CS194788B2 - Method of producing depot steroid esters - Google Patents

Method of producing depot steroid esters

Info

Publication number
CS194788B2
CS194788B2 CS768342A CS834276A CS194788B2 CS 194788 B2 CS194788 B2 CS 194788B2 CS 768342 A CS768342 A CS 768342A CS 834276 A CS834276 A CS 834276A CS 194788 B2 CS194788 B2 CS 194788B2
Authority
CS
Czechoslovakia
Prior art keywords
steroid esters
producing
depot steroid
producing depot
esters
Prior art date
Application number
CS768342A
Other languages
Czech (cs)
English (en)
Inventor
Paul-Eberhard Schulze
Ulrich Speck
Dieter Bittler
Rudolf Wiechert
Bernard Acksteiner
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of CS194788B2 publication Critical patent/CS194788B2/cs

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0033Androstane derivatives substituted in position 17 alfa and 17 beta
    • C07J1/004Androstane derivatives substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0048Alkynyl derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0081Substituted in position 17 alfa and 17 beta
    • C07J1/0088Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096Alkynyl derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J11/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J21/00Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005Ketals
    • C07J21/006Ketals at position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J31/00Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C07J5/0046Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
    • C07J5/0053Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa not substituted in position 16
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J53/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002Carbocyclic rings fused
    • C07J53/0043 membered carbocyclic rings
    • C07J53/0053 membered carbocyclic rings in position 12
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J53/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002Carbocyclic rings fused
    • C07J53/0043 membered carbocyclic rings
    • C07J53/0083 membered carbocyclic rings in position 15/16

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CS768342A 1975-12-19 1976-12-17 Method of producing depot steroid esters CS194788B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2558076A DE2558076C2 (de) 1975-12-19 1975-12-19 Depot-Steroidester, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Präparate

Publications (1)

Publication Number Publication Date
CS194788B2 true CS194788B2 (en) 1979-12-31

Family

ID=5965325

Family Applications (1)

Application Number Title Priority Date Filing Date
CS768342A CS194788B2 (en) 1975-12-19 1976-12-17 Method of producing depot steroid esters

Country Status (35)

Country Link
US (1) US4119626A (it)
JP (1) JPS5278860A (it)
AT (1) AT357704B (it)
AU (1) AU507111B2 (it)
BE (1) BE849553A (it)
BG (2) BG30475A3 (it)
CA (1) CA1086305A (it)
CH (1) CH630097A5 (it)
CS (1) CS194788B2 (it)
DD (1) DD132270A5 (it)
DE (1) DE2558076C2 (it)
DK (1) DK146629C (it)
EG (1) EG12383A (it)
ES (1) ES454297A1 (it)
FI (1) FI57263C (it)
FR (1) FR2335231A1 (it)
GB (1) GB1554199A (it)
GR (1) GR62084B (it)
HU (1) HU179343B (it)
IE (1) IE44320B1 (it)
IL (1) IL50981A (it)
IT (1) IT1065783B (it)
LU (1) LU76398A1 (it)
MX (1) MX3798E (it)
NL (1) NL7614023A (it)
NO (2) NO145620C (it)
NZ (1) NZ182890A (it)
PH (1) PH13907A (it)
PL (1) PL105525B1 (it)
PT (1) PT65973B (it)
RO (1) RO75383A (it)
SE (1) SE428930B (it)
SU (1) SU648105A3 (it)
YU (1) YU293176A (it)
ZA (1) ZA767510B (it)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7613248A (nl) * 1976-11-26 1978-05-30 Akzo Nv Werkwijze voor het bereiden van nieuwe steroid- esters.
DE2848423A1 (de) * 1978-11-08 1980-05-29 Merck Patent Gmbh Hydrocortisonester, diese enthaltende pharmazeutische zubereitungen und verfahren zu ihrer herstellung
US4507290A (en) * 1981-04-07 1985-03-26 World Health Organization Esters of 17 α-ethynyl 19-nor-testosterone and 17 α-ethynyl-18-homo-19-nor-testosterone and pharmaceutical compositions containing the same
DE3133082A1 (de) * 1981-08-18 1983-03-10 Schering Ag, 1000 Berlin Und 4619 Bergkamen Neue hydrocortison-derivate, ihre herstellung und verwendung
JPS59184200A (ja) * 1983-03-31 1984-10-19 Takeda Chem Ind Ltd ステロイド化合物、その製造法及び薬剤
DE3511588A1 (de) * 1985-03-27 1986-10-02 Schering AG, Berlin und Bergkamen, 1000 Berlin Waessrige kristallsuspension von steroidglykoestern
JPH02139518U (it) * 1989-04-25 1990-11-21
DE4232521A1 (de) * 1992-09-22 1994-03-24 Schering Ag Gestagen wirksame 4,5;11,12-Estradiene, Verfahren zu ihrer Herstellung, diese Estradiene enthaltende Arzneimittel sowie deren Verwendung zur Herstellung von Arzneimitteln

