CN1571670A - 弗利班西林在治疗性障碍中的用途 - Google Patents

弗利班西林在治疗性障碍中的用途 Download PDF

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Publication number
CN1571670A
CN1571670A CNA028208285A CN02820828A CN1571670A CN 1571670 A CN1571670 A CN 1571670A CN A028208285 A CNA028208285 A CN A028208285A CN 02820828 A CN02820828 A CN 02820828A CN 1571670 A CN1571670 A CN 1571670A
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CN
China
Prior art keywords
acid
sexual
sexual demand
demand
purposes
Prior art date
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Pending
Application number
CNA028208285A
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English (en)
Chinese (zh)
Inventor
肯尼思·R·埃文斯
佛朗哥·博西尼
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Original Assignee
Boehringer Ingelheim Pharma GmbH and Co KG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by Boehringer Ingelheim Pharma GmbH and Co KG filed Critical Boehringer Ingelheim Pharma GmbH and Co KG
Publication of CN1571670A publication Critical patent/CN1571670A/zh
Pending legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Endocrinology (AREA)
  • Psychiatry (AREA)
  • Reproductive Health (AREA)
  • Pain & Pain Management (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CNA028208285A 2001-10-20 2002-10-04 弗利班西林在治疗性障碍中的用途 Pending CN1571670A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01125020 2001-10-20
EP01125020.6 2001-10-20

Related Child Applications (3)

Application Number Title Priority Date Filing Date
CN201110009433XA Division CN102058597A (zh) 2001-10-20 2002-10-04 弗利班西林在治疗性障碍中的用途
CNA2008101316858A Division CN101347431A (zh) 2001-10-20 2002-10-04 弗利班西林在治疗性障碍中的用途
CN2011100094486A Division CN102125557A (zh) 2001-10-20 2002-10-04 弗利班西林在治疗性障碍中的用途

Publications (1)

Publication Number Publication Date
CN1571670A true CN1571670A (zh) 2005-01-26

Family

ID=8179028

Family Applications (4)

Application Number Title Priority Date Filing Date
CNA028208285A Pending CN1571670A (zh) 2001-10-20 2002-10-04 弗利班西林在治疗性障碍中的用途
CN201110009433XA Pending CN102058597A (zh) 2001-10-20 2002-10-04 弗利班西林在治疗性障碍中的用途
CNA2008101316858A Pending CN101347431A (zh) 2001-10-20 2002-10-04 弗利班西林在治疗性障碍中的用途
CN2011100094486A Pending CN102125557A (zh) 2001-10-20 2002-10-04 弗利班西林在治疗性障碍中的用途

Family Applications After (3)

Application Number Title Priority Date Filing Date
CN201110009433XA Pending CN102058597A (zh) 2001-10-20 2002-10-04 弗利班西林在治疗性障碍中的用途
CNA2008101316858A Pending CN101347431A (zh) 2001-10-20 2002-10-04 弗利班西林在治疗性障碍中的用途
CN2011100094486A Pending CN102125557A (zh) 2001-10-20 2002-10-04 弗利班西林在治疗性障碍中的用途

Country Status (31)

Country Link
US (9) US7151103B2 (OSRAM)
EP (2) EP1446122B1 (OSRAM)
JP (3) JP2005506370A (OSRAM)
KR (3) KR20090130196A (OSRAM)
CN (4) CN1571670A (OSRAM)
AR (2) AR037109A1 (OSRAM)
AT (1) ATE327757T1 (OSRAM)
AU (1) AU2002333894B2 (OSRAM)
BR (1) BR0213358A (OSRAM)
CA (1) CA2458067C (OSRAM)
CY (1) CY1105082T1 (OSRAM)
DE (1) DE60211937T2 (OSRAM)
DK (1) DK1446122T5 (OSRAM)
EA (1) EA007274B1 (OSRAM)
EC (1) ECSP045069A (OSRAM)
ES (1) ES2266632T3 (OSRAM)
HR (1) HRP20040352B1 (OSRAM)
HU (1) HUP0401023A3 (OSRAM)
IL (2) IL160389A0 (OSRAM)
ME (1) MEP42808A (OSRAM)
MX (1) MXPA04003666A (OSRAM)
MY (1) MY127290A (OSRAM)
NO (1) NO325556B1 (OSRAM)
NZ (1) NZ532079A (OSRAM)
PL (1) PL208744B1 (OSRAM)
PT (1) PT1446122E (OSRAM)
RS (1) RS50876B (OSRAM)
SI (1) SI1446122T1 (OSRAM)
UA (1) UA78974C2 (OSRAM)
WO (1) WO2003035072A1 (OSRAM)
ZA (1) ZA200401366B (OSRAM)

