CO5210949A1 - Trifluorometilalquilaminotriazolopirimidinas fungicidas - Google Patents

Trifluorometilalquilaminotriazolopirimidinas fungicidas

Info

Publication number
CO5210949A1
CO5210949A1 CO99059982A CO99059982A CO5210949A1 CO 5210949 A1 CO5210949 A1 CO 5210949A1 CO 99059982 A CO99059982 A CO 99059982A CO 99059982 A CO99059982 A CO 99059982A CO 5210949 A1 CO5210949 A1 CO 5210949A1
Authority
CO
Colombia
Prior art keywords
formula
jpeg
optically active
atom
emi file
Prior art date
Application number
CO99059982A
Other languages
English (en)
Inventor
Waldemar Pfrengle
Klaus-Juerge Pees
Albert Guido
Paul Carter
Annerose Rehnig
Tuyl Cotter Henry Van
Original Assignee
Basf Agrochemical Products Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Agrochemical Products Bv filed Critical Basf Agrochemical Products Bv
Publication of CO5210949A1 publication Critical patent/CO5210949A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/82—Purification; Separation; Stabilisation; Use of additives
    • C07C209/86—Separation
    • C07C209/88—Separation of optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Una 7-(1,1,1-trifluoroalc-2-ilamino)-triazolopirimidina ópticamente activa de fórmula l<EMI FILE="99059982_1" ID="1" IMF=JPEG >en la cualR1 representa un grupo alquilo C1-6;CH* indica un átomo de carbono quiral;Hal representa un átomo de halógeno,L1 a L5 cada uno representa independientemente un átomo de hidrógeno o halógeno o un grupo alquilo, alcoxi o nitro, caracterizado porque el exceso enantiomérico del (S)-enantiómero es por lo menos 70%.Un proceso para la preparación de un compuesto ópticamente activo de fórmula I como se define en cualquiera de las reivindicaciones precedentes que comprendeTratar un compuesto de fórmula ll<EMI FILE="99059982_2" ID="2" IMF=JPEG >en la cualL1 a L5 y Hal son como se definen en la reivindicación 1 y con una amina ópticamente activa de fórmula III<EMI FILE="99059982_3" ID="3" IMF=JPEG >en la cualR1 y R2 son como se definieron en la reivindicación 1,M representa un átomo de hidrógeno o un átomo de metal libre o complejado, y el exceso enantiomérico del (S)-enantiómero es de por lo menos 70%, a una temperatura de reacción en el rango de 0°C a 70°C, y en presencia de una base.
CO99059982A 1998-09-25 1999-09-22 Trifluorometilalquilaminotriazolopirimidinas fungicidas CO5210949A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US09/160,894 US5986135A (en) 1998-09-25 1998-09-25 Fungicidal trifluoromethylalkylamino-triazolopyrimidines

Publications (1)

Publication Number Publication Date
CO5210949A1 true CO5210949A1 (es) 2002-10-30

Family

ID=22578919

Family Applications (1)

Application Number Title Priority Date Filing Date
CO99059982A CO5210949A1 (es) 1998-09-25 1999-09-22 Trifluorometilalquilaminotriazolopirimidinas fungicidas

Country Status (16)

Country Link
US (2) US5986135A (es)
EP (2) EP1468984A1 (es)
JP (1) JP2000119275A (es)
KR (1) KR100598727B1 (es)
CN (1) CN1218947C (es)
AR (1) AR021827A1 (es)
AT (1) ATE274516T1 (es)
BR (1) BR9904354A (es)
CO (1) CO5210949A1 (es)
DE (1) DE69919647T2 (es)
DK (1) DK0989130T3 (es)
ES (1) ES2227975T3 (es)
PT (1) PT989130E (es)
SI (1) SI0989130T1 (es)
TW (1) TWI225061B (es)
ZA (1) ZA995673B (es)

