CS197276B2 - Method of producing new 1,5,10,10a-tetrahydrothiazolo/3,4-b/isoquinolines - Google Patents
Method of producing new 1,5,10,10a-tetrahydrothiazolo/3,4-b/isoquinolines Download PDFInfo
- Publication number
- CS197276B2 CS197276B2 CS765082A CS508276A CS197276B2 CS 197276 B2 CS197276 B2 CS 197276B2 CS 765082 A CS765082 A CS 765082A CS 508276 A CS508276 A CS 508276A CS 197276 B2 CS197276 B2 CS 197276B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- formula
- hydrogen
- pyridyl
- tetrahydroisoquinoline
- tetrahydrothiazolo
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/12—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
- C07D217/14—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
- C07D217/16—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Pain & Pain Management (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CS776704A CS197277B2 (cs) | 1975-08-06 | 1977-10-14 | Zpustli) výroby nových l,5,19,10a-tetrahydroihiazolo- [ 3,4-b jisochinolinových derivátů |
CS778474A CS197278B2 (cs) | 1975-08-06 | 1977-10-14 | Způsob výroby derivátů l,5,13,10a-t3traIiydroUiiazoIn- [ 3,4-b 1 isochinolinu |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7524523A FR2320098A1 (fr) | 1975-08-06 | 1975-08-06 | Nouveaux derives de la thiazilo (3,4-b) isoquinoleine, leur preparation et les compositions qui les contiennent |
FR7614935A FR2351655A1 (fr) | 1976-05-18 | 1976-05-18 | Nouveau derive de la thiazolo (3,4-b) isoquinoleine, sa preparation et les compositions qui le contiennent |
Publications (1)
Publication Number | Publication Date |
---|---|
CS197276B2 true CS197276B2 (en) | 1980-04-30 |
Family
ID=26219017
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CS765082A CS197276B2 (en) | 1975-08-06 | 1976-08-03 | Method of producing new 1,5,10,10a-tetrahydrothiazolo/3,4-b/isoquinolines |
Country Status (26)
Country | Link |
---|---|
US (1) | US4064247A (es) |
JP (1) | JPS5219699A (es) |
AR (2) | AR211868A1 (es) |
AT (2) | AT350054B (es) |
AU (1) | AU505316B2 (es) |
CA (1) | CA1073909A (es) |
CH (1) | CH612682A5 (es) |
CS (1) | CS197276B2 (es) |
DE (1) | DE2635516C3 (es) |
DK (1) | DK141069B (es) |
ES (2) | ES450530A1 (es) |
FI (1) | FI60214C (es) |
GB (1) | GB1503091A (es) |
HU (1) | HU173003B (es) |
IE (1) | IE44379B1 (es) |
IL (1) | IL50208A (es) |
LU (1) | LU75540A1 (es) |
MX (1) | MX3639E (es) |
NL (1) | NL169076C (es) |
NO (1) | NO762729L (es) |
NZ (1) | NZ181693A (es) |
OA (1) | OA05403A (es) |
PL (2) | PL108413B1 (es) |
PT (1) | PT65442B (es) |
SE (1) | SE422065B (es) |
SU (2) | SU629881A3 (es) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NL7800383A (nl) * | 1977-01-20 | 1978-07-24 | Rhone Poulenc Ind | Nieuwe isochinolinederivaten, de bereiding ervan en preparaten die de isochinolinederivaten bevatten. |
FR2412545A1 (fr) * | 1977-12-23 | 1979-07-20 | Rhone Poulenc Ind | Nouveaux derives de l'isoquinoleine, leur preparation et les compositions pharmaceutiques qui les contiennent |
NL7800385A (nl) * | 1977-02-04 | 1978-08-08 | Rhone Poulenc Ind | Nieuwe indoolderivaten, werkwijzen ter berei- ding ervan en preparaten die de nieuwe deriva- ten bevatten. |
FR2412554A2 (fr) * | 1977-12-23 | 1979-07-20 | Rhone Poulenc Ind | Nouveaux derives de l'indole, leur preparation et les compositions qui les contiennent |
FR2433023A2 (fr) * | 1978-08-09 | 1980-03-07 | Rhone Poulenc Ind | Nouveaux derives de l'isoquinoleine, leur preparation et les compositions qui les contiennent |
FR2408615A1 (fr) * | 1977-11-10 | 1979-06-08 | Rhone Poulenc Ind | Nouveaux derives de l'isoquinoleine, leur preparation et les compositions qui les contiennent |
