CS227007B2 - Method of preparing carbazol-4-yl oxypropanolamine derivatives - Google Patents

Method of preparing carbazol-4-yl oxypropanolamine derivatives Download PDF

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Publication number
CS227007B2
CS227007B2 CS792434A CS243479A CS227007B2 CS 227007 B2 CS227007 B2 CS 227007B2 CS 792434 A CS792434 A CS 792434A CS 243479 A CS243479 A CS 243479A CS 227007 B2 CS227007 B2 CS 227007B2
Authority
CS
Czechoslovakia
Prior art keywords
carbazol
yloxy
formula
ethylamino
theory
Prior art date
Application number
CS792434A
Other languages
Czech (cs)
English (en)
Inventor
Fritz Dr Wiedemann
Wolfgang Dr Kampe
Max Dr Thiel
Gisbert Dr Sponer
Egon Dr Roesch
Karl Prof Dr Dietmann
Original Assignee
Boehringer Mannheim Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6036838&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CS227007(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Mannheim Gmbh filed Critical Boehringer Mannheim Gmbh
Priority to CS792434A priority Critical patent/CS227047B2/cs
Publication of CS227007B2 publication Critical patent/CS227007B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/64—Oxygen atoms

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CS792434A 1978-04-13 1979-04-10 Method of preparing carbazol-4-yl oxypropanolamine derivatives CS227007B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS792434A CS227047B2 (cs) 1978-04-13 1982-08-20 Způsob výroby derivátů karbazol-4-yloxypropanolaminu

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19782815926 DE2815926A1 (de) 1978-04-13 1978-04-13 Neue carbazolyl-(4)-oxy-propanolamin-derivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
CS227007B2 true CS227007B2 (en) 1984-04-16

Family

ID=6036838

Family Applications (2)

Application Number Title Priority Date Filing Date
CS792434A CS227007B2 (en) 1978-04-13 1979-04-10 Method of preparing carbazol-4-yl oxypropanolamine derivatives
CS914200A CS420091A3 (en) 1978-04-13 1991-12-31 Derivatives of carbazol-4-yloxy-propanol amine, process of their preparation and medicament containing these compounds

Family Applications After (1)

Application Number Title Priority Date Filing Date
CS914200A CS420091A3 (en) 1978-04-13 1991-12-31 Derivatives of carbazol-4-yloxy-propanol amine, process of their preparation and medicament containing these compounds

Country Status (23)

Country Link
US (1) US4503067A (xx)
EP (1) EP0004920B1 (xx)
JP (2) JPS54157558A (xx)
AT (1) AT375639B (xx)
AU (1) AU522975B2 (xx)
BG (1) BG61419B2 (xx)
CA (1) CA1129416A (xx)
CS (2) CS227007B2 (xx)
DD (1) DD143607A5 (xx)
DE (2) DE2815926A1 (xx)
DK (1) DK154555C (xx)
ES (1) ES479396A1 (xx)
FI (1) FI70406C (xx)
HK (1) HK2385A (xx)
HU (1) HU179433B (xx)
IL (1) IL57020A (xx)
LT (1) LT2628B (xx)
LU (1) LU88320I2 (xx)
MX (1) MX9203380A (xx)
NL (1) NL930110I2 (xx)
SG (1) SG52284G (xx)
SU (1) SU810079A3 (xx)
ZA (1) ZA791732B (xx)

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US4076829A (en) * 1974-11-16 1978-02-28 Boehringer Mannheim Gmbh Aminopropanol compounds and compositions for the treatment of cardiac and circulatory diseases
US4115409A (en) * 1975-12-05 1978-09-19 Imperial Chemical Industries Limited Alkanolamine derivatives
GB1508208A (en) * 1975-12-05 1978-04-19 Ici Ltd Amide derivatives

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DE2815926A1 (de) 1979-10-18
AU4582079A (en) 1979-10-18
ZA791732B (en) 1980-05-28
EP0004920A1 (de) 1979-10-31
JPS63258416A (ja) 1988-10-25
FI70406C (fi) 1986-09-19
SU810079A3 (ru) 1981-02-28
ES479396A1 (es) 1980-04-16
AT375639B (de) 1984-08-27
DE2960553D1 (en) 1981-11-05
LT2628B (lt) 1994-04-25
FI70406B (fi) 1986-03-27
SG52284G (en) 1985-03-29
CA1129416A (en) 1982-08-10
MX9203380A (es) 1992-09-01
US4503067A (en) 1985-03-05
EP0004920B1 (de) 1981-08-05
AU522975B2 (en) 1982-07-08
IL57020A (en) 1982-07-30
DD143607A5 (de) 1980-09-03
HU179433B (en) 1982-10-28
NL930110I2 (nl) 1994-12-01
BG61419B2 (bg) 1997-07-31
JPH0123462B2 (xx) 1989-05-02
JPS54157558A (en) 1979-12-12
DK154555B (da) 1988-11-28
HK2385A (en) 1985-01-18
IL57020A0 (en) 1979-07-25
DK141979A (da) 1979-10-14
DK154555C (da) 1989-06-19
CS420091A3 (en) 1992-04-15
LU88320I2 (de) 1994-05-04
FI791142A (fi) 1979-10-14
ATA276279A (de) 1984-01-15
NL930110I1 (nl) 1993-10-18

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