Cited By (11)

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US7923449B2 (en) 2005-10-29 2011-04-12 Boehringer Ingelheim International Gmbh Benzimidazolone derivatives for the treatment of premenstrual and other female sexual disorders
US8227476B2 (en) 2005-08-03 2012-07-24 Sprout Pharmaceuticals, Inc. Use of flibanserin in the treatment of obesity
US8227471B2 (en) 2001-10-20 2012-07-24 Sprout Pharmaceuticals, Inc. Treating sexual desire disorders with flibanserin
US8512748B2 (en) 2006-08-25 2013-08-20 Boehringer Ingelheim International Gmbh Controlled release system and method for manufacturing the same
CN103251598A (zh) * 2005-11-08 2013-08-21 贝林格尔.英格海姆国际有限公司 氟班色林在治疗绝经前性欲障碍中的用途
US8545886B2 (en) 2006-08-14 2013-10-01 Boehringer Ingelheim International Gmbh Extended release tablet formulations of flibanserin and method for manufacturing the same
US8658207B2 (en) 2006-08-14 2014-02-25 Boehringer Ingelheim International Gmbh Extended release tablet formulations of flibanserin and method for manufacturing the same
CN104926734A (zh) * 2015-07-07 2015-09-23 苏州立新制药有限公司 氟班色林的制备方法
US9763936B2 (en) 2006-06-30 2017-09-19 Sprout Pharmaceuticals, Inc. Flibanserin for the treatment of urinary incontinence and related diseases
US10166230B2 (en) 2007-09-12 2019-01-01 Sprout Pharmaceuticals Inc. Treatment of vasomotor symptoms
US10675280B2 (en) 2001-10-20 2020-06-09 Sprout Pharmaceuticals, Inc. Treating sexual desire disorders with flibanserin

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US20040048877A1 (en) * 2002-05-22 2004-03-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmaceutical compositions containing flibanserin
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US20050239798A1 (en) * 2004-04-22 2005-10-27 Boehringer Ingelheim Pharmaceuticals, Inc. Method for the treatment of premenstrual and other female sexual disorders
KR101292492B1 (ko) 2004-05-11 2013-08-01 이모셔널 브레인 비.브이. 약제학적 제형물 및 여성 성기능 부전의 치료에서 그것의용도
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US20060211685A1 (en) * 2005-03-04 2006-09-21 Boehringer Ingelheim International Gmbh Pharmaceutical compositions for the treatment and/or prevention of depression
WO2006119884A2 (en) * 2005-05-06 2006-11-16 Boehringer Ingelheim International Gmbh Method for the treatment of drug abuse with flibanserin
CA2608363A1 (en) * 2005-05-19 2006-11-23 Boehringer Ingelheim International Gmbh Method for the treatment of drug-induced sexual dysfunction
WO2006125041A1 (en) * 2005-05-19 2006-11-23 Boehringer Ingelheim International Gmbh Method for the treatment of sexual dysfunctions due to medical conditions
CA2614833A1 (en) * 2005-07-12 2007-01-18 Boehringer Ingelheim International Gmbh Pharmaceutical composition comprising 2, 3-disubstituted tropanes for the treatment of disorders of sexual desire
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EP1790343A1 (en) 2005-11-11 2007-05-30 Emotional Brain B.V. Pharmaceuticals formulations and uses thereof in the treatment of female sexual dysfunction
EP2010505B1 (en) * 2006-03-28 2012-12-05 Atir Holding S.A. Heterocyclic compounds and uses thereof in the treatment of sexual disorders
EA200802208A1 (ru) * 2006-05-09 2009-04-28 Бёрингер Ингельхайм Интернациональ Гмбх Применение флибансерина для лечения расстройств полового влечения в постклимактерический период
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CA2657045A1 (en) * 2006-07-14 2008-01-17 Boehringer Ingelheim International Gmbh Combinations of flibanserin with caffeine, process for their preparation and use thereof as medicaments
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US8722682B2 (en) 2006-12-20 2014-05-13 Sprout Pharmaceuticals, Inc. Sulfated benzimidazolone derivatives having mixed serotonin receptor affinity
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CA2686480A1 (en) 2008-12-15 2010-06-15 Boehringer Ingelheim International Gmbh New salts
DE102011012712A1 (de) 2011-03-01 2012-09-06 Frank Lehmann-Horn Verwendung von Aldosteron-Rezeptor-Antagonisten zur Behandlung von weiblicher sexueller Dysfunktion
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