CS189731B2 - Method of producing new derivatives of 3-aminoindazolcarboxylic acid - Google Patents

Method of producing new derivatives of 3-aminoindazolcarboxylic acid

Info

Publication number
CS189731B2
CS189731B2 CS758165A CS816575A CS189731B2 CS 189731 B2 CS189731 B2 CS 189731B2 CS 758165 A CS758165 A CS 758165A CS 816575 A CS816575 A CS 816575A CS 189731 B2 CS189731 B2 CS 189731B2
Authority
CS
Czechoslovakia
Prior art keywords
aminoindazolcarboxylic
acid
producing new
new derivatives
derivatives
Prior art date
Application number
CS758165A
Other languages
Czech (cs)
English (en)
Inventor
Karl H Mayer
Siegfried Petersen
Erich Klauke
Friedrich Hoffmeister
Wolfgang Wuttke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of CS189731B2 publication Critical patent/CS189731B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CS758165A 1974-12-13 1975-12-02 Method of producing new derivatives of 3-aminoindazolcarboxylic acid CS189731B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
CS189731B2 true CS189731B2 (en) 1979-04-30

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
CS758165A CS189731B2 (en) 1974-12-13 1975-12-02 Method of producing new derivatives of 3-aminoindazolcarboxylic acid

Country Status (27)

Country Link
US (1) US4051252A (en:Method)
JP (1) JPS5182266A (en:Method)
AT (1) AT343653B (en:Method)
BE (1) BE836528A (en:Method)
CA (1) CA1059523A (en:Method)
CH (1) CH622250A5 (en:Method)
CS (1) CS189731B2 (en:Method)
DD (1) DD125484A5 (en:Method)
DE (1) DE2458965C3 (en:Method)
DK (1) DK137082C (en:Method)
ES (1) ES443429A1 (en:Method)
FI (1) FI753493A7 (en:Method)
FR (1) FR2293928A1 (en:Method)
GB (1) GB1490306A (en:Method)
HK (1) HK52580A (en:Method)
HU (1) HU173557B (en:Method)
IE (1) IE42208B1 (en:Method)
IL (1) IL48642A (en:Method)
KE (1) KE3078A (en:Method)
LU (1) LU73993A1 (en:Method)
NL (1) NL7514521A (en:Method)
NO (1) NO145382C (en:Method)
PL (1) PL99858B1 (en:Method)
SE (1) SE419645B (en:Method)
SU (1) SU604487A3 (en:Method)
YU (1) YU315275A (en:Method)
ZA (1) ZA757777B (en:Method)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
CN1926132B (zh) * 2000-09-15 2010-12-29 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的吡唑化合物
EP1698627A1 (en) * 2000-09-15 2006-09-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
MXPA03002291A (es) 2000-09-15 2003-06-06 Vertex Pharma Compuestos de pirazol utiles como inhibidores de proteina cinasa.
ATE340172T1 (de) 2000-12-21 2006-10-15 Vertex Pharma Pyrazolverbindungen als protein- kinasehemmer
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
EP1820503B1 (en) 2001-09-26 2012-02-22 Pfizer Italia S.r.l. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
WO2003066629A2 (en) * 2002-02-06 2003-08-14 Vertex Pharmaceuticals Incorporated Heteroaryl compounds useful as inhibitors of gsk-3
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
AU2003218215A1 (en) 2002-03-15 2003-09-29 Vertex Pharmaceuticals, Inc. Azolylaminoazines as inhibitors of protein kinases
ES2411655T3 (es) 2002-05-17 2013-07-08 Pfizer Italia S.R.L. Derivados de aminoindazol activos como inhibidores de quinasas, procedimiento para su preparación y composiciones farmacéuticas que los comprenden
MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
DE60308387T2 (de) 2002-08-02 2007-09-20 Vertex Pharmaceuticals Inc., Cambridge Pyrazolenthaltende zusammensetzungen und ihre verwendung als gsk-3 inhibitoren
WO2004041285A1 (en) * 2002-10-31 2004-05-21 Amgen Inc. Antiinflammation agents
WO2004072029A2 (en) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
WO2005056547A2 (en) * 2003-12-04 2005-06-23 Vertex Pharmaceuticals Incorporated Quinoxalines useful as inhibitors of protein kinases
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
ATE542814T1 (de) 2005-08-18 2012-02-15 Vertex Pharma Pyrazinkinaseinhibitoren
AR056763A1 (es) * 2005-11-03 2007-10-24 Vertex Pharma Aminopirimidinas sustituidas con tiazol o pirazol,utiles como agentes anticancer y composiciones farmaceuticas que las contienen.
KR101118932B1 (ko) * 2006-04-14 2012-02-27 아보트 러보러터리즈 바닐로이드 서브타입 1(ｖｒ1) 수용체를 억제하는 인다졸릴우레아의 제조방법
WO2008057940A1 (en) 2006-11-02 2008-05-15 Vertex Pharmaceuticals Incorporated Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
MX2009006690A (es) 2006-12-19 2009-07-31 Vertex Pharma Aminopirimidinas utiles como inhibidores de proteinas cinasas.
JP2010520887A (ja) 2007-03-09 2010-06-17 バーテックス ファーマシューティカルズ インコーポレイテッド 蛋白キナーゼの阻害剤として有用なアミノピリジン
MX2009009590A (es) 2007-03-09 2009-11-10 Vertex Pharma Aminopirimidinas utiles como inhibidores de proteinas cinasas.
CA2680029A1 (en) 2007-03-09 2008-09-18 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
EP2146982A2 (en) 2007-04-13 2010-01-27 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
EP2152696B1 (en) 2007-05-02 2014-09-24 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
CA2685876A1 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
JP5572087B2 (ja) * 2007-05-02 2014-08-13 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼ阻害として有用なアミノピリミジン
AU2008257044A1 (en) * 2007-05-24 2008-12-04 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
NZ582879A (en) * 2007-07-31 2012-03-30 Vertex Pharma Process for preparing 5-fluoro-1h-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof
MX2011002312A (es) * 2008-09-03 2011-04-26 Vertex Pharma Co-cristales y formulaciones farmaceuticas que comprenden los mismos.
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
AU2013293650B2 (en) 2012-07-24 2017-05-25 Bial- Portela & Ca, S.A. Urea compounds and their use as enzyme inhibitors
EP2882712A2 (en) * 2012-07-27 2015-06-17 BIAL - Portela & Cª S.A. Process for the synthesis of substituted urea compounds
WO2015012708A1 (en) 2013-07-24 2015-01-29 BIAL - PORTELA & Cª, S.A. Imidazolecarboxamides and their use as faah inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3277100A (en) * 1963-05-31 1966-10-04 Du Pont Novel substituted pyrazoles
NL6707299A (en:Method) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
DE2458965C3 (de) 1979-10-11
NL7514521A (nl) 1976-06-15
DK137082B (da) 1978-01-16
CA1059523A (en) 1979-07-31
NO145382B (no) 1981-11-30
KE3078A (en) 1980-10-03
IE42208B1 (en) 1980-06-18
JPS5182266A (en) 1976-07-19
DE2458965A1 (de) 1976-06-16
DD125484A5 (en:Method) 1977-04-20
IE42208L (en) 1976-06-13
FI753493A7 (en:Method) 1976-06-14
LU73993A1 (en:Method) 1976-11-11
SE7513990L (sv) 1976-06-14
BE836528A (fr) 1976-06-11
PL99858B1 (pl) 1978-08-31
SE419645B (sv) 1981-08-17
IL48642A (en) 1979-12-30
DE2458965B2 (de) 1979-02-22
AU8717075A (en) 1977-06-09
GB1490306A (en) 1977-11-02
AT343653B (de) 1978-06-12
FR2293928B1 (en:Method) 1979-09-21
ATA939775A (de) 1977-10-15
SU604487A3 (ru) 1978-04-25
NO754024L (en:Method) 1976-06-15
DK137082C (da) 1978-06-19
HK52580A (en) 1980-09-26
NO145382C (no) 1982-03-10
FR2293928A1 (fr) 1976-07-09
CH622250A5 (en:Method) 1981-03-31
YU315275A (en) 1982-02-28
ES443429A1 (es) 1977-04-16
ZA757777B (en) 1976-11-24
IL48642A0 (en) 1976-02-29
US4051252A (en) 1977-09-27
DK567275A (da) 1976-06-14
HU173557B (hu) 1979-06-28

