CN1849328A - 新型14和15元环化合物 - Google Patents

新型14和15元环化合物 Download PDF

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Publication number
CN1849328A
CN1849328A CNA2004800192646A CN200480019264A CN1849328A CN 1849328 A CN1849328 A CN 1849328A CN A2004800192646 A CNA2004800192646 A CN A2004800192646A CN 200480019264 A CN200480019264 A CN 200480019264A CN 1849328 A CN1849328 A CN 1849328A
Authority
CN
China
Prior art keywords
alkyl
group
hydrogen
ethyl
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CNA2004800192646A
Other languages
English (en)
Chinese (zh)
Inventor
S·阿利霍兹克
A·K·福雷斯特
R·L·亚维斯特
G·拉扎雷夫斯基
D·帕夫洛维克
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Fidelta doo
Original Assignee
Glaxo Group Ltd
Pliva Istrazivacki Institut doo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd, Pliva Istrazivacki Institut doo filed Critical Glaxo Group Ltd
Publication of CN1849328A publication Critical patent/CN1849328A/zh
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CNA2004800192646A 2003-05-13 2004-05-11 新型14和15元环化合物 Pending CN1849328A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0310986.5A GB0310986D0 (en) 2003-05-13 2003-05-13 Novel compounds
GB0310986.5 2003-05-13

Publications (1)

Publication Number Publication Date
CN1849328A true CN1849328A (zh) 2006-10-18

Family

ID=9957984

Family Applications (1)

Application Number Title Priority Date Filing Date
CNA2004800192646A Pending CN1849328A (zh) 2003-05-13 2004-05-11 新型14和15元环化合物

Country Status (22)

Country Link
US (1) US7569550B2 (https=)
EP (1) EP1628988B1 (https=)
JP (1) JP2007502313A (https=)
KR (1) KR20060026407A (https=)
CN (1) CN1849328A (https=)
AR (1) AR044309A1 (https=)
AT (1) ATE341560T1 (https=)
AU (1) AU2004238528A1 (https=)
BR (1) BRPI0410246A (https=)
CA (1) CA2525452A1 (https=)
CL (1) CL2004001010A1 (https=)
DE (1) DE602004002696T2 (https=)
DK (1) DK1628988T3 (https=)
ES (1) ES2273255T3 (https=)
GB (1) GB0310986D0 (https=)
HR (1) HRP20060448T3 (https=)
MX (1) MXPA05012163A (https=)
PL (1) PL1628988T3 (https=)
PT (1) PT1628988E (https=)
RU (1) RU2005134908A (https=)
WO (1) WO2004101586A1 (https=)
ZA (1) ZA200509079B (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111574575A (zh) * 2020-04-29 2020-08-25 北京理工大学 一种含有大环内酯基的喹喏酮衍生物、制备方法及应用

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0424961D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
GB0424958D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
WO2007054295A1 (en) * 2005-11-09 2007-05-18 Glaxo Group Limited New 4*-substituted erythromycin derivative
PT1851236E (pt) * 2005-01-13 2010-10-25 Glaxosmithkline Zagreb Macrólidos com actividade anti-inflamatória
JP2008540503A (ja) 2005-05-10 2008-11-20 グラクソスミスクライン・イストラジヴァッキ・センタル・ザグレブ・ドルズバ・ゼー・オメイェノ・オドゴヴォルノスティオ 細菌感染症の処置に有用なエーテル結合マクロライド
EP1945652A1 (en) * 2005-11-09 2008-07-23 Glaxo Group Limited Macrolones
TW201038277A (en) 2009-01-30 2010-11-01 Glaxosmithkline Zagreb Anti-inflammatory macrolide

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1990011288A1 (en) * 1989-03-28 1990-10-04 Abbott Laboratories Erythromycin derivatives
AU3710695A (en) * 1995-04-27 1996-11-18 Laboratorios Aranda, S.A. De C.V. Quinolonylcarboxyerythromycin derivatives and pharmaceutical compositions containing them
JP2002502366A (ja) * 1996-05-07 2002-01-22 アボット・ラボラトリーズ ３―デスクラジノース―２，３―無水エリスロマイシン誘導体
GB0025688D0 (en) * 2000-10-19 2000-12-06 Glaxo Group Ltd Macrolides
JP4311203B2 (ja) * 2001-08-08 2009-08-12 大正製薬株式会社 １１ａ−アザライド化合物及びその製造方法
GB0127349D0 (en) 2001-11-14 2002-01-02 Glaxo Group Ltd Macrolides

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111574575A (zh) * 2020-04-29 2020-08-25 北京理工大学 一种含有大环内酯基的喹喏酮衍生物、制备方法及应用
CN111574575B (zh) * 2020-04-29 2022-05-17 北京理工大学 一种含有大环内酯基的喹喏酮衍生物、制备方法及应用

Also Published As

Publication number Publication date
CL2004001010A1 (es) 2005-03-18
WO2004101586A1 (en) 2004-11-25
AR044309A1 (es) 2005-09-07
EP1628988B1 (en) 2006-10-04
AU2004238528A1 (en) 2004-11-25
US7569550B2 (en) 2009-08-04
DE602004002696D1 (de) 2006-11-16
MXPA05012163A (es) 2006-05-19
DE602004002696T2 (de) 2007-08-16
ATE341560T1 (de) 2006-10-15
CA2525452A1 (en) 2004-11-25
DK1628988T3 (da) 2007-02-05
ZA200509079B (en) 2007-02-28
GB0310986D0 (en) 2003-06-18
JP2007502313A (ja) 2007-02-08
HRP20060448T3 (hr) 2007-03-31
PL1628988T3 (pl) 2007-03-30
KR20060026407A (ko) 2006-03-23
US20070185117A1 (en) 2007-08-09
BRPI0410246A (pt) 2006-05-16
PT1628988E (pt) 2007-01-31
ES2273255T3 (es) 2007-05-01
RU2005134908A (ru) 2006-06-27
EP1628988A1 (en) 2006-03-01

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Legal Events

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C06 Publication
PB01 Publication
C10 Entry into substantive examination
SE01 Entry into force of request for substantive examination
C02 Deemed withdrawal of patent application after publication (patent law 2001)
WD01 Invention patent application deemed withdrawn after publication

Open date: 20061018