CS276785B6 - PROCESS FOR PREPARING NOVEL DERIVATIVES OF 1H,3H-PYRROLO-(1,2-c)THIAZOLE-7-CARBOXAMIDE - Google Patents

PROCESS FOR PREPARING NOVEL DERIVATIVES OF 1H,3H-PYRROLO-(1,2-c)THIAZOLE-7-CARBOXAMIDE Download PDF

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Publication number
CS276785B6
CS276785B6 CS901252A CS125290A CS276785B6 CS 276785 B6 CS276785 B6 CS 276785B6 CS 901252 A CS901252 A CS 901252A CS 125290 A CS125290 A CS 125290A CS 276785 B6 CS276785 B6 CS 276785B6
Authority
CS
Czechoslovakia
Prior art keywords
pyridyl
group
phenyl
mixture
solution
Prior art date
Application number
CS901252A
Other languages
Czech (cs)
English (en)
Other versions
CS125290A3 (en
Inventor
Claude James
Daniel Lave
Francoise Soler
Original Assignee
Rhone Poulenc Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante
Publication of CS125290A3 publication Critical patent/CS125290A3/cs
Publication of CS276785B6 publication Critical patent/CS276785B6/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
CS901252A 1989-03-17 1990-03-15 PROCESS FOR PREPARING NOVEL DERIVATIVES OF 1H,3H-PYRROLO-(1,2-c)THIAZOLE-7-CARBOXAMIDE CS276785B6 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8903510A FR2644456B1 (fr) 1989-03-17 1989-03-17 Nouveaux derives du 1h, 3h-pyrrolo(1,2-c)thiazolecarboxamide-7, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (2)

Publication Number Publication Date
CS125290A3 CS125290A3 (en) 1992-03-18
CS276785B6 true CS276785B6 (en) 1992-08-12

Family

ID=9379793

Family Applications (2)

Application Number Title Priority Date Filing Date
CS904389A CS438990A3 (en) 1989-03-17 1990-03-15 Process for preparing novel derivatives of 1h,3h-pyrrolo-(1,2-c)thiazole-7-carboxamide
CS901252A CS276785B6 (en) 1989-03-17 1990-03-15 PROCESS FOR PREPARING NOVEL DERIVATIVES OF 1H,3H-PYRROLO-(1,2-c)THIAZOLE-7-CARBOXAMIDE

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CS904389A CS438990A3 (en) 1989-03-17 1990-03-15 Process for preparing novel derivatives of 1h,3h-pyrrolo-(1,2-c)thiazole-7-carboxamide

Country Status (24)

