CS363490A3 (en) 1992-11-18
MX9203701A (es) 1992-09-01
PT83763A (de) 1986-12-01
FI865058A0 (fi) 1986-12-11
DK536386A (da) 1987-09-21
AU6516886A (en) 1987-09-24
FI864498A0 (fi) 1986-11-05

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Legal Events

Date Code Title Description
IF00 In force as of 2000-06-30 in czech republic
MK4A Patent expired

Effective date: 20061216