HUP0401023A2 - Flibanserin alkalmazása szexuális zavarok kezelésére - Google Patents

Flibanserin alkalmazása szexuális zavarok kezelésére

Info

Publication number
HUP0401023A2
HUP0401023A2 HU0401023A HUP0401023A HUP0401023A2 HU P0401023 A2 HUP0401023 A2 HU P0401023A2 HU 0401023 A HU0401023 A HU 0401023A HU P0401023 A HUP0401023 A HU P0401023A HU P0401023 A2 HUP0401023 A2 HU P0401023A2
Authority
HU
Hungary
Prior art keywords
acid
flibanserin
sexual desire
disorders
treatment
Prior art date
Application number
HU0401023A
Other languages
English (en)
Inventor
Franco Borsini
Kenneth Robert Evans
Original Assignee
Boehringer Ingelheim Pharma Gmbh & Co. Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma Gmbh & Co. Kg filed Critical Boehringer Ingelheim Pharma Gmbh & Co. Kg
Publication of HUP0401023A2 publication Critical patent/HUP0401023A2/hu
Publication of HUP0401023A3 publication Critical patent/HUP0401023A3/hu

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pain & Pain Management (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

A találmány tárgya flibanserin (1-[2-{4-[3-(trifluormetil)-fenil]-1-piperazinil}-etil]-2,3-dihidro-1(1-benzimidazol-2-on) alkalmazása,adott esetben gyógyszerészetileg elfogadható savaddíciós sóiformájában, a csökkent aktivitású szexuális vágy rendellenesség, aszexuális vágy elvesztése, a szexuális vágy hiánya, a csökkent vagygátolt szexuális vágy körébe tartozó rendellenességek kezeléséreszolgáló gyógyszer előállítására. A flibanserin gyógyszerészetilegelfogadható savaddíciós sóit borostánykősav, hidrogén-bromid, ecetsav,fumársav, maleinsav, metánszulfonsav, tejsav, foszforsav, sósav,kénsav, borkősav, citromsav és elegyeik valamelyikével képezik. Aflibanserint 0,1 és 400 mg/nap közötti tartományba eső adagokbanalkalmazzák. Ó
HU0401023A 2001-10-20 2002-10-04 Use of flibanserin in the treatment of sexual disorders HUP0401023A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01125020 2001-10-20
PCT/EP2002/011103 WO2003035072A1 (en) 2001-10-20 2002-10-04 Use of flibanserin in the treatment of sexual disorders

Publications (2)

Publication Number Publication Date
HUP0401023A2 true HUP0401023A2 (hu) 2004-08-30
HUP0401023A3 HUP0401023A3 (en) 2004-10-28

Family

ID=8179028

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0401023A HUP0401023A3 (en) 2001-10-20 2002-10-04 Use of flibanserin in the treatment of sexual disorders

Country Status (31)

Country Link
US (9) US7151103B2 (hu)
EP (2) EP1446122B1 (hu)
JP (3) JP2005506370A (hu)
KR (3) KR20040047931A (hu)
CN (4) CN101347431A (hu)
AR (2) AR037109A1 (hu)
AT (1) ATE327757T1 (hu)
AU (1) AU2002333894B2 (hu)
BR (1) BR0213358A (hu)
CA (1) CA2458067C (hu)
CY (1) CY1105082T1 (hu)
DE (1) DE60211937T2 (hu)
DK (1) DK1446122T5 (hu)
EA (1) EA007274B1 (hu)
EC (1) ECSP045069A (hu)
ES (1) ES2266632T3 (hu)
HR (1) HRP20040352B1 (hu)
HU (1) HUP0401023A3 (hu)
IL (2) IL160389A0 (hu)
ME (1) MEP42808A (hu)
MX (1) MXPA04003666A (hu)
MY (1) MY127290A (hu)
NO (1) NO325556B1 (hu)
NZ (1) NZ532079A (hu)
PL (1) PL208744B1 (hu)
PT (1) PT1446122E (hu)
RS (1) RS50876B (hu)
SI (1) SI1446122T1 (hu)
UA (1) UA78974C2 (hu)
WO (1) WO2003035072A1 (hu)
ZA (1) ZA200401366B (hu)

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