Similar Documents

Publication Publication Date Title
CS189731B2 (en) Method of producing new derivatives of 3-aminoindazolcarboxylic acid
JPS53101385A (en) Method of producing phenyllpyrimidine
CS188985B2 (en) Method of producing aryl-1-azolylmethanes
CS190478B2 (en) Method of producing novel biphenylyl derivatives
CS194749B2 (en) Method of producing novel derivatives of 3-sulphonyl-ox!-crotonic acid
CS189709B2 (en) Method of producing 6-d-/-/-alpha-amino-alpha-/p-acetoxyphenylacetamido/penicillanic acid
CS188235B2 (en) Method of producing new derivatives ryfamicine
CS191264B2 (en) Method of producing new pyridobenzodiazepinones
CS188938B2 (en) Method of producing xanthene-9-spiro-4-piperidines
CS183850B2 (en) Method of producing 5-fluor-2-methyl-1-/p-methyl-sulphinylbenzyliden/-3-indenylacetic acid
SU677666A3 (en) Method of producing 7l-or extradiols
YU118575A (en) Process for obtaining new derivatives of 13-thiaprostanoic acid
CS190489B2 (en) Method of producing novel derivatives of prostanoic acid
HU170859B (hu) Sposob poluchenija novykh proizvodnykh 6-skobka-al'fa-ureido-fenilacetilamido-skobka zakryta-penam-3-karbonovojj kisloty
CS189635B2 (en) Method of producing bromderivatives of 4-imido-thioazetidin-2-one
CS192518B2 (en) Method of producing derivatives of 3-cinnolincarboxylic acid
CS182298B2 (en) Method of producing substituted benzendisulphon-amides
CS187333B2 (en) Method of producing derivatives of prostanoic acid
HU171053B (hu) Sposob poluchenija novykh proizvodnykh 7-skobka-2-ureido-acetamido-skobka zakryta-3-geterociklicheskijj-tiometil-cef-3-em-4-karbonovojj kisloty
CS189753B2 (en) Method of producing derivatives of prostanic acid
HU175345B (hu) Sposob poluchenija novykh proizvodnykh 15-gidroksi-16s- i -16r-alkil-prost-5-en-13-in-karbonovykh kislot
CS188945B2 (en) Method of producing 1-aryluracils
CS185675B2 (en) Method of producing 7-amino-delta up3-cephem derivatives
CS181278B2 (en) Method of producing cephalosporane acid derivatives
BG25086A3 (en) A method of obtaining derivatives of thiazolidinon-acetic acid