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB660199A (en) * 1947-09-13 1951-10-31 Sterling Drug Inc Acyloxyalkanoates of hydroxylated hormones
GB817735A (en) * 1955-08-26 1959-08-06 Lab Francais Chimiotherapie Improvements in or relating to steroidal compounds
US3082222A (en) * 1958-03-26 1963-03-19 Ott Erwin Steroid acid-esters and salts thereof, and method of making the same
FR1326329A (fr) * 1959-10-28 1963-05-10 Préparation de sels d'hormones solubles dans l'eau et dans les lipides
US3629245A (en) * 1965-05-14 1971-12-21 Roussel Uclaf 16 17-isoxazolino-delta-1 3 5(10)-gonatrienes
US3856956A (en) * 1967-02-02 1974-12-24 Boots Pure Drug Co Ltd 17-acyloxysteroids and their manufacture
GB1253828A (en) * 1967-10-25 1971-11-17 Shionogi & Co 2,3-EPITHIO-5alpha-ANDROST-6-ENE STEROIDS
US3916002A (en) * 1973-12-17 1975-10-28 Taubert Hans Dieter Oligomeric steroid esters, process for their production, and therapeutic compositions containing the same

Also Published As

Publication number Publication date
FI57263C (fi) 1980-07-10
YU293176A (en) 1982-08-31
HU179343B (en) 1982-10-28
NO145620B (no) 1982-01-18
NO145620C (no) 1982-04-28
FR2335231B1 (it) 1980-03-14
IE44320B1 (en) 1981-10-21
PH13907A (en) 1980-10-27
PT65973B (en) 1978-06-16
DD132270A5 (de) 1978-09-13
US4119626A (en) 1978-10-10
SE428930B (sv) 1983-08-01
IL50981A0 (en) 1977-01-31
DK566076A (da) 1977-06-20
NO147717C (no) 1983-06-01
DK146629C (da) 1984-04-30
BE849553A (fr) 1977-06-17
FR2335231A1 (fr) 1977-07-15
FI763544A (it) 1977-06-20
IT1065783B (it) 1985-03-04
ES454297A1 (es) 1977-12-16
FI57263B (fi) 1980-03-31
CA1086305A (en) 1980-09-23
DK146629B (da) 1983-11-21
NZ182890A (en) 1980-05-08
GB1554199A (en) 1979-10-17
DE2558076C2 (de) 1983-12-15
PL105525B1 (pl) 1979-10-31
JPS5278860A (en) 1977-07-02
CH630097A5 (de) 1982-05-28
SE7614107L (sv) 1977-06-20
SU648105A3 (ru) 1979-02-15
IE44320L (en) 1977-06-19
ZA767510B (en) 1977-11-30
NO764284L (it) 1977-06-21
EG12383A (en) 1979-06-30
NO803670L (no) 1977-06-21
AT357704B (de) 1980-07-25
JPS6131115B2 (it) 1986-07-17
GR62084B (en) 1979-02-21
NL7614023A (nl) 1977-06-21
MX3798E (es) 1981-07-22
AU2073776A (en) 1978-06-29
DE2558076A1 (de) 1977-06-30
AU507111B2 (en) 1980-02-07
PT65973A (en) 1977-01-01
BG30475A3 (en) 1981-06-15
NO147717B (no) 1983-02-21
BG31504A3 (en) 1982-01-15
LU76398A1 (it) 1977-06-10
ATA935576A (de) 1979-12-15
IL50981A (en) 1980-09-16
RO75383A (ro) 1980-11-30

Similar Documents

Publication Publication Date Title
JPS51115409A (en) Method of producing ethyridene diacetate
CS188263B2 (en) Method of producing new biphenyloxyderivatives
BG27550A3 (en) Method of obtaining of thiazolinyl- or thiazinyl- benzimidazole esters
JPS523010A (en) Acetylene glycol and method of producing same
CS189737B2 (en) Method of producing new trichlormethylamidines
PT65402A (en) 3-oximes of d-17alpha-ethynyl-19-nortestosterone esters and method
CS194788B2 (en) Method of producing depot steroid esters
JPS51146407A (en) Method of producing 22aminoonnbutanol
JPS5253807A (en) Method of producing 22aminoo11alcohol
JPS51138618A (en) Method of producing iminodiacetonitlile
JPS52102212A (en) Method of producing halogenoacetal from ester
JPS51139818A (en) Method of producing combined panels
JPS5220194A (en) Method of producing metallic can
JPS51148634A (en) Method of producing hydrogennoccluding metal
CH612117A5 (en) Method of producing sawn-timber elements
JPS5268908A (en) Method of producing motor
JPS5219719A (en) Method of making combined panel
JPS5236616A (en) Method of producing 22chloroalkanal
JPS5212958A (en) Method of producing ice
JPS5270687A (en) Method of producing metallic can
JPS5271311A (en) Method of producing ironnsiliconnaluminium alloy
CS181443B1 (en) Method of producing glycol esters
JPS51139859A (en) Method of producing cases
JPS5251066A (en) Method of producing pidan
JPS5221360A (en) Method of producing eggroll