Country Link
US (1) US5086051A (no)
EP (1) EP0388309B1 (no)
JP (1) JPH02289586A (no)
KR (1) KR900014408A (no)
AT (1) ATE102210T1 (no)
BG (1) BG51159A3 (no)
CA (1) CA2012343A1 (no)
CS (2) CS438990A3 (no)
DD (1) DD297822A5 (no)
DE (1) DE69006872T2 (no)
DK (1) DK0388309T3 (no)
ES (1) ES2062432T3 (no)
FI (1) FI92069C (no)
FR (1) FR2644456B1 (no)
IE (1) IE63313B1 (no)
IL (1) IL93760A (no)
MA (1) MA21771A1 (no)
MX (1) MX26542A (no)
NO (1) NO172392C (no)
NZ (1) NZ232960A (no)
PL (1) PL284321A1 (no)
PT (1) PT93485B (no)
TN (1) TNSN90030A1 (no)
ZA (1) ZA902033B (no)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW214545B (no) * 1992-02-17 1993-10-11 Ciba Geigy Ag
US5639782A (en) * 1992-03-04 1997-06-17 Center For Innovative Technology Neolignan derivatives as platelet activating factor receptor antagonists and 5-lipoxygenase inhibitors
US5530141A (en) * 1992-03-04 1996-06-25 Center For Innovative Technology 2,4-diaryl-1,3-dithiolanes; 2,4-diaryl-1,3-dioxolanes; 2,4-diaryl-1,3-oxathiolanes; and 2,5-diaryl-1,3-oxathiolanes for the treatment of disorders mediated by platelet activating factor or products of 5-lipoxygenase
US5648486A (en) * 1992-07-13 1997-07-15 Cytomed, Inc. Compounds and methods for the treatment of inflammatory and immune disorders
US5463083A (en) * 1992-07-13 1995-10-31 Cytomed, Inc. Compounds and methods for the treatment of cardiovascular, inflammatory and immune disorders
DE69329550T2 (de) 1992-07-13 2001-05-31 Cytomed, Inc. 2,5-diaryl tetrahydro-thiopene, -furane und analoge zur behandlung von entzündungs-und immunkrankheiten
US5358938A (en) * 1992-07-13 1994-10-25 Cytomed, Inc. Compounds and methods for the treatment of disorders mediated by platelet activating factor or products of 5-lipoxygenase
US5434151A (en) * 1992-08-24 1995-07-18 Cytomed, Inc. Compounds and methods for the treatment of disorders mediated by platelet activating factor or products of 5-lipoxygenase
TW266206B (no) * 1993-04-28 1995-12-21 Takeda Pharm Industry Co Ltd
US5703093A (en) * 1995-05-31 1997-12-30 Cytomed, Inc. Compounds and methods for the treatment of cardiovascular, inflammatory and immune disorders
US5792776A (en) * 1994-06-27 1998-08-11 Cytomed, Inc., Compounds and methods for the treatment of cardiovascular, inflammatory and immune disorders
US5750565A (en) * 1995-05-25 1998-05-12 Cytomed, Inc. Compounds and methods for the treatment of cardiovascular, inflammatory and immune disorders
US5891895A (en) * 1996-04-15 1999-04-06 Takeda Chemical Industries, Ltd. Hydroxypyridine derivatives their production and use
WO2007020945A1 (ja) * 2005-08-19 2007-02-22 National Institute Of Advanced Industrial Science And Technology 色可逆変化表示装置用電極体及びその製造方法、並びに色可逆変化表示装置及び色可逆変化調光装置
WO2009125434A2 (en) * 2008-04-07 2009-10-15 Cadila Healthcare Limited Oxime derivatives
WO2014192023A1 (en) * 2013-05-22 2014-12-04 Cadila Healthcare Limited Novel compounds suitable for the treatment of dyslipidemia

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2541280B1 (fr) * 1983-01-13 1985-06-21 Rhone Poulenc Sante Nouveaux derives du 1h, 3h-pyrrolo (1,2c) thiazolecarboxamide-7, leur preparation et les medicaments qui les contiennent
FR2601016B1 (fr) * 1986-07-04 1988-10-07 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2601015B1 (fr) * 1986-07-04 1988-08-05 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
NO901237D0 (no) 1990-03-16
ATE102210T1 (de) 1994-03-15
KR900014408A (ko) 1990-10-23
BG51159A3 (en) 1993-02-15
MX26542A (es) 1993-09-01
DE69006872T2 (de) 1994-06-30
FI901325A0 (fi) 1990-03-16
DK0388309T3 (da) 1994-04-11
MA21771A1 (fr) 1990-10-01
NO172392C (no) 1993-07-14
FI92069B (fi) 1994-06-15
CS125290A3 (en) 1992-03-18
FR2644456B1 (fr) 1991-07-05
EP0388309A3 (fr) 1991-07-24
DD297822A5 (de) 1992-01-23
IL93760A (en) 1994-08-26
CS438990A3 (en) 1992-03-18
ZA902033B (en) 1990-12-28
TNSN90030A1 (fr) 1991-03-05
IE63313B1 (en) 1995-04-05
PT93485A (pt) 1990-11-07
FI92069C (fi) 1994-09-26
US5086051A (en) 1992-02-04
EP0388309B1 (fr) 1994-03-02
NZ232960A (en) 1991-02-26
EP0388309A2 (fr) 1990-09-19
ES2062432T3 (es) 1994-12-16
IE900984L (en) 1990-09-17
JPH02289586A (ja) 1990-11-29
NO172392B (no) 1993-04-05
DE69006872D1 (de) 1994-04-07
IL93760A0 (en) 1990-12-23
FR2644456A1 (fr) 1990-09-21
PT93485B (pt) 1996-02-29
CA2012343A1 (fr) 1990-09-17
NO901237L (no) 1990-09-18
PL284321A1 (en) 1991-07-29

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