SU797580A3 (ru) * | 1977-11-10 | 1981-01-15 | Рон-Пуленк Эндюстри (Фирма) | Способ получени производных изохино-лиНА, иХ СОлЕй, РАцЕМАТОВ или ОпТичЕС-КиХ изОМЕРОВ |
FR2456110A2 (fr) * | 1979-05-09 | 1980-12-05 | Rhone Poulenc Ind | Nouveaux derives de l'isoquinoleine, leur preparation et les compositions qui les contiennent |
FR2468613A2 (fr) * | 1979-10-29 | 1981-05-08 | Rhone Poulenc Ind | Nouveaux derives de la thienopyridine, leur preparation et les medicaments qui les contiennent |
NL7908655A (nl) * | 1978-12-07 | 1980-06-10 | Rhone Poulenc Ind | Nieuwe thienopyridine-derivaten, de bereiding ervan, alsmede farmaceutische preparaten, die de nieuwe derivaten bevatten. |
NL8002540A (nl) * | 1979-05-09 | 1980-11-11 | Rhone Poulenc Ind | Nieuwe isochinoline derivaten, werkwijzen ter bereiding ervan en farmaceutische preparaten, die de nieuwe derivaten bevatten. |
HU181232B (en) * | 1979-12-04 | 1983-06-28 | Rhone Poulenc Ind | Process for preparing new derivatives of thiazolo-isoquinoline |
US4269842A (en) * | 1979-12-05 | 1981-05-26 | Rhone-Poulenc Industries | Method for treating rhinoviral complaints |
FR2624861B1 (fr) * | 1987-12-21 | 1990-06-01 | Delalande Sa | Carbamates tricycliques, leur procede de preparation et leur application en therapeutique |
US5059692A (en) * | 1989-09-01 | 1991-10-22 | Hiroyoshi Hidaka | Novel compounds exhibiting a vasodilating activity and inhibitory activity for platelet aggregation |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3455933A (en) * | 1966-11-15 | 1969-07-15 | American Home Prod | Thiazolo and thiazino isoquinoline derivatives |
HU170680B (es) * | 1973-05-30 | 1977-08-28 |
-
1976
- 1976-07-29 OA OA55901A patent/OA05403A/xx unknown
- 1976-07-29 NL NLAANVRAGE7608444,A patent/NL169076C/xx not_active IP Right Cessation
- 1976-08-02 GB GB32128/76A patent/GB1503091A/en not_active Expired
- 1976-08-03 CS CS765082A patent/CS197276B2/cs unknown
- 1976-08-04 IL IL50208A patent/IL50208A/xx unknown
- 1976-08-04 CA CA258,441A patent/CA1073909A/fr not_active Expired
- 1976-08-05 PT PT65442A patent/PT65442B/pt unknown
- 1976-08-05 SE SE7608808A patent/SE422065B/xx unknown
- 1976-08-05 AR AR264233A patent/AR211868A1/es active
- 1976-08-05 MX MX762133U patent/MX3639E/es unknown
- 1976-08-05 LU LU75540A patent/LU75540A1/xx unknown
- 1976-08-05 NZ NZ181693A patent/NZ181693A/xx unknown
- 1976-08-05 AU AU16615/76A patent/AU505316B2/en not_active Expired
- 1976-08-05 CH CH1004176A patent/CH612682A5/xx not_active IP Right Cessation
- 1976-08-05 HU HU76RO00000892A patent/HU173003B/hu unknown
- 1976-08-05 NO NO762729A patent/NO762729L/no unknown
- 1976-08-05 DK DK353876AA patent/DK141069B/da not_active IP Right Cessation
- 1976-08-05 IE IE1728/76A patent/IE44379B1/en unknown
- 1976-08-05 US US05/711,963 patent/US4064247A/en not_active Expired - Lifetime
- 1976-08-05 JP JP51093548A patent/JPS5219699A/ja active Granted
- 1976-08-06 DE DE2635516A patent/DE2635516C3/de not_active Expired
- 1976-08-06 ES ES450530A patent/ES450530A1/es not_active Expired
- 1976-08-06 PL PL1976211043A patent/PL108413B1/pl unknown
- 1976-08-06 AT AT586476A patent/AT350054B/de not_active IP Right Cessation
- 1976-08-06 FI FI762256A patent/FI60214C/fi not_active IP Right Cessation
- 1976-08-06 SU SU762386213A patent/SU629881A3/ru active
- 1976-08-06 PL PL1976191674A patent/PL108034B1/pl unknown
- 1976-11-04 ES ES452987A patent/ES452987A1/es not_active Expired
-
1977
- 1977-03-28 AR AR267010A patent/AR211170A1/es active
- 1977-07-26 SU SU772504520A patent/SU635874A3/ru active
-
1978
- 1978-06-01 AT AT397778A patent/AT351544B/de not_active IP Right Cessation
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