CN1518550A - 用于预防和治疗疱疹病毒感染的咪唑并[1,2-a]吡啶衍生物 - Google Patents

用于预防和治疗疱疹病毒感染的咪唑并[1,2-a]吡啶衍生物 Download PDF

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Publication number
CN1518550A
CN1518550A CNA028124499A CN02812449A CN1518550A CN 1518550 A CN1518550 A CN 1518550A CN A028124499 A CNA028124499 A CN A028124499A CN 02812449 A CN02812449 A CN 02812449A CN 1518550 A CN1518550 A CN 1518550A
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China
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imidazo
pyridin
het
cyclopentylamino
pyrimidinyl
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Pending
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CNA028124499A
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English (en)
Chinese (zh)
Inventor
K���ŵ���ɭ
K·古德蒙森
����� Լ�������
B·A·约翰斯
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SmithKline Beecham Corp
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SmithKline Beecham Corp
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Publication of CN1518550A publication Critical patent/CN1518550A/zh
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CNA028124499A 2001-06-21 2002-06-10 用于预防和治疗疱疹病毒感染的咪唑并[1,2-a]吡啶衍生物 Pending CN1518550A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30000901P 2001-06-21 2001-06-21
US60/300,009 2001-06-21

Publications (1)

Publication Number Publication Date
CN1518550A true CN1518550A (zh) 2004-08-04

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CNA028124499A Pending CN1518550A (zh) 2001-06-21 2002-06-10 用于预防和治疗疱疹病毒感染的咪唑并[1,2-a]吡啶衍生物

Country Status (19)

Country Link
US (3) US7186714B2 (https=)
EP (1) EP1401836B1 (https=)
JP (1) JP2005500315A (https=)
KR (1) KR20040018281A (https=)
CN (1) CN1518550A (https=)
AT (1) ATE337316T1 (https=)
BR (1) BR0210464A (https=)
CA (1) CA2451008A1 (https=)
CO (1) CO5540312A2 (https=)
CZ (1) CZ20033518A3 (https=)
DE (1) DE60214179T2 (https=)
ES (1) ES2271273T3 (https=)
HU (1) HUP0400266A2 (https=)
IL (1) IL158667A0 (https=)
MX (1) MXPA03011906A (https=)
NO (1) NO20035583D0 (https=)
PL (1) PL366827A1 (https=)
WO (1) WO2003000689A1 (https=)
ZA (1) ZA200308726B (https=)

Cited By (5)

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US8207189B2 (en) 2006-11-30 2012-06-26 Nihon Medi-Physics Co., Ltd. Compound having affinity for amyloid
US8303935B2 (en) 2006-05-19 2012-11-06 Nihon Medi-Physics Co., Ltd. Alkoxy substituted imidazo[1,2-a]pyridines having affinity for amyloid
US8658132B2 (en) 2007-02-13 2014-02-25 Nihon Medi-Physics Co., Ltd. Method for production of radiation diagnostic imaging agent
CN110483504A (zh) * 2019-08-02 2019-11-22 桂林理工大学 以DMF为甲酰化试剂构建2-（2-萘基）咪唑[1,2-a]吡啶-3-醛的新方法
CN110483506A (zh) * 2019-08-02 2019-11-22 桂林理工大学 以DMF为甲酰化试剂构建2-（2-噻吩基）咪唑[1,2-a]吡啶-3-醛的新方法

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JP6642942B2 (ja) 2013-12-30 2020-02-12 アレイ バイオファーマ、インコーポレイテッド セリン／トレオニンキナーゼ阻害剤
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Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8303935B2 (en) 2006-05-19 2012-11-06 Nihon Medi-Physics Co., Ltd. Alkoxy substituted imidazo[1,2-a]pyridines having affinity for amyloid
US8207189B2 (en) 2006-11-30 2012-06-26 Nihon Medi-Physics Co., Ltd. Compound having affinity for amyloid
US8658132B2 (en) 2007-02-13 2014-02-25 Nihon Medi-Physics Co., Ltd. Method for production of radiation diagnostic imaging agent
CN110483504A (zh) * 2019-08-02 2019-11-22 桂林理工大学 以DMF为甲酰化试剂构建2-（2-萘基）咪唑[1,2-a]吡啶-3-醛的新方法
CN110483506A (zh) * 2019-08-02 2019-11-22 桂林理工大学 以DMF为甲酰化试剂构建2-（2-噻吩基）咪唑[1,2-a]吡啶-3-醛的新方法
CN110483506B (zh) * 2019-08-02 2022-04-19 桂林理工大学 以DMF为甲酰化试剂构建2-(2-噻吩基)咪唑[1,2-a]吡啶-3-醛的新方法

Also Published As

Publication number Publication date
HUP0400266A2 (hu) 2004-08-30
NO20035583D0 (no) 2003-12-15
EP1401836B1 (en) 2006-08-23
CA2451008A1 (en) 2003-01-03
CO5540312A2 (es) 2005-07-29
WO2003000689A1 (en) 2003-01-03
MXPA03011906A (es) 2004-03-26
PL366827A1 (en) 2005-02-07
ZA200308726B (en) 2005-02-10
ES2271273T3 (es) 2007-04-16
BR0210464A (pt) 2004-07-20
ATE337316T1 (de) 2006-09-15
US7186714B2 (en) 2007-03-06
DE60214179T2 (de) 2007-01-04
US20070135451A1 (en) 2007-06-14
EP1401836A1 (en) 2004-03-31
DE60214179D1 (de) 2006-10-05
US20060167252A1 (en) 2006-07-27
CZ20033518A3 (en) 2004-05-12
US20050228004A1 (en) 2005-10-13
JP2005500315A (ja) 2005-01-06
KR20040018281A (ko) 2004-03-02
IL158667A0 (en) 2004-05-12

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