CS270411B2 - Method of new 4 halogen anthracycline glycosides production - Google Patents

Method of new 4 halogen anthracycline glycosides production Download PDF

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Publication number
CS270411B2
CS270411B2 CS846052A CS605284A CS270411B2 CS 270411 B2 CS270411 B2 CS 270411B2 CS 846052 A CS846052 A CS 846052A CS 605284 A CS605284 A CS 605284A CS 270411 B2 CS270411 B2 CS 270411B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
protecting group
compounds
process according
compound
Prior art date
Application number
CS846052A
Other languages
Czech (cs)
English (en)
Other versions
CS605284A2 (en
Inventor
Antonio Suarato
Sergio Penco
Fernando Giuliani
Federico Arcamone
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of CS605284A2 publication Critical patent/CS605284A2/cs
Publication of CS270411B2 publication Critical patent/CS270411B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
CS846052A 1983-08-11 1984-08-09 Method of new 4 halogen anthracycline glycosides production CS270411B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB838321676A GB8321676D0 (en) 1983-08-11 1983-08-11 4'-haloanthrocycline glycosides

Publications (2)

Publication Number Publication Date
CS605284A2 CS605284A2 (en) 1989-11-14
CS270411B2 true CS270411B2 (en) 1990-06-13

Family

ID=10547171

Family Applications (1)

Application Number Title Priority Date Filing Date
CS846052A CS270411B2 (en) 1983-08-11 1984-08-09 Method of new 4 halogen anthracycline glycosides production

Country Status (19)

Country Link
JP (1) JPS6058997A (da)
AT (1) AT384226B (da)
AU (1) AU563396B2 (da)
BE (1) BE900336A (da)
CA (1) CA1250833A (da)
CH (1) CH660740A5 (da)
CS (1) CS270411B2 (da)
DE (1) DE3428945A1 (da)
DK (1) DK381884A (da)
FI (1) FI78109C (da)
FR (1) FR2554450B1 (da)
GB (2) GB8321676D0 (da)
GR (1) GR80046B (da)
HU (1) HU194266B (da)
IT (1) IT1209576B (da)
NL (1) NL8402477A (da)
SE (1) SE8404005L (da)
SU (1) SU1579465A3 (da)
ZA (1) ZA846147B (da)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2159518A (en) * 1984-06-08 1985-12-04 Erba Farmitalia New anthracyclines and process for manufacture
GB8414619D0 (en) * 1984-06-08 1984-07-11 Erba Farmitalia Anthracyclines
DE3500017A1 (de) * 1985-01-02 1986-07-10 Farmitalia Carlo Erba S.p.A., Mailand/Milano 4'-haloanthracyclinester
GB2218087B (en) * 1988-04-22 1991-01-30 Erba Carlo Spa 4-demethoxy-4'-deoxy-4'iodo anthracycline glycosides
AU601857B2 (en) * 1988-06-30 1990-09-20 Pharmacia & Upjohn S.P.A. A new antitumor agent obtained by microbial stereoselective reduction of 4'-deoxy-4'-iododoxorubicin
MA21995A1 (fr) * 1989-11-13 1991-07-01 Menarini Farma Ind Nouvelles fluoronaphthacenediones,leurs derives glycozyles et leurs procedes de fabrication .
GB9418260D0 (en) * 1994-09-09 1994-10-26 Erba Carlo Spa Anthracycline derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR892943A (fr) * 1942-03-06 1944-05-24 Ig Farbenindustrie Ag Procédé pour épurer la dilactone gamma céto-pimélique
US4345070A (en) * 1980-09-29 1982-08-17 Farmitalia Carlo Erba S.P.A. Process for the preparation of 4'-deoxy-daunorubicin and 4'-deoxy-doxorubicin
US4438105A (en) * 1982-04-19 1984-03-20 Farmaitalia Carlo Erba S.P.A 4'-Iododerivatives of anthracycline glycosides

Also Published As

Publication number Publication date
GB8420237D0 (en) 1984-09-12
NL8402477A (nl) 1985-03-01
DK381884D0 (da) 1984-08-08
FI78109B (fi) 1989-02-28
GB2144744B (en) 1986-12-03
CS605284A2 (en) 1989-11-14
FR2554450A1 (fr) 1985-05-10
SU1579465A3 (ru) 1990-07-15
ZA846147B (en) 1985-03-27
CA1250833A (en) 1989-03-07
DE3428945A1 (de) 1985-02-28
DK381884A (da) 1985-02-12
SE8404005D0 (sv) 1984-08-07
GR80046B (en) 1984-12-10
HU194266B (en) 1988-01-28
JPS6058997A (ja) 1985-04-05
AT384226B (de) 1987-10-12
FI78109C (fi) 1989-06-12
SE8404005L (sv) 1985-02-12
IT8422232A0 (it) 1984-08-06
ATA253884A (de) 1987-03-15
FR2554450B1 (fr) 1987-01-30
AU563396B2 (en) 1987-07-09
BE900336A (fr) 1985-02-11
AU3168584A (en) 1985-02-14
FI843110A0 (fi) 1984-08-08
GB2144744A (en) 1985-03-13
HUT35691A (en) 1985-07-29
GB8321676D0 (en) 1983-09-14
FI843110A (fi) 1985-02-12
IT1209576B (it) 1989-08-30
CH660740A5 (de) 1987-06-15

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