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KR20040015358A (ko) * 2001-07-18 2004-02-18 바스프 악티엔게젤샤프트 살진균제인 치환된 6-(2-톨릴)-트리아졸로피리미딘
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UA80304C2 (en) 2002-11-07 2007-09-10 Basf Ag Substituted 6-(2-halogenphenyl)triazolopyrimidines
EP1684763B1 (en) * 2003-09-24 2008-06-18 Wyeth Holdings Corporation 6-aryl-7-halo-imidazo[1,2-a]pyrimidines as anticancer agent
US7419982B2 (en) * 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
ATE432077T1 (de) * 2003-09-24 2009-06-15 Wyeth Corp 5-arylpyrimidine als anti-krebs-mittel
ES2279452T3 (es) * 2003-09-24 2007-08-16 Wyeth Holdings Corporation 6-((sustituido)fenil)triazolopirimidinas como agentes antineoplasicos.
DE10347090A1 (de) 2003-10-10 2005-05-04 Bayer Cropscience Ag Synergistische fungizide Wirkstoffkombinationen
DE10349501A1 (de) 2003-10-23 2005-05-25 Bayer Cropscience Ag Synergistische fungizide Wirkstoffkombinationen
MY179926A (en) 2003-12-08 2020-11-19 Wyeth Corp Process for the preparation of tubulin inhibitors
MXPA06005987A (es) * 2003-12-17 2006-08-23 Basf Ag 6-(2-cloro-4-alcoxi-fenil)-triazolopirimidinas, procedimientos para su preparacion y el uso de las mimas para combatir hongos nocivos, asi como productos que las contienen.
WO2005058903A1 (de) * 2003-12-17 2005-06-30 Basf Aktiengesellschaft 6-(2,4,6-trihalogenphenyl)-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
PE20050594A1 (es) * 2003-12-17 2005-10-18 Basf Ag 6-(2-fluoro-4-alcoxifenil)-triazolopirimidinas y procedimientos para su preparacion
AU2005254665A1 (en) * 2004-06-22 2005-12-29 Basf Aktiengesellschaft Use of 6-(2-tolyl)-triazolopyrimidines as fungicides, novel 6-(2-tolyl)-triazolopyrimidines, method for the production thereof, use thereof for controlling harmful fungi, and agents containing the same
US20080032889A1 (en) * 2004-06-22 2008-02-07 Basf Aktiengesellschaft 6-(2-Fluorophenyl)-Triazolopyrimidines, Method For The Production Thereof, Use Thereof For Controlling Harmful Fungi, And Agents Containing The Same
US20080248952A1 (en) * 2004-07-08 2008-10-09 Basf Aktiengesellschaft Substituted 6-Phenyl-7-Aminotriazolopyrimidines, Method for the Production Thereof, Their Use for Controlling Pathogenic Fungi, and Agents Containing These Compounds
BRPI0608712A2 (pt) * 2005-03-18 2010-12-07 Basf Ag processo para a preparação de composto, e, uso do composto
DE102005015677A1 (de) 2005-04-06 2006-10-12 Bayer Cropscience Ag Synergistische fungizide Wirkstoffkombinationen
DE102005026482A1 (de) 2005-06-09 2006-12-14 Bayer Cropscience Ag Wirkstoffkombinationen
MX2007015376A (es) 2005-06-09 2008-02-14 Bayer Cropscience Ag Combinaciones de productos activos.
BRPI0612673A2 (pt) * 2005-06-27 2016-11-29 Basf Ag processo para preparar compostos, compostos, e, uso de compostos
CN101208289A (zh) * 2005-06-27 2008-06-25 巴斯福股份公司 生产取代的苯基丙二酸酯中间体化合物的方法及其在生产5,7-二羟基-6-(2,4,6-三氟苯基)[1,2,4]三唑并[1,5-a]嘧啶中的用途
AR059649A1 (es) * 2006-02-28 2008-04-16 Basf Ag 6- fenil 7-amino - amino (1,2,4) -triazolo (1,5-a) pirimidinas y su su uso para el combate de hongos daninos
DE102006023263A1 (de) 2006-05-18 2007-11-22 Bayer Cropscience Ag Synergistische Wirkstoffkombinationen
JP5142492B2 (ja) * 2006-08-01 2013-02-13 東ソー株式会社 （１−メチル−２，２，２−トリフルオロ）エチルアミン類およびその製造方法
WO2008084082A1 (de) * 2007-01-11 2008-07-17 Basf Se Verfahren zur herstellung arylsubstituierter anellierter pyrimidine
DE102007045920B4 (de) 2007-09-26 2018-07-05 Bayer Intellectual Property Gmbh Synergistische Wirkstoffkombinationen
WO2010108507A2 (de) 2009-03-25 2010-09-30 Bayer Cropscience Ag Synergistische wirkstoffkombinationen
MX2012000566A (es) 2009-07-16 2012-03-06 Bayer Cropscience Ag Combinaciones sinergicas de principios activos con feniltriazoles.
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US9649317B2 (en) 2012-09-19 2017-05-16 The Trustees Of The University Of Pennsylvania Heterocyclic compounds and their use for the treatment of neurodegenerative tauopathies
CN103709072B (zh) * 2012-09-29 2015-06-24 中国科学院化学研究所 一种光活性三氟甲基胺类化合物及其制备方法
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Also Published As

Publication number Publication date
ZA995673B (en) 2000-03-30
EP1468984A1 (en) 2004-10-20
TWI225061B (en) 2004-12-11
JP2000119275A (ja) 2000-04-25
DE69919647D1 (de) 2004-09-30
DE69919647T2 (de) 2005-09-01
CN1250052A (zh) 2000-04-12
US5986135A (en) 1999-11-16
CN1218947C (zh) 2005-09-14
KR20000023437A (ko) 2000-04-25
KR100598727B1 (ko) 2006-07-13
US6204269B1 (en) 2001-03-20
PT989130E (pt) 2004-12-31
DK0989130T3 (da) 2004-11-29
EP0989130A1 (en) 2000-03-29
ATE274516T1 (de) 2004-09-15
BR9904354A (pt) 2000-09-12
SI0989130T1 (en) 2004-12-31
ES2227975T3 (es) 2005-04-01
EP0989130B1 (en) 2004-08-25
AR021827A1 (es) 2002-08-07

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