CS234003B2 - Method of aryl-phenylindenes and aryl-phenylnaphalenes preparation - Google Patents

Method of aryl-phenylindenes and aryl-phenylnaphalenes preparation Download PDF

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Publication number
CS234003B2
CS234003B2 CS766972A CS697276A CS234003B2 CS 234003 B2 CS234003 B2 CS 234003B2 CS 766972 A CS766972 A CS 766972A CS 697276 A CS697276 A CS 697276A CS 234003 B2 CS234003 B2 CS 234003B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
hydrogen
compound
alkoxy
carbon atoms
Prior art date
Application number
CS766972A
Other languages
Czech (cs)
English (en)
Inventor
Tulio Suarez
Charles D Jones
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of CS234003B2 publication Critical patent/CS234003B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/088—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46—Friedel-Crafts reactions
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/65—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by splitting-off hydrogen atoms or functional groups; by hydrogenolysis of functional groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/673—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CS766972A 1975-10-28 1976-10-28 Method of aryl-phenylindenes and aryl-phenylnaphalenes preparation CS234003B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/625,992 US4017546A (en) 1975-10-28 1975-10-28 Novel antifertility agents

Publications (1)

Publication Number Publication Date
CS234003B2 true CS234003B2 (en) 1985-03-14

Family

ID=24508497

Family Applications (1)

Application Number Title Priority Date Filing Date
CS766972A CS234003B2 (en) 1975-10-28 1976-10-28 Method of aryl-phenylindenes and aryl-phenylnaphalenes preparation

Country Status (31)

Country Link
US (2) US4017546A (ja)
JP (1) JPS5253844A (ja)
AR (1) AR221031A1 (ja)
AT (1) AT347443B (ja)
AU (1) AU503883B2 (ja)
BE (1) BE847717A (ja)
BG (1) BG27556A3 (ja)
CA (1) CA1064926A (ja)
CH (1) CH624375A5 (ja)
CS (1) CS234003B2 (ja)
DD (1) DD127462A5 (ja)
DE (1) DE2647906C2 (ja)
DK (1) DK484676A (ja)
ES (1) ES452736A1 (ja)
FR (1) FR2329265A1 (ja)
GB (1) GB1562806A (ja)
GR (1) GR61239B (ja)
HU (1) HU176092B (ja)
IE (1) IE43642B1 (ja)
IL (1) IL50414A (ja)
MX (1) MX4320E (ja)
NL (1) NL7611973A (ja)
NZ (1) NZ182426A (ja)
PH (2) PH13486A (ja)
PL (1) PL106987B1 (ja)
PT (1) PT65754B (ja)
RO (1) RO70754A (ja)
SE (1) SE431086B (ja)
SU (1) SU654164A3 (ja)
YU (1) YU262176A (ja)
ZA (1) ZA766441B (ja)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4017546A (en) * 1975-10-28 1977-04-12 Eli Lilly And Company Novel antifertility agents
US4400543A (en) * 1975-10-28 1983-08-23 Eli Lilly And Company 3-Phenyl-4-benzoyl-1,2-dihydronaphthalenes
US4230862A (en) * 1975-10-28 1980-10-28 Eli Lilly And Company Antifertility compounds
US4323707A (en) * 1975-10-28 1982-04-06 Eli Lilly And Company Antifertility compounds
US5552401A (en) * 1995-02-28 1996-09-03 Eli Lilly And Company 2-benzyl-3-arylbenzothiophenes
US6107346A (en) * 1997-08-11 2000-08-22 Eli Lilly And Company Methods for treating hyperlipidemia

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2551316A (en) * 1948-02-20 1951-05-01 Searle & Co 9-aminoalkyl 9-alkanoyl 9, 10 dihydroanthracenes
US3396169A (en) * 1966-10-26 1968-08-06 Upjohn Co Substituted 2-phenyl-1-(tertiary-aminoalkoxy) phenyl-3, 4-dihydronaphthalenes
US3274213A (en) * 1961-09-05 1966-09-20 Upjohn Co Alkoxy-substituted 2-phenyl-1-(tertiary-aminoalkoxy)phenyl-3, 4-dihydronaphthalenes
US3862232A (en) * 1963-07-03 1975-01-21 Upjohn Co 1-(p-hydroxyphenyl)-2-phenyl-6-(2-diethylaminoethoxy)-3,4-dihydronaphthalene and the salts thereof
US3293263A (en) * 1963-12-09 1966-12-20 Upjohn Co Diphenylbenzocycloalkenes
US3519675A (en) * 1964-06-01 1970-07-07 Upjohn Co 1,2-diphenyl-3,4-dihydronaphthalenes and 2,3-diphenylindenes
US3320271A (en) * 1964-06-01 1967-05-16 Upjohn Co 1, 2-diphenyl-3, 4-dihydronaphthalenes and 2, 3-diphenylindenes
US3483293A (en) * 1967-12-15 1969-12-09 Upjohn Co Method for controlling birds and rodents
US4017546A (en) * 1975-10-28 1977-04-12 Eli Lilly And Company Novel antifertility agents

Also Published As

Publication number Publication date
DD127462A5 (ja) 1977-09-28
ES452736A1 (es) 1978-01-16
AU503883B2 (en) 1979-09-27
PL106987B1 (pl) 1980-01-31
AT347443B (de) 1978-12-27
IL50414A (en) 1980-09-16
ATA800676A (de) 1978-05-15
SE431086B (sv) 1984-01-16
JPS6114141B2 (ja) 1986-04-17
CA1064926A (en) 1979-10-23
FR2329265B1 (ja) 1980-05-16
BE847717A (fr) 1977-04-28
JPS5253844A (en) 1977-04-30
DK484676A (da) 1977-04-29
HU176092B (en) 1980-12-28
US4075223A (en) 1978-02-21
NZ182426A (en) 1978-11-13
GR61239B (en) 1978-10-12
MX4320E (es) 1982-03-24
RO70754A (ro) 1982-10-26
DE2647906C2 (de) 1985-01-31
PT65754A (en) 1976-11-01
FR2329265A1 (fr) 1977-05-27
PH14545A (en) 1981-09-24
US4017546A (en) 1977-04-12
CH624375A5 (ja) 1981-07-31
NL7611973A (nl) 1977-05-02
SU654164A3 (ru) 1979-03-25
ZA766441B (en) 1978-06-28
YU262176A (en) 1982-05-31
GB1562806A (en) 1980-03-19
DE2647906A1 (de) 1977-05-05
IL50414A0 (en) 1976-11-30
BG27556A3 (en) 1979-11-12
SE7611952L (sv) 1977-04-29
IE43642L (en) 1977-04-28
AR221031A1 (es) 1980-12-30
PH13486A (en) 1980-05-21
IE43642B1 (en) 1981-04-22
PT65754B (en) 1978-04-27
AU1740776A (en) 1978-03-09

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