CN1250549C - 吲哚衍生物及其作为5－ht2b和5－ht2c受体配体的应用 - Google Patents
吲哚衍生物及其作为5－ht2b和5－ht2c受体配体的应用 Download PDFInfo
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- CN1250549C CN1250549C CNB018213510A CN01821351A CN1250549C CN 1250549 C CN1250549 C CN 1250549C CN B018213510 A CNB018213510 A CN B018213510A CN 01821351 A CN01821351 A CN 01821351A CN 1250549 C CN1250549 C CN 1250549C
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Classifications
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Addiction (AREA)
- Child & Adolescent Psychology (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
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- Psychology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0031724.8 | 2000-12-27 | ||
| GB0031724A GB0031724D0 (en) | 2000-12-27 | 2000-12-27 | Indole derivatives |
| GB0119820A GB0119820D0 (en) | 2001-08-14 | 2001-08-14 | Indole derivatives |
| GB0119820.9 | 2001-08-14 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN1483034A CN1483034A (zh) | 2004-03-17 |
| CN1250549C true CN1250549C (zh) | 2006-04-12 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNB018213510A Expired - Fee Related CN1250549C (zh) | 2000-12-27 | 2001-12-14 | 吲哚衍生物及其作为5－ht2b和5－ht2c受体配体的应用 |
Country Status (16)
Families Citing this family (61)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE60330864D1 (de) | 2002-06-19 | 2010-02-25 | Biovitrum Ab Publ | Neue verbindungen, deren verwendung und herstellung |
| US7105526B2 (en) | 2002-06-28 | 2006-09-12 | Banyu Pharmaceuticals Co., Ltd. | Benzimidazole derivatives |
| US7772188B2 (en) | 2003-01-28 | 2010-08-10 | Ironwood Pharmaceuticals, Inc. | Methods and compositions for the treatment of gastrointestinal disorders |
| CL2004000826A1 (es) | 2003-04-25 | 2005-03-04 | Pfizer | Uso de un agonista para el receptor 5-ht2c para preparar un medicamento util en el tratamiento de la incontinencia urinaria provocada por estres, con la condicion de que el agonista no sea 1-[6-cloro-5-(trifluorometil)-2-piridinil]piperazina (org-129 |
| GB0314967D0 (en) * | 2003-06-26 | 2003-07-30 | Hoffmann La Roche | Piperazine derivatives |
| CN1902177A (zh) | 2003-09-22 | 2007-01-24 | 万有制药株式会社 | 新哌啶衍生物 |
| WO2005097127A2 (en) | 2004-04-02 | 2005-10-20 | Merck & Co., Inc. | Method of treating men with metabolic and anthropometric disorders |
| US8685924B2 (en) | 2004-08-25 | 2014-04-01 | Takeda Pharmaceutical Company Limited | Preventives/remedies for stress urinary incontinence and method of screening the same |
| KR101123549B1 (ko) | 2004-11-01 | 2012-04-18 | 아밀린 파마슈티칼스, 인크. | 비만 및 관련 장애의 치료 |
| BRPI0517955A (pt) * | 2004-11-01 | 2008-10-21 | Wyeth Corp | indolizinas substituìdas e derivados como agentes de snc |
| US8394765B2 (en) | 2004-11-01 | 2013-03-12 | Amylin Pharmaceuticals Llc | Methods of treating obesity with two different anti-obesity agents |
| US20090286723A1 (en) | 2005-02-11 | 2009-11-19 | Amylin Pharmaceuticals, Inc. | Hybrid Polypeptides with Selectable Properties |
| US7737155B2 (en) | 2005-05-17 | 2010-06-15 | Schering Corporation | Nitrogen-containing heterocyclic compounds and methods of use thereof |
| AU2006253312B2 (en) | 2005-05-30 | 2011-08-18 | Msd K.K. | Novel piperidine derivative |
| AU2006277253A1 (en) | 2005-08-10 | 2007-02-15 | Msd K.K. | Pyridone compound |
| EP2330125A3 (en) | 2005-08-11 | 2012-12-12 | Amylin Pharmaceuticals, Inc. | Hybrid polypeptides with selectable properties |
| AU2006282260A1 (en) | 2005-08-24 | 2007-03-01 | Msd K.K. | Phenylpyridone derivative |
| EP1939194A4 (en) | 2005-09-07 | 2010-12-08 | Banyu Pharma Co Ltd | AROMATIC SUBSTITUTED BICYLIC PYRIDONE DERIVATIVE |
| RU2008116844A (ru) | 2005-09-29 | 2009-11-10 | Мерк энд Ко., Инк. (US) | Ацилированные производные спиропиперидина как модуляторы рецептора меланокортина-4 |
| KR20080059233A (ko) | 2005-10-21 | 2008-06-26 | 노파르티스 아게 | 레닌 억제제, 및 항이상지질혈증제 및/또는 항비만제의조합물 |
| AU2006307046A1 (en) | 2005-10-27 | 2007-05-03 | Msd K.K. | Novel benzoxathiin derivative |
| AU2006312557B2 (en) | 2005-11-10 | 2011-12-08 | Msd K.K. | Aza-substituted spiro derivative |
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| TW270114B (enrdf_load_stackoverflow) | 1993-10-22 | 1996-02-11 | Hoffmann La Roche | |
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- 2001-12-14 ES ES01989597T patent/ES2291374T3/es not_active Expired - Lifetime
- 2001-12-14 US US10/017,978 patent/US6610685B2/en not_active Expired - Fee Related
- 2001-12-14 WO PCT/EP2001/014781 patent/WO2002051844A1/en active IP Right Grant
- 2001-12-14 DE DE60129841T patent/DE60129841T2/de not_active Expired - Lifetime
- 2001-12-14 KR KR10-2003-7008679A patent/KR100539143B1/ko not_active Expired - Fee Related
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| MXPA03005915A (es) | 2003-09-10 |
| CA2432085A1 (en) | 2002-07-04 |
| AR035722A1 (es) | 2004-07-07 |
| ES2291374T3 (es) | 2008-03-01 |
| KR20030063476A (ko) | 2003-07-28 |
| DE60129841D1 (de) | 2007-09-20 |
| EP1347979B1 (en) | 2007-08-08 |
| AU2002228007B2 (en) | 2007-06-21 |
| UY27097A1 (es) | 2002-07-31 |
| CA2432085C (en) | 2009-02-24 |
| DE60129841T2 (de) | 2008-04-17 |
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| EP1347979A1 (en) | 2003-10-01 |
| PE20020911A1 (es) | 2002-10-22 |
| JP4094950B2 (ja) | 2008-06-04 |
| WO2002051844A1 (en) | 2002-07-04 |
| CN1483034A (zh) | 2004-03-17 |
| BR0116605A (pt) | 2003-09-30 |
| JP2004517852A (ja) | 2004-06-17 |
| AU2002228007B8 (en) | 2002-07-08 |
| KR100539143B1 (ko) | 2005-12-26 |
| ATE369368T1 (de) | 2007-08-15 |
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