CS238611B2 - Preparation method of sulphone-amides - Google Patents

Preparation method of sulphone-amides Download PDF

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Publication number
CS238611B2
CS238611B2 CS809599A CS959980A CS238611B2 CS 238611 B2 CS238611 B2 CS 238611B2 CS 809599 A CS809599 A CS 809599A CS 959980 A CS959980 A CS 959980A CS 238611 B2 CS238611 B2 CS 238611B2
Authority
CS
Czechoslovakia
Prior art keywords
ethyl
acid
yield
carbon atoms
theory
Prior art date
Application number
CS809599A
Other languages
Czech (cs)
English (en)
Inventor
Ernst Ch Witte
Hans P Wolff
Karlheinz Stegmeier
Egon Roesch
Original Assignee
Boehringer Mannheim Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Mannheim Gmbh filed Critical Boehringer Mannheim Gmbh
Publication of CS238611B2 publication Critical patent/CS238611B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Devices That Are Associated With Refrigeration Equipment (AREA)
CS809599A 1980-01-07 1980-12-31 Preparation method of sulphone-amides CS238611B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19803000377 DE3000377A1 (de) 1980-01-07 1980-01-07 Neue sulfonamide, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
CS238611B2 true CS238611B2 (en) 1985-12-16

Family

ID=6091629

Family Applications (1)

Application Number Title Priority Date Filing Date
CS809599A CS238611B2 (en) 1980-01-07 1980-12-31 Preparation method of sulphone-amides

Country Status (22)

Country Link
US (1) US4443477A (nl)
EP (1) EP0031954B1 (nl)
JP (1) JPS56100757A (nl)
AT (1) ATE6641T1 (nl)
AU (1) AU538993B2 (nl)
CA (1) CA1241341A (nl)
CS (1) CS238611B2 (nl)
DD (1) DD157190A5 (nl)
DE (2) DE3000377A1 (nl)
ES (1) ES498308A0 (nl)
FI (1) FI73667C (nl)
GR (1) GR72486B (nl)
HK (1) HK68887A (nl)
IE (1) IE50657B1 (nl)
IL (1) IL61834A (nl)
PH (1) PH18739A (nl)
PL (1) PL127050B1 (nl)
PT (1) PT72305B (nl)
SG (1) SG2387G (nl)
SU (1) SU1088664A3 (nl)
YU (1) YU42995B (nl)
ZA (1) ZA8132B (nl)

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US4959383A (en) * 1988-10-31 1990-09-25 E. R. Squibb & Sons, Inc. Phenylsulfone alkenoic acids, derivatives thereof, compositions containing same and method of use
US4975452A (en) * 1989-06-02 1990-12-04 E. R. Squibb & Sons, Inc. Geminally substituted thiaheterocyclic carboxylic acids and derivatives thereof
US5106991A (en) * 1989-06-02 1992-04-21 E. R. Squibb & Sons, Inc. Geminally substituted thiaheterocyclic carboxylic acids and derivatives thereof
US5153214A (en) * 1989-06-28 1992-10-06 Ciba-Geigy Corporation Certain (arylsulfonamido- and imidazolyl-)-substituted carboxylic acids and derivatives thereof and use for suppressing thromboxane activity
US5025025A (en) * 1989-06-28 1991-06-18 Ciba-Geigy Corporation (Arylsulfonamido- and pyridyl-)-substituted carboxylic acids and derivatives thereof and use for suppressing thromboxane activity
DE4010536A1 (de) * 1990-04-02 1991-10-10 Boehringer Mannheim Gmbh Pharmazeutische waessrige loesung von 4-(2-(benzolsulfonylamino)-ethyl)-phenoxyessigsaeure
FR2665440B1 (fr) * 1990-07-31 1994-02-04 Lipha Nouveaux cycloalkylsulfonamides substitues, procedes de preparation et medicaments les contenant.
US5189211A (en) * 1990-08-01 1993-02-23 Taisho Pharmaceutical Co., Ltd. Sulfonamide derivatives
US5409959A (en) * 1991-01-29 1995-04-25 Genelabs Incorporated Antithrombotic treatment with calix(n)arene compounds
DE4109735A1 (de) * 1991-03-25 1992-10-01 Boehringer Mannheim Gmbh Neue sulfonamide, verfahren zu ihrer herstellung und arzneimittel, die diese verbindungen enthalten
US5280034A (en) * 1991-08-23 1994-01-18 E. R. Squibb & Sons, Inc. Bis-heterocyclic prostaglandin analogs
US5827868A (en) * 1991-10-07 1998-10-27 E. R. Squibb & Sons, Inc. Prostaglandin analogs
TW219358B (nl) * 1991-12-20 1994-01-21 Hokuriku Pharmaceutical
GB9220137D0 (en) * 1992-09-23 1992-11-04 Pfizer Ltd Therapeutic agents
JPH0753505A (ja) * 1992-10-01 1995-02-28 Hokuriku Seiyaku Co Ltd ベンゼンスルホンアミド誘導体及びその用途
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FR2760235B1 (fr) * 1997-02-28 1999-04-09 Adir Nouveaux derives de benzenesulfonylamine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
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SA109300309B1 (ar) 2008-05-20 2013-01-22 باير شيرنج فارما ايه جي مشتقات فينيل وبنزو داي أوكسينيل إندازول بها استبدال
EP2303013A1 (en) * 2008-07-07 2011-04-06 Fasgen, Inc. Novel compounds, pharmaceutical compositions containing same, methods of use for same, and methods for preparing same
CN110776447A (zh) 2012-09-20 2020-02-11 坦普尔大学 取代的烷基二芳基衍生物、制备方法和用途
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Also Published As

Publication number Publication date
EP0031954A3 (en) 1981-11-11
CA1241341A (en) 1988-08-30
PT72305B (de) 1981-12-17
FI73667C (fi) 1987-11-09
YU881A (en) 1983-10-31
YU42995B (en) 1989-02-28
GR72486B (nl) 1983-11-14
SU1088664A3 (ru) 1984-04-23
JPS6352625B2 (nl) 1988-10-19
DE3000377A1 (de) 1981-07-09
PT72305A (de) 1981-02-01
PL127050B1 (en) 1983-09-30
SG2387G (en) 1987-11-13
ZA8132B (en) 1982-02-24
EP0031954B1 (de) 1984-03-14
AU6597481A (en) 1981-07-16
EP0031954A2 (de) 1981-07-15
ATE6641T1 (de) 1984-03-15
PL229072A1 (nl) 1982-04-26
HK68887A (en) 1987-10-02
AU538993B2 (en) 1984-09-06
FI804085L (fi) 1981-07-08
IL61834A (en) 1984-06-29
PH18739A (en) 1985-09-16
IL61834A0 (en) 1981-01-30
DE3067068D1 (en) 1984-04-19
ES8200655A1 (es) 1981-12-01
JPS56100757A (en) 1981-08-12
ES498308A0 (es) 1981-12-01
IE810006L (en) 1981-07-07
IE50657B1 (en) 1986-06-11
US4443477A (en) 1984-04-17
DD157190A5 (de) 1982-10-20
FI73667B (fi) 1987